VINCENZI, Fabrizio
VINCENZI, Fabrizio
Dipartimento di Medicina Traslazionale e per la Romagna
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
file con accesso da definire2023 Oliva, Paola; Suresh, R Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J; Tosh, Dilip K; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation
file con accesso da definire2013 Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S.
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold To Obtain Potent and Selective Human A(3) Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition (dagger).
file con accesso da definire2009 Lenzi, O.; Colotta, V.; Catarzi, D.; Varano, F.; Poli, D.; Filacchioni, G.; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Paoletta, S.; Morizzo, E.; Moro, S.
4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives
2022 Catarzi, D.; Varano, F.; Vigiani, E.; Calenda, S.; Melani, F.; Varani, K.; Vincenzi, F.; Pasquini, S.; Mennini, N.; Nerli, G.; Dal Ben, D.; Volpini, R.; Colotta, V.
7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A(1) and A(2A) adenosine receptors. Molecular modeling and pharmacological studies
2014 Squarcialupi, L; Colotta, V; Catarzi, D; Varano, F; Betti, M; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Porta, N; Ciancetta, A; Moro, S.
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
[3H]MRE2029F20 a new selective antagonist radioligand for the human A2B adenosine receptors.
file con accesso da definire2005 Borea, Pier Andrea; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Benini, Annalisa; Cattabriga, Elena; Baraldi, Pier Giovanni
A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach.
file con accesso da definire2012 Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spalluto, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
A(2A) adenosine receptors are differentially modulated by pharmacological treatments in rheumatoid arthritis patients and their stimulation ameliorates adjuvant-induced arthritis in rats
file con accesso da definire2013 Vincenzi, Fabrizio; Padovan, Melissa; Targa, Martina; Corciulo, Carmen; Giacuzzo, Sarah; Merighi, Stefania; Gessi, Stefania; Govoni, Marcello; Borea, Pa; Varani, Katia
A(2A) adenosine receptors are up-regulated in lymphocytes from amyotrophic lateral sclerosis patients
file con accesso da definire2013 Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Casetta, Ilaria; Gentile, Mauro; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea; P., Popoli; Varani, Katia
A(2B) adenosine receptors stimulate IL-6 production in primary murine microglia through p38 MAPK kinase pathway
2017 Merighi, Stefania; Bencivenni, Serena; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea; Gessi, Stefania
A1 Adenosine Receptor Partial Agonists and Allosteric Modulators: Advancing Toward the Clinic?
2020 Vincenzi, F.; Pasquini, S.; Battistello, E.; Merighi, S.; Gessi, S.; Borea, P. A.; Varani, K.
A2A Adenosine Receptor Antagonists in Neurodegenerative Diseases
2022 Merighi, Stefania; Borea, Pier Andrea; Varani, Katia; Vincenzi, Fabrizio; Jacobson, Kenneth A; Gessi, Stefania
A2A Adenosine Receptor as a Potential Biomarker and a Possible Therapeutic Target in Alzheimer's Disease
2021 Gessi, Stefania; Poloni, Tino Emanuele; Negro, Giulia; Varani, Katia; Pasquini, Silvia; Vincenzi, Fabrizio; Borea, Pier Andrea; Merighi, Stefania
A2A adenosine receptor overexpression and functionality, as well as TNF-alpha levels, correlate with motor symptoms in Parkinson's disease.
file con accesso da definire2010 Varani, Katia; Vincenzi, Fabrizio; Tosi, Alice; Gessi, Stefania; Casetta, Ilaria; Granieri, Gino; Fazio, Patrik; Leung, E; Maclennan, S; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea
A2A adenosine receptor upregulation correlates with disease activity in patients with systemic lupus erythematosus
file con accesso da definire2016 Bortoluzzi, Alessandra; Vincenzi, Fabrizio; Govoni, Marcello; Padovan, Melissa; Ravani, Annalisa; Borea, Pier Andrea; Varani, Katia
A2A Adenosine Receptor: A Possible Therapeutic Target for Alzheimer's Disease by Regulating NLRP3 Inflammasome Activity?
2022 Merighi, Stefania; Nigro, Manuela; Travagli, Alessia; Pasquini, Silvia; Borea, Pier Andrea; Varani, Katia; Vincenzi, Fabrizio; Gessi, Stefania
A2A adenosine receptors and chronic caffeine intake in human neutrophils
file con accesso da definire2005 Varani, Katia; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Belardinelli, L.; Borea, Pier Andrea
A2A adenosine receptors and chronic caffeine intake in human neutrophils
file con accesso da definire2005 Varani, Katia; Portaluppi, Francesco; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Belardinelli, L.; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
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2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators | 2023 | Oliva, Paola; Suresh, R Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J; Tosh, Dilip K;... Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A | file con accesso da definire |
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 2022 | Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Va...leria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation | 2013 | Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo,... Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S. | file con accesso da definire |
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold To Obtain Potent and Selective Human A(3) Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition (dagger). | 2009 | Lenzi, O.; Colotta, V.; Catarzi, D.; Varano, F.; Poli, D.; Filacchioni, G.; Varani, Katia; Vincen...zi, Fabrizio; Borea, Pier Andrea; Paoletta, S.; Morizzo, E.; Moro, S. | file con accesso da definire |
4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives | 2022 | Catarzi, D.; Varano, F.; Vigiani, E.; Calenda, S.; Melani, F.; Varani, K.; Vincenzi, F.; Pasquini..., S.; Mennini, N.; Nerli, G.; Dal Ben, D.; Volpini, R.; Colotta, V. | |
7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A(1) and A(2A) adenosine receptors. Molecular modeling and pharmacological studies | 2014 | Squarcialupi, L; Colotta, V; Catarzi, D; Varano, F; Betti, M; Varani, Katia; Vincenzi, Fabrizio; ...Borea, Pier Andrea; Porta, N; Ciancetta, A; Moro, S. | |
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
[3H]MRE2029F20 a new selective antagonist radioligand for the human A2B adenosine receptors. | 2005 | Borea, Pier Andrea; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Benini..., Annalisa; Cattabriga, Elena; Baraldi, Pier Giovanni | file con accesso da definire |
A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach. | 2012 | Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spallut...o, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
A(2A) adenosine receptors are differentially modulated by pharmacological treatments in rheumatoid arthritis patients and their stimulation ameliorates adjuvant-induced arthritis in rats | 2013 | Vincenzi, Fabrizio; Padovan, Melissa; Targa, Martina; Corciulo, Carmen; Giacuzzo, Sarah; Merighi,... Stefania; Gessi, Stefania; Govoni, Marcello; Borea, Pa; Varani, Katia | file con accesso da definire |
A(2A) adenosine receptors are up-regulated in lymphocytes from amyotrophic lateral sclerosis patients | 2013 | Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Casetta, Ilaria; Gentile, Mauro; Granieri, ...Enrico Gavino Giuseppe; Borea, Pier Andrea; P., Popoli; Varani, Katia | file con accesso da definire |
A(2B) adenosine receptors stimulate IL-6 production in primary murine microglia through p38 MAPK kinase pathway | 2017 | Merighi, Stefania; Bencivenni, Serena; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea; Ges...si, Stefania | |
A1 Adenosine Receptor Partial Agonists and Allosteric Modulators: Advancing Toward the Clinic? | 2020 | Vincenzi, F.; Pasquini, S.; Battistello, E.; Merighi, S.; Gessi, S.; Borea, P. A.; Varani, K. | |
A2A Adenosine Receptor Antagonists in Neurodegenerative Diseases | 2022 | Merighi, Stefania; Borea, Pier Andrea; Varani, Katia; Vincenzi, Fabrizio; Jacobson, Kenneth A; Ge...ssi, Stefania | |
A2A Adenosine Receptor as a Potential Biomarker and a Possible Therapeutic Target in Alzheimer's Disease | 2021 | Gessi, Stefania; Poloni, Tino Emanuele; Negro, Giulia; Varani, Katia; Pasquini, Silvia; Vincenzi,... Fabrizio; Borea, Pier Andrea; Merighi, Stefania | |
A2A adenosine receptor overexpression and functionality, as well as TNF-alpha levels, correlate with motor symptoms in Parkinson's disease. | 2010 | Varani, Katia; Vincenzi, Fabrizio; Tosi, Alice; Gessi, Stefania; Casetta, Ilaria; Granieri, Gino;... Fazio, Patrik; Leung, E; Maclennan, S; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea | file con accesso da definire |
A2A adenosine receptor upregulation correlates with disease activity in patients with systemic lupus erythematosus | 2016 | Bortoluzzi, Alessandra; Vincenzi, Fabrizio; Govoni, Marcello; Padovan, Melissa; Ravani, Annalisa;... Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
A2A Adenosine Receptor: A Possible Therapeutic Target for Alzheimer's Disease by Regulating NLRP3 Inflammasome Activity? | 2022 | Merighi, Stefania; Nigro, Manuela; Travagli, Alessia; Pasquini, Silvia; Borea, Pier Andrea; Varan...i, Katia; Vincenzi, Fabrizio; Gessi, Stefania | |
A2A adenosine receptