TRAPELLA, Claudio

TRAPELLA, Claudio  

Dipartimento di Scienze chimiche, farmaceutiche ed agrarie  

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Titolo Data di pubblicazione Autore(i) File
(L)-Monomethyl Tyrosine (Mmt): New Synthetic Strategy via Bulky ‘Forced-Traceless’ Regioselective Pd-Catalyzed C(sp2)–H Activation 2023 Illuminati, Davide; Trapella, Claudio; Zanirato, Vinicio; Guerrini, Remo; Albanese, Valentina; St...uraro, Chiara; Stragapede, Simona; Malfacini, Davide; Compagnin, Greta; Catani, Martina; Fantinati, Anna file con accesso da definire
1,3,8-Triazaspiro compounds and their use as medicaments for the treatment of reperfusion injury. 2019 Pinton, Paolo; Ferrari, Roberto; Giorgi, Carlotta; Trapella, Claudio; Preti, Delia; Morciano, Gia...mpaolo file con accesso da definire
1,3,8-Triazaspiro[4.5]decane Derivatives Inhibit Permeability Transition Pores through a FO-ATP Synthase c Subunit Glu119-Independent Mechanism That Prevents Oligomycin A-Related Side Effects 2023 Pedriali, G.; Ramaccini, D.; Bouhamida, E.; Branchini, A.; Turrin, G.; Tonet, E.; Scala, A.; Pate...rgnani, S.; Pinotti, M.; Trapella, C.; Giorgi, C.; Tremoli, E.; Campo, G.; Morciano, G.; Pinton, P. file con accesso da definire
1,4-Dithiane-2,5-diol: An Attractive Platform for the Synthesis of Sulfur-Containing Functionalized Heterocycles 2018 Zamberlan, Francesco; Fantinati, Anna; Trapella, Claudio
1-Benzyl-N-[3-[spiroisobenzofuran-1(3H),4′-piperidin-1-yl]propyl]pyrrolidine-2-carboxamide (Compound 24) antagonizes NOP receptor-mediated potassium channel activation in rat periaqueductal gray slices 2009 Liao, Y. Y.; Trapella, Claudio; Chiou, L. C. file con accesso da definire
1‐cyclohexyl‐x‐methoxybenzene derivatives, novel psychoactive substances seized on the internet market. Synthesis and in vivo pharmacological studies in mice 2017 Fantinati, Anna; Ossato, Andrea; Bianco, Sara; Canazza, Isabella; De Giorgio, F; Trapella, Claudi...o; Marti, Matteo
6-N,N-dimethylamino-2,3-naphthalimide: A new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides 2006 Vazquez, Me; Blanco, Jb; Salvadori, Severo; Trapella, Claudio; Argazzi, Roberto; Bryant, Sd; Jins...maa, Y; Lazarus, Lh; Negri, L; Giannini, E; Lattanzi, R; Colucci, M; Balboni, G. file con accesso da definire
[D-Pen(p-tBuBzl)5]NPS, a novel ligand for the neuropeptide S receptor: structure activity and pharmacological studies 2014 Ruzza, Chiara; L., del Zoppo; Malfacini, Davide; Pela', Michela; Trapella, Claudio; P., Grieco; S...alvadori, Severo; Calo', Girolamo; Guerrini, Remo file con accesso da definire
A Cationic Contrast Agent in X-ray Imaging of Articular Cartilage: Pre-Clinical Evaluation of Diffusion and Attenuation Properties 2022 Fantoni, Simone; Gabucci, Ilenia; Cardarelli, Paolo; Paternò, Gianfranco; Taibi, Angelo; Cristofo...ri, Virginia; Trapella, Claudio; Bazzani, Armando; Assenza, Marta; Zanna Bonacorsi, Alice; Conti, Daniele; Baruffaldi, Fabio
A Convenient Route to Enantiomerically Pure 2-Substituted Methyl Glycerate Derivatives 2003 Ley, S. V.; Trapella, Claudio; Michel, P. file con accesso da definire
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism 2017 Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, M...aria Camilla; Trapella, Claudio; Calo', Girolamo
A linear allergic contact dermatitis to p-tert-butylphenol formaldehyde resin sectorially present in a neoprene orthopedic brace: role of spectroscopy 2012 Corazza, Monica; S., Zauli; Bernardi, Tatiana; Trapella, Claudio; Benetti, Simonetta; Virgili, Anna file con accesso da definire
A new amido-phosphine of dichloroacetic acid as an active ligand for metals of pharmaceutical interest. Synthesis, characterization and tests of antiproliferative and pro-apoptotic activity 2019 Marvelli, L.; Ferretti, V.; Bertolasi, V.; Lampronti, I.; Gambari, R.; Trapella, C.; Turrin, G.; ...Bonotto, F.; Moriello, A.; Bergamini, P.
A new synthetic approach to 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidyl]-3-ethyl-1,3-dihydro-benzimidazol-2-one (J-113397), the first non-peptide ORL-1 receptor antagonist 2001 DE RISI, Carmela; Pollini, Gian Piero; Trapella, Claudio; Peretto, I.; Ronzoni, S.; Giardina, G. ...A. M. file con accesso da definire
A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ. 2014 Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pela', Michela; Molinari, Stefano; Cerlesi, Ma...ria Camilla; Malfacini, Davide; Rizzi, Anna; Salvadori, Severo; Calo', Girolamo file con accesso da definire
A proteomic approach to investigate the mechanism of action of anticancer peptides 2013 F., Genovese; A., Gualandi; L., Taddia; M., Caselli; G., Ponterini; S., Ferrari; G., Marverti; Gu...errini, Remo; Pela', Michela; G., Pavesi; Trapella, Claudio; M. P., Costi file con accesso da definire
An alternative enzymatic route to the ergogenic ketone body ester (R)-3-hydroxybutyl (r)-3-hydroxybutyrate 2021 Zaccone, F.; Venturi, V.; Giovannini, P. P.; Trapella, C.; Narducci, M.; Fournier, H.; Fantinati, A.
Antinociceptive action of NOP and opioid receptor agonists in the mouse orofacial formalin test 2017 Rizzi, Anna; Ruzza, Chiara; Bianco, Sara; Trapella, Claudio; Calo', Girolamo file con accesso da definire
Anxiolytic and antidepressant-like activities of UFP-512, a novel selective delta opiold receptor agonist 2006 Vergura, Raffaella; Balboni, G; Spagnolo, Barbara; Gavioli, Elaine Cristina; Lambert, Dg; Mcdonal...d, J; Trapella, Claudio; Regoli, Domenico; Salvadori, Severo; Calo', Girolamo file con accesso da definire
Anxiolytic- and antidepressant-like activities of H-Dmt-Tic-NH-CH(CH2-COOH)-Bid (UFP-512), a novel selective delta opioid receptor agonist 2008 Vergura, Raffaella; G., Balboni; Spagnolo, Barbara; Gavioli, Elaine Cristina; D. G., Lambert; J.,... Mcdonald; Trapella, Claudio; L. H., Lazarus; Regoli, Domenico; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo file con accesso da definire