BARALDI, Pier Giovanni
 Distribuzione geografica
Continente #
NA - Nord America 42.427
AS - Asia 21.789
EU - Europa 20.194
SA - Sud America 3.359
AF - Africa 512
OC - Oceania 43
Continente sconosciuto - Info sul continente non disponibili 33
Totale 88.357
Nazione #
US - Stati Uniti d'America 41.658
FI - Finlandia 8.286
SG - Singapore 7.626
CN - Cina 5.863
DE - Germania 3.424
BR - Brasile 2.595
UA - Ucraina 2.333
VN - Vietnam 2.165
HK - Hong Kong 1.902
TR - Turchia 1.834
GB - Regno Unito 1.364
IT - Italia 1.208
RU - Federazione Russa 908
SE - Svezia 872
FR - Francia 795
IN - India 462
JP - Giappone 462
MX - Messico 344
CA - Canada 314
BD - Bangladesh 311
AR - Argentina 273
PL - Polonia 259
ZA - Sudafrica 207
IQ - Iraq 179
NL - Olanda 148
ID - Indonesia 131
ES - Italia 113
PK - Pakistan 111
CO - Colombia 110
BE - Belgio 103
EC - Ecuador 94
MA - Marocco 89
TW - Taiwan 87
SA - Arabia Saudita 80
VE - Venezuela 76
CL - Cile 67
UZ - Uzbekistan 66
MY - Malesia 61
KR - Corea 57
LT - Lituania 57
PH - Filippine 53
PY - Paraguay 52
AE - Emirati Arabi Uniti 49
CZ - Repubblica Ceca 47
EG - Egitto 47
AT - Austria 37
IL - Israele 36
TN - Tunisia 36
KE - Kenya 33
AU - Australia 32
IR - Iran 30
PE - Perù 29
BO - Bolivia 28
JO - Giordania 27
UY - Uruguay 27
NP - Nepal 26
EU - Europa 24
IE - Irlanda 24
CR - Costa Rica 21
AZ - Azerbaigian 20
GR - Grecia 20
TH - Thailandia 20
CH - Svizzera 19
DZ - Algeria 18
ET - Etiopia 18
RO - Romania 18
KZ - Kazakistan 17
PS - Palestinian Territory 17
AL - Albania 16
JM - Giamaica 15
HU - Ungheria 14
BH - Bahrain 13
KG - Kirghizistan 13
LB - Libano 13
OM - Oman 13
BG - Bulgaria 12
MD - Moldavia 12
PA - Panama 12
PT - Portogallo 12
SK - Slovacchia (Repubblica Slovacca) 12
SY - Repubblica araba siriana 11
TT - Trinidad e Tobago 11
HR - Croazia 10
LV - Lettonia 10
NO - Norvegia 10
NZ - Nuova Zelanda 10
AO - Angola 9
BY - Bielorussia 9
DO - Repubblica Dominicana 9
RS - Serbia 9
SN - Senegal 9
HN - Honduras 8
MN - Mongolia 8
NI - Nicaragua 8
CI - Costa d'Avorio 7
SV - El Salvador 7
GT - Guatemala 6
MT - Malta 6
MU - Mauritius 6
XK - ???statistics.table.value.countryCode.XK??? 6
Totale 88.245
Città #
Helsinki 7.702
Singapore 4.981
Ashburn 4.042
Woodbridge 3.789
Fairfield 3.580
Dallas 2.772
Houston 2.484
Jacksonville 2.450
San Jose 2.431
Chandler 2.073
Ann Arbor 1.911
Hong Kong 1.779
Santa Clara 1.627
Beijing 1.546
Seattle 1.529
Wilmington 1.378
Cambridge 1.093
Izmir 805
Nanjing 776
Ho Chi Minh City 694
Los Angeles 532
Princeton 513
Hanoi 494
New York 468
Tokyo 422
Boardman 405
Lauterbourg 396
Munich 367
San Diego 323
Ferrara 271
Shenyang 263
São Paulo 249
Milan 236
Shanghai 226
Hefei 220
Nanchang 213
Warsaw 209
Mexico City 199
Tianjin 182
London 178
Orem 158
Hebei 157
Falkenstein 154
San Mateo 153
Changsha 149
Bremen 144
Chicago 143
Addison 141
Jiaxing 121
Brooklyn 118
Council Bluffs 118
Frankfurt am Main 115
Dearborn 114
Dong Ket 114
Turku 112
Jinan 111
The Dalles 109
Montreal 106
Chennai 99
Brussels 98
Da Nang 95
Philadelphia 95
Buffalo 92
Johannesburg 90
Amsterdam 88
Baghdad 88
Haiphong 88
Atlanta 87
Falls Church 86
Moscow 86
Norwalk 84
Rio de Janeiro 84
Kunming 79
San Francisco 79
Redwood City 78
Zhengzhou 76
Denver 75
Guangzhou 72
Phoenix 68
Toronto 68
Stockholm 66
Boston 61
Taipei 60
Mountain View 59
Poplar 58
Tashkent 58
Manchester 57
Belo Horizonte 54
Brasília 54
Mumbai 53
Ningbo 51
Jakarta 48
Auburn Hills 47
Orange 47
Hải Dương 46
Des Moines 44
Verona 44
Dhaka 43
Ankara 42
Quito 41
Totale 61.033
Nome #
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists 3.095
1,4-Diketones via Isoxazole Intermediates 3.074
1,2,3-triazolo[5,4-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new class of A(2A) adenosine receptor antagonists 3.044
Nuovo impiego di poliammidi eterocicliche e benzoeterocicliche strutturalmente correlate all'antibiotico naturale Distamicina A 1.964
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1 528
The use of phase-transfer catalysis for the N-alkylation of indole. 514
Medicinal Chemistry, Pharmacology, and Clinical Implications of TRPV1 Receptor Antagonists 329
A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy 313
A glance at adenosine receptors: Novel target for antitumor therapy 308
Synthesis and Structure Activity Relationship Investigation of Triazolo[1,5-a]pyrimidines as CB2 Cannabinoid Receptor Inverse Agonists 297
A new, efficient synthesis of muscimol (5-ammoniomethylisoxazol-3-olate). 294
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents 294
1-methyl-3-nitro-5-methoxycarbonyl pyrazole 292
A facile, efficient synthesis of 2-substituted-4-hydroxy-2-cyclopenten-1-ones 290
