PRETI, Delia
 Distribuzione geografica
Continente #
NA - Nord America 7.606
EU - Europa 2.895
AS - Asia 1.233
SA - Sud America 12
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 3
AF - Africa 2
Totale 11.757
Nazione #
US - Stati Uniti d'America 7.595
DE - Germania 1.076
CN - Cina 742
UA - Ucraina 474
IT - Italia 422
TR - Turchia 375
GB - Regno Unito 264
RU - Federazione Russa 220
SE - Svezia 187
FI - Finlandia 110
VN - Vietnam 66
PL - Polonia 58
BE - Belgio 35
FR - Francia 23
HK - Hong Kong 16
CA - Canada 10
IN - India 9
KR - Corea 9
EU - Europa 6
NL - Olanda 6
BR - Brasile 4
CL - Cile 4
AR - Argentina 3
AU - Australia 3
ES - Italia 3
IR - Iran 3
JP - Giappone 3
LT - Lituania 3
PK - Pakistan 3
IE - Irlanda 2
IL - Israele 2
PT - Portogallo 2
SG - Singapore 2
AT - Austria 1
BG - Bulgaria 1
CH - Svizzera 1
DK - Danimarca 1
EG - Egitto 1
GR - Grecia 1
HR - Croazia 1
ID - Indonesia 1
KH - Cambogia 1
MA - Marocco 1
MC - Monaco 1
MN - Mongolia 1
MX - Messico 1
PE - Perù 1
RO - Romania 1
RS - Serbia 1
SK - Slovacchia (Repubblica Slovacca) 1
Totale 11.757
Città #
Fairfield 1.100
Woodbridge 1.035
Ann Arbor 606
Ashburn 574
Houston 534
Jacksonville 531
Chandler 500
Seattle 422
Wilmington 401
Cambridge 338
Ferrara 199
Izmir 182
Beijing 177
Nanjing 151
Princeton 131
San Diego 108
Boardman 85
Shanghai 85
Dong Ket 64
Milan 58
Warsaw 58
Bremen 57
Nanchang 50
Shenyang 49
New York 41
Tianjin 36
Brussels 35
Dearborn 35
San Mateo 32
Changsha 31
Hebei 30
Falls Church 27
Jiaxing 27
Redwood City 27
Mountain View 25
London 21
Addison 20
Philadelphia 18
Zhengzhou 18
Washington 17
Kunming 16
Jinan 15
Auburn Hills 14
Hong Kong 14
Munich 14
Duncan 13
Indiana 13
Norwalk 12
Orange 12
Des Moines 11
Ferrara di Monte Baldo 11
Helsinki 11
Los Angeles 11
Tappahannock 10
Guangzhou 9
Bari 8
Kilburn 8
Mcallen 8
Montréal 8
Ningbo 7
Padova 7
Verona 7
Chicago 6
Haikou 6
Hangzhou 6
Lanzhou 6
Bologna 5
Prescot 5
Augusta 4
Düsseldorf 4
Grassano 4
Rome 4
West Jordan 4
Xian 4
Yellow Springs 4
Bournemouth 3
Chongqing 3
Florence 3
Leawood 3
Lugo 3
Mysore 3
Taizhou 3
Waban 3
Wandsworth 3
Aversa 2
Buenos Aires 2
Calvizzano 2
Dublin 2
Frankfurt am Main 2
Hanoi 2
Hefei 2
Hyderabad 2
Isola della Scala 2
Rimini 2
San Jose 2
Torino 2
Toronto 2
Triggiano 2
Walnut 2
Acton 1
Totale 8.294
Nome #
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists 287
History and perspectives of A2A adenosine receptor antagonists as potential therapeutic agents 140
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization 137
Synthesis and preliminary biological evaluation of new anti-tubulin agents containing different benzoheterocycles 135
Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors 135
Design, synthesis and growth inhibition activity of bis-epoxyethyl derivatives of stallimycin modified on the amidino moiety 132
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2. 131
Water-Soluble Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines as Human A3 Adenosine Receptor Antagonists 131
Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor 131
Discovery and Optimization of a Series of 2-Aryl-4-Amino-5-(3 ',4 ',5 '-trimethoxybenzoyl)Thiazoles as Novel Anticancer Agents 130
1,3,8-Triazaspiro compounds and their use as medicaments for the treatment of reperfusion injury. 130
DNA minor groove binders as potential antitumor and antimicrobial agents 129
New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A 3 adenosine receptor antagonists 129
The involvement of the TRPA1 receptor in a mouse model of sympathetically maintained neuropathic pain 128
From tyrosine to glycine: Synthesis and biological activity of potent antagonists of the purinergic P2X(7) receptor 127
Hybrid molecules based on distamycin A as potential antitumor agents 127
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon 126
Novel 8-heterocyclyl xanthine derivatives in drug development - An update 126
The TRPA1 channel mediates the analgesic action of dipyrone and pyrazolone derivatives 126
null 124
Discovery of Novel 1,3,8-Triazaspiro[4.5]decane Derivatives That Target the c Subunit of F1/FO-Adenosine Triphosphate (ATP) Synthase for the Treatment of Reperfusion Damage in Myocardial Infarction 123
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[(4- arylpiperazin-1-yl)methyl]-5-substituted-thiophenes. Effect of the 5-modification on allosteric enhancer activity at the A1 adenosine receptor 123
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2. 122
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors 121
Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxyphenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents 121
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation 121
null 121
Pyrazolo [4,3-e][1,2,4]triazolo[1,5-c]pyrimidine template: Organic and medicinal chemistry approach 120
Recent improvements in the development of A2B adenosine receptor agonists. 120
null 120
null 118
A3 adenosine receptor antagonists: History and future perspectives 117
Structure-and conformation-Activity studies of nociceptin/orphanin FQ receptor dimeric ligands 117
N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor 116
Synthesis and Biological Evaluation of 1-Methyl-2-(3’,4’,5’-Trimethoxybenzoyl)-3-Amino Indoles as a New Class of Antimitotic Agents and Tubulin Inhibitors 114
Transient receptor potential ankyrin receptor 1 is a novel target for pro-tussive agents 113
Microwave-assisted synthesis of substituted 2,4-diarylthiazoles and their evaluation as anticancer agents 112
null 112
Medicinal Chemistry of A3 Adenosine Receptor Modulators: Pharmacological Activities and Therapeutic Implications 111
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N- (substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor 111
Allosteric enhancers for A(1) adenosine receptor 110
null 110
Recent improvements in the development of A2B adenosine receptor agonists 110
Transient Receptor Potential Ankyrin 1 (TRPA1) Channel as Emerging Target for Novel Analgesics and Anti-Inflammatory Agents 110
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists 110
The blockade of transient receptor potential ankirin 1 (TRPA1) signalling mediates antidepressant- and anxiolytic-like actions in mice 110
Oxaliplatin elicits mechanical and cold allodynia in rodents via TRPA1 receptor stimulation 109
null 109
Structure-activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A(3) adenosine receptor antagonists. 108
Concise Synthesis and Biological Evaluation of 2-Aroyl-5-Amino Benzo[b]thiophene Derivatives As a Novel Class of Potent Antimitotic Agents 108
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene 108
Hybrid molecules between distamycin A and active moieties of antitumor agents 108
Ozone-induced hypertussive responses in rabbits and guinea pigs 105
Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach 103
null 103
Activation of TRPA1 on dural afferents: a potential mechanism of headache pain 102
Neuropeptide S receptor ligands: a patent review (2005-2016) 102
The P2X7 receptor as a therapeutic target. 101
Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor 101
Recent developments in the field of adenosine receptor ligands. 99
The 'headache tree' via umbellulone and TRPA1 activates the trigeminovascular system. 99
C subunit of F1/FO-ATP synthase as target for preventing the detrimental effect of myocardial ischemia/reperfusion injury 99
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists 98
New 2-arylpyrazolo[4,3-c]quinoline derivates as potent and selective human A3 adenosine receptor antagonists 97
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor 96
null 96
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked heterocycles as template for the adenosine receptor antagonism: medicinal chemistry approach and SAR considerations. 95
Biased Agonism at Nociceptin/Orphanin FQ Receptors: A Structure Activity Study on N/OFQ(1-13)-NH2 95
Synthesis and biological evaluation of 2-substituted-4-(3 ',4 ',5 '-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents 94
Acetaminophen, via its reactive metabolite N-acetyl-p-benzo-quinoneimine and transient receptor potential ankyrin-1 stimulation, causes neurogenic inflammation in the airways and other tissues in rodents 94
[H-3]-MRE 2029-F20, a selective antagonist radioligand for the human A(2B) adenosine receptors 92
null 92
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists 91
Synthesis and biological evaluation of 2-aroyl-4-phenyl-5-hydroxybenzofurans as a new class of antitubulin agents 91
Tetrabranched Hetero-Conjugated Peptides as Bifunctional Agonists of the NOP and Mu Opioid Receptors 90
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor 89
Recent developments in the field of A(2A) and A(3) adenosine receptor antagonists 87
null 87
New strategies for the synthesis of A(3) adenosine receptor antagonists 87
null 87
Hybrid molecules containing benzo[4,5]imidazo[1,2-d][1,2,4]thiadiazole and alpha-bromoacryloyl moieties as potent apoptosis inducers on human myeloid leukaemia cells 86
Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors 86
TRP channels as therapeutic targets in airway disorders: a patent review 85
Design, synthesis, and biological evaluation of C-9- and C-2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c] pyrimidines as new A(2A) and A(3) adenosine receptors antagonists 84
null 84
New pyrrolo[2,1-f]purine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives as potent and selective human A(3) adenosine receptor antagonists 83
Preparation of fused purine derivatives as adenosine A3 receptor modulators. 83
null 83
null 82
Preparation of fused purine derivatives as adenosine A3 receptor modulators. 81
Design, synthesis and biological evaluation of hybrid molecules containing conjugated styryl ketone and α-bromoacryloyl moieties 80
Discovery of novel fetal hemoglobin inducers for β-thalassemia by small chemical library screening 80
Recent developments in the field of A2B and A3 adenosine receptors antagonists 79
Pharmacological profile of the neuropeptide S receptor: Dynamic mass redistribution studies 77
Adenosine Modulates HIF-1 alpha, VEGF, IL-8, and Foam Cell Formation in a Human Model of Hypoxic Foam Cells 75
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A(3) adenosine receptor antagonists 75
The acyl-glucuronide metabolite of ibuprofen has analgesic and anti-inflammatory effects via the TRPA1 channel 75
Recent improvements in the field of A(3) adenosine receptor ligands 74
Role of TRPA1 receptors in skin inflammation induced by volatile chemical irritants in mice 74
null 73
Totale 10.695
Categoria #
all - tutte 41.986
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 1.078
Totale 43.064


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019899 0 0 0 0 0 0 0 0 0 0 359 540
2019/20202.469 378 94 83 356 180 285 226 240 208 231 141 47
2020/20211.854 183 134 91 184 85 183 83 217 59 281 186 168
2021/20221.365 62 127 137 55 88 61 84 57 47 105 140 402
2022/20231.270 132 86 23 181 239 171 53 92 169 9 64 51
2023/2024619 59 96 49 25 60 137 41 90 25 19 18 0
Totale 11.938