BARALDI, Pier Giovanni
BARALDI, Pier Giovanni
Dipartimento di Scienze Chimiche e Farmaceutiche (attivo dal 01/01/2012 al 31/12/2022)
1,2,3-triazolo[5,4-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new class of A(2A) adenosine receptor antagonists
file con accesso da definire1996 Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G; PINEDA DE LAS INFANTAS, Mj; Zocchi, C; Ferrara, S; Dionisotti, S.
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists
file con accesso da definire2008 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea
1,4-Diketones via Isoxazole Intermediates
1979 Barco, Achille; Benetti, Simonetta; Pollini, Gian Piero; Baraldi, Pier Giovanni; Guarneri, Mario; Vicentini, Chiara Beatrice
1-methyl-3-nitro-5-methoxycarbonyl pyrazole
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.
1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors
file con accesso da definire1999 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.
1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors
file con accesso da definire1996 Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINEDA DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia
2,3a,5,6,7,7a-Hexahydro-3H,4H-benzothiophene-3,4-dione and cyclopenta[b]tetrahydrothiophene-3,4-dione enolate anions as synthetic equivalents to cyclohex-2-enone and cyclopent-2-enone C-2-carbanions.
file con accesso da definire1984 Baraldi, Pier Giovanni; Barco, Achille; Benetti, Simonetta; Pollini, Gian Piero; Zanirato, Vinicio
2-Arylamino-4-Amino-5-Aroylthiazoles. "One-Pot" Synthesis and Biological Evaluation of a New Class of Inhibitors of Tubulin Polymerization.
file con accesso da definire2009 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Basso, G.; Viola, G.; Khedr, M.; Balzarini, J.; Mahboobi, S.; Sellmer, A.; Brancale, A.; Hamel, E.
3,5-Disubstituted isoxazoles as a latent aldol moiety: application to the synthesis of (±)-[6]-gingerol.
file con accesso da definire1981 Barco, Achille; Benetti, Simonetta; Baraldi, Pier Giovanni; Guarneri, Mario; Pollini, Gian Piero; Simoni, Daniele
3,5-Disubstituted isoxazoles as synthons for (±)-pyrenophorin and (±)-vermiculine synthesis.
file con accesso da definire1983 Baraldi, Pier Giovanni; Barco, Achille; Benetti, Simonetta; Moroder, Fabio; Pollini, Gian Piero; Simoni, Daniele
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
5'-Phosphoramidates and 5'-diphosphates of 2'-O-allyl-β-D- arabinofuranosyl-uracil, -cytosine, and -adenine: Inhibition of ribonucleotide reductase
file con accesso da definire1999 Manfredini, Stefano; Baraldi, Pier Giovanni; Durini, Elisa; Vertuani, Silvia; Balzarini, Jan; DE CLERCQ, Erik; Karlsson, Anna; Buzzoni, Valentina; Thelander, Lars
5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists.
file con accesso da definire2006 Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G.
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility
file con accesso da definire2002 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation
2012 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1
file con accesso da definire2000 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Leoni, A; Bianchi, Nicoletta; Feriotto, Giordana; Rutigliano, C; Mischiati, Carlo; Gambari, Roberto
[3H]-MRE 2029-F20, a novel selective antagonist radioligand, for the pharmacological and biochemical characterization of A2B receptors.
file con accesso da definire2006 Gessi, Stefania; Varani, Katia; Merighi, Stefania; Cattabriga, Elena; Szabadkai, Y.; Rizzuto, Rosario; Klotz, K. N.; Leung, E.; Maclennan, S.; Baraldi, Pier Giovanni; Borea, Pier Andrea
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,2,3-triazolo[5,4-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new class of A(2A) adenosine receptor antagonists | 1996 | Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G; PINEDA DE LAS INFANTAS, Mj; Zocchi, C; Fe...rrara, S; Dionisotti, S. | file con accesso da definire |
| 1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists | 2008 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 1,4-Diketones via Isoxazole Intermediates | 1979 | Barco, Achille; Benetti, Simonetta; Pollini, Gian Piero; Baraldi, Pier Giovanni; Guarneri, Mario;... Vicentini, Chiara Beatrice | |
| 1-methyl-3-nitro-5-methoxycarbonyl pyrazole | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G. | file con accesso da definire |
| 1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors | 1999 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G. | file con accesso da definire |
| 1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors | 1996 | Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINED...A DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia | file con accesso da definire |
| 2,3a,5,6,7,7a-Hexahydro-3H,4H-benzothiophene-3,4-dione and cyclopenta[b]tetrahydrothiophene-3,4-dione enolate anions as synthetic equivalents to cyclohex-2-enone and cyclopent-2-enone C-2-carbanions. | 1984 | Baraldi, Pier Giovanni; Barco, Achille; Benetti, Simonetta; Pollini, Gian Piero; Zanirato, Vinicio | file con accesso da definire |
| 2-Arylamino-4-Amino-5-Aroylthiazoles. "One-Pot" Synthesis and Biological Evaluation of a New Class of Inhibitors of Tubulin Polymerization. | 2009 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Basso, ...G.; Viola, G.; Khedr, M.; Balzarini, J.; Mahboobi, S.; Sellmer, A.; Brancale, A.; Hamel, E. | file con accesso da definire |
| 3,5-Disubstituted isoxazoles as a latent aldol moiety: application to the synthesis of (±)-[6]-gingerol. | 1981 | Barco, Achille; Benetti, Simonetta; Baraldi, Pier Giovanni; Guarneri, Mario; Pollini, Gian Piero;... Simoni, Daniele | file con accesso da definire |
| 3,5-Disubstituted isoxazoles as synthons for (±)-pyrenophorin and (±)-vermiculine synthesis. | 1983 | Baraldi, Pier Giovanni; Barco, Achille; Benetti, Simonetta; Moroder, Fabio; Pollini, Gian Piero; ...Simoni, Daniele | file con accesso da definire |
| 3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Bra...ncale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro | |
| 5'-Phosphoramidates and 5'-diphosphates of 2'-O-allyl-β-D- arabinofuranosyl-uracil, -cytosine, and -adenine: Inhibition of ribonucleotide reductase | 1999 | Manfredini, Stefano; Baraldi, Pier Giovanni; Durini, Elisa; Vertuani, Silvia; Balzarini, Jan; DE ...CLERCQ, Erik; Karlsson, Anna; Buzzoni, Valentina; Thelander, Lars | file con accesso da definire |
| 5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists. | 2006 | Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier ...Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G. | file con accesso da definire |
| 7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
| 7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility. | 2001 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility | 2002 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, ...E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility. | 2001 | Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation | 2012 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, S...tefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia | |
| [2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1 | 2000 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Leoni, A; B...ianchi, Nicoletta; Feriotto, Giordana; Rutigliano, C; Mischiati, Carlo; Gambari, Roberto | file con accesso da definire |
| [3H]-MRE 2029-F20, a novel selective antagonist radioligand, for the pharmacological and biochemical characterization of A2B receptors. | 2006 | Gessi, Stefania; Varani, Katia; Merighi, Stefania; Cattabriga, Elena; Szabadkai, Y.; Rizzuto, Ros...ario; Klotz, K. N.; Leung, E.; Maclennan, S.; Baraldi, Pier Giovanni; Borea, Pier Andrea | file con accesso da definire |