A3 adenosine receptor antagonists: History and future perspectives 286
The A3 adenosine receptor: history and perspectives 281
A [3+2] nitrile oxide intermolecular cycloaddition approach to 4,5-dihydro-3(2H)-furanone and 3(2H)-furanone ring systems: application to the formal synthesis of (±)-ascofuranone and geiparvarin. 278
Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor 276
Positive allosteric modulation of A1 adenosine receptors as a novel and promising therapeutic strategy for anxiety 276
A formal total synthesis (±)-forskolin through [3+2] nitrile oxide cycloaddition chemistry 270
3,5-Disubstituted isoxazoles as a latent aldol moiety: Application to the synthesis of (±)-[6]-gingerol 268
Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole 268
Azaprostaglandin Analogues. Synthesis and Biological Properties of 11-Azaprostaglandin Derivatives 267
A synthetic approach for the preparation of rigid analogs of 1,3-dipropyl-7-methyl-8-aryl/heteroarylstyryl xanthines 264
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization 263
A convenient synthesis of unsymmetrically substituted terphenyls of biologically active stilbenes via a double Suzuki cross-coupling protocol 263
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation 262
Allosteric modulators for the A1-adenosine receptor 256
2,3a,5,6,7,7a-Hexahydro-3H,4H-benzothiophene-3,4-dione and cyclopenta[b]tetrahydrothiophene-3,4-dione enolate anions as synthetic equivalents to cyclohex-2-enone and cyclopent-2-enone C-2-carbanions. 255
Adenosine receptors and human melanoma 255
Design, synthesis, in vitro, and in vivo anticancer and antiangiogenic activity of novel 3-arylaminobenzofuran derivatives targeting the colchicine site on tubulin 255
A [3 + 2] nitrile oxide cycloaddition approach to retinoids 253
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists 253
Design, synthesis, DNA binding, and biological evaluation of water-soluble hybrid molecules containing two pyrazole analogues of the alkylating cyclopropylpyrroloindole (CPI) subunit of the antitumor agent CC-1065 and polypyrrole minor groove binders 252
[H-3]-MRE 2029-F20, a selective antagonist radioligand for the human A(2B) adenosine receptors 250
[H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors 245
A new nitrile oxide based synthesis of the antitumor agent geiparvarin 244
3,5-Disubstituted Isoxazoles as Synthons for (±)-Pyrenophorin and (±)-Vermiculine Synthesis 244
New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A 3 adenosine receptor antagonists 244
N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor 241
DNA minor groove binders as potential antitumor and antimicrobial agents 241
Pyrazolo [4,3-e][1,2,4]triazolo[1,5-c]pyrimidine template: Organic and medicinal chemistry approach 240
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2. 240
Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents 239
Allosteric enhancers for A(1) adenosine receptor 238
2-Arylamino-4-amino-5-aroylthiazoles. "One-pot" synthesis and biological evaluation of a new class of inhibitors of tubulin polymerization 238
Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffolds 237
Design, synthesis and in vitro cytotoxicity of a cis-dichloroplatinum(II) complex linked to the minor groove binder stallimycin 236
History and perspectives of A2A adenosine receptor antagonists as potential therapeutic agents 236
Binding of hybrid molecules containing pyrrolo [2,1-c][1,4]benzodiazepine (PBD) and oligopyrrole carriers to the human immunodeficiency type 1 virus TAR-RNA 231
Blockade of A2A receptors plus L-DOPA after nigrostriatal lesion results in GAD67 mRNA changes different from L-DOPA alone in the rat globus pallidus and substantia nigra reticulata 230
Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor 229
A new direct glycosylation of pyrimidine, pyrazole, imidazole and purine heterocycles via their N-tetrahydropyranyl (THP) derivatives 229
Active γ-manganese dioxide promoted conversion of 4,5-dihydro-1,2-oxazoles to 1,2-oxazoles. 228
Pyrazole phenylcyclohexylcarbamates as inhibitors of human fatty acid amide hydrolases (FAAH) 228
null 227
From tyrosine to glycine: Synthesis and biological activity of potent antagonists of the purinergic P2X(7) receptor 226
Adenosine Receptor Antagonists: Translating Medicinal Chemistry and Pharmacology into Clinical Utility 226
Synthesis and preliminary biological evaluation of new anti-tubulin agents containing different benzoheterocycles 225
One-pot reaction to obtain N,N'-disubstituted guanidines of pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine scaffold as human A3 adenosine receptor antagonists 225
Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation 225
5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists. 224
Novel 8-heterocyclyl xanthine derivatives in drug development - An update 224
1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors 223
Bis-epoxyethyl derivatives of distamycin A modified on the amidino moiety: Induction of production of fetal hemoglobin in human erythroid precursor cells 222
Hybrid molecules between distamycin A and active moieties of antitumor agents 222
A3 adenosine receptors in human neutrophils and promyelocytic HL60 cells: a pharmacological and biochemical study 221
Carboxyl activation in peptide synthesis using 4-oximino-pyrazol-5-ones 221
Hybrid molecules based on distamycin A as potential antitumor agents 219
Synthesis, in vitro antiproliferative activity, and DNA-binding properties of hybrid molecules containing pyrrolo[2,1-c][1,4] benzodiazepine and minor-groove-binding oligopyrrole carriers 219
A one-pot glycosylation of tetrahydropyranyl (THP) ether intermediates 218
Geiparvarin analogs. 2. Synthesis and cytostatic activity of 5-(4-arylbutadienyl)-3(2H)-furanones and of N-substituted 3-(4-oxo-2-furanyl)-2-buten-2-yl carbamates. 218
Adenosine receptors as mediators of both cell proliferation and cell death of cultured human melanoma cells 217
Current status of A1 adenosine receptor allosteric enhancers 217
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2 216
Biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptors 216
A new simple synthesis of a-substituted acrylonitriles 214
Ethyl 2,4-dioxoalkanoates as starting materials for a convenient route to 3(2H)-furanones and 3(2H)-furanimines 213
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon 213
Synthesis of hybrid distamycin-cysteine labeled with 99mTc: a model for a novel class of cancer imaging agents 213
[3H]-MRE 2029-F20, a novel selective antagonist radioligand, for the pharmacological and biochemical characterization of A2B receptors. 213
Methyl 4-oxothiolane-3-carboxylate and methyl 2-methyl-4-oxothiolane-3- carboxylate anions as synthetic equivalents of α-acrylate and α-crotonate anions. Formal synthesis of integerrinecic acid 212
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors 212
Transient receptor potential ankyrin receptor 1 is a novel target for pro-tussive agents 212
A mild one-pot synthesis of thieno[3,4-c]pyrazoles and their conversion into pyrazole analogs of o-quinodimethane 210
Structure-activity relationship studies of a new series of imidazo[2,1-f] purinones as potent and selective A3 adenosine receptor antagonists 210
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor 210
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists 209
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor 209
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked Heterocycles as template for the adenosine receptor antagonism: Medicinal chemistry approach and sar considerations 209
7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility. 209
Discovery and Optimization of a Series of 2-Aryl-4-Amino-5-(3 ',4 ',5 '-trimethoxybenzoyl)Thiazoles as Novel Anticancer Agents 209
A new synthetic approach to indazole synthesis 209
Cinnamoyl nitrogen mustard derivatives of pyrazole analogues of tallimustine modified at the amidino moiety: design, synthesis, molecular modeling and antitumor activity studies 208
[3H]MRE2029F20 a new selective antagonist radioligand for the human A2B adenosine receptors. 208
Modulation of metalloproteinase-9 in U87MG glioblastoma cells by A3 adenosine receptors 207
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility 207
Design, synthesis and growth inhibition activity of bis-epoxyethyl derivatives of stallimycin modified on the amidino moiety 206
Synthesis of conformationally constrained analogues of KN62, a potent antagonist of the P2X7-receptor 205
A new synthetic approach to pyrazolo[3,4-c]-1,2,5-oxadiazoles 205
Totale 34.608
Categoria #
all - tutte 338.202
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 3.331
Totale 341.533


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021553 0 0 0 0 0 0 0 0 0 0 0 553
2021/20225.094 159 470 372 291 373 250 208 243 197 361 528 1.642
2022/20234.800 508 249 108 646 881 773 145 390 611 31 286 172
2023/20242.411 243 307 129 82 170 287 95 394 28 60 56 560
2024/20259.331 291 294 752 335 1.154 770 273 638 1.285 1.084 1.377 1.078
2025/202636.220 2.653 1.709 4.045 3.576 3.659 1.892 3.275 1.339 9.919 3.179 886 88
Totale 88.836