PACIFICO, Salvatore

PACIFICO, Salvatore  

Dipartimento di Scienze chimiche, farmaceutiche ed agrarie  

Mostra records
Risultati 1 - 20 di 58 (tempo di esecuzione: 0.026 secondi).
Titolo Data di pubblicazione Autore(i) File
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism 2017 Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, M...aria Camilla; Trapella, Claudio; Calo', Girolamo
A Peptidic Thymidylate-Synthase Inhibitor Loaded on Pegylated Liposomes Enhances the Antitumour Effect of Chemotherapy Drugs in Human Ovarian Cancer Cells 2020 Marverti, Gaetano; Gozzi, Gaia; Maretti, Eleonora; Lauriola, Angela; Severi, Leda; Sacchetti, Fra...ncesca; Losi, Lorena; Pacifico, Salvatore; Ferrari, Stefania; Ponterini, Glauco; Leo, Eliana; Costi, Maria Paola; D'Arca, Domenico
Activation of nociceptin/orphanin FQ receptors inhibits contextual fear memory reconsolidation 2017 Rekik, Khaoula; Faria Da Silva, Raquel; Colom, Morgane; Pacifico, Salvatore; Zaveri, Nurulain T; ...Calo', Girolamo; Rampon, Claire; Frances, Bernard; Mouledous, Lionel file con accesso da definire
Age, Sex, Hypertension and HDL-C Alter Serum BACE1 Activity in Cognitively Normal Subjects: Implications for Alzheimer's Disease 2022 Cervellati, C; Vergallo, A; Trentini, A; Campo, G; Vieceli Dalla Sega, F; Bonaccorsi, G; Rosta, V...; Renzini, C; Pacifico, S; Passaro, A; Hampel, H; Zuliani, G; Rizzo, P
Ageing Curtails the Diversity and Functionality of Nascent CD8+ T Cell Responses against SARS-CoV-2 2023 Proietto, Davide; Dallan, Beatrice; Gallerani, Eleonora; Albanese, Valentina; Llewellyn-Lacey, Si...an; Price, David A.; Appay, Victor; Pacifico, Salvatore; Caputo, Antonella; Nicoli, Francesco; Gavioli, Riccardo
alpha-Diketones as acyl anion equivalents: a non-enzymatic thiamine-promoted route to aldehyde ketone coupling in PEG(400) as recyclable medium 2011 Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina;... Pacifico, Salvatore; Massi, Alessandro file con accesso da definire
alpha-Diketones as acyl anion equivalents: new enzymatic and non-enzymatic thiamine-promoted routes to aldehyde-ketone coupling 2011 Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina;... Massi, Alessandro; Pacifico, Salvatore file con accesso da definire
Biased Agonism at Nociceptin/Orphanin FQ Receptors: A Structure Activity Study on N/OFQ(1-13)-NH2 2020 Pacifico, S.; Ferrari, F.; Albanese, V.; Marzola, E.; Neto, J. A.; Ruzza, C.; Calo, G.; Preti, D....; Guerrini, R.
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth 2018 Saxena, P; Severi, L; Santucci, M; Taddia, L; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C;... Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp
Conveying a newly designed hydrophilic anti-human thymidylate synthase peptide to cisplatin resistant cancer cells: are pH-sensitive liposomes more effective than conventional ones? 2017 Sacchetti, Francesca; D'Arca, Domenico; Genovese, Filippo; Pacifico, Salvatore; Maretti, E; Hanus...kova, M; Iannuccelli, V; Costi, Mp; Leo, E. file con accesso da definire
Cyclic peptides acting as allosteric inhibitors of human thymidylate synthase and cancer cell growth 2019 Pacifico, S.; Santucci, M.; Luciani, R.; Saxena, P.; Linciano, P.; Ponterini, G.; Lauriola, A.; D...'Arca, D.; Marverti, G.; Guerrini, R.; Costi, M. P.
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones 2016 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna...; Manfredini, Stefano; Pacifico, Salvatore; Liekens, Sandra; Balzarini, Jan
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth. 2022 Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; H Salo-Ahen, Outi M; Carosati, Emanuele; F...ranchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; DI BENEDETTO CARDINALE, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Gaetana Moschella, Maria; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela; Giovannetti, Elisa; J Peters, Godefridus; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; M Stroud, Robert; C Wade, Rebecca; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Paola Costi, Maria file con accesso da definire
Dimethyl Sulfoxide and N,N-dimethylformamide as Umpolung Pre-catalysts in Cross Benzoin Reactions of alpha-Diketones with Aldehydes 2013 Bortolini, Olga; Massi, Alessandro; Giovannini, Pier Paolo; Pacifico, Salvatore; Ragno, Daniele; ...Zaghi, Anna file con accesso da definire
Discovery of Novel 1,3,8-Triazaspiro[4.5]decane Derivatives That Target the c Subunit of F1/FO-Adenosine Triphosphate (ATP) Synthase for the Treatment of Reperfusion Damage in Myocardial Infarction 2018 Morciano, Giampaolo; Preti, Delia; Pedriali, Gaia; Aquila, Giorgio; Missiroli, Sonia; Fantinati, ...Anna; Caroccia, Natascia; Pacifico, Salvatore; Bonora, Massimo; Talarico, Anna; Morganti, Claudia; Rizzo, Paola; Ferrari, Roberto; Wieckowski, Mariusz R.; Campo, Gianluca; Giorgi, Carlotta; Trapella, Claudio; Pinton, Paolo
Discovery of novel fetal hemoglobin inducers for β-thalassemia by small chemical library screening 2020 Breveglieri, G; Pacifico, Salvatore; Zuccato, Cristina; Cosenza, Lucia Carmela; Sultan, Shaiq; D'...Aversa, Elisabetta; Gambari, Roberto; Preti, Delia; Trapella, Claudio; Guerrini, Remo; Borgatti, Monica
Effects of non-peptide nociceptin/orphanin FQ receptor ligands on methylphenidate-induced hyperactivity in mice: Implications for bipolar disorders 2020 Asth, Laila; Tiago, Pamella R. F.; Costa, Layse R. F.; Holanda, Victor A. D.; Pacifico, Salvatore...; Zaveri, Nurulain T.; Calo', Girolamo; Ruzza, Chiara; Gavioli, Elaine C.
Expeditious Synthesis and Biological Characterization of Enantio-Enriched (-)-Nutlin-3 2017 Fantinati, Anna; Bianco, Sara; Cristofori, Virginia; Cavazzini, Alberto; Catani, Martina; Zanirat...o, Vinicio; Pacifico, Salvatore; Rimondi, Erika; Milani, Daniela; Voltan, Rebecca; Secchiero, Paola; Trapella, Claudio
Fluorometric detection of protein-ligand engagement: The case of phosphodiesterase5 2018 Di Rocco, G; Martinelli, I; Pacifico, S; Guerrini, R; Cichero, E; Fossa, P; Franchini, S; Cardare...lli, S; Giorgi, M; Sola, M; Ponterini, G.
Folic Acid-Peptide Conjugates Combine Selective Cancer Cell Internalization with Thymidylate Synthase Dimer Interface Targeting 2021 Marverti, G.; Marraccini, C.; Martello, A.; D'Arca, D.; Pacifico, S.; Guerrini, R.; Spyrakis, F.;... Gozzi, G.; Lauriola, A.; Santucci, M.; Cannazza, G.; Tagliazucchi, L.; Cazzato, A. S.; Losi, L.; Ferrari, S.; Ponterini, G.; Costi, M. P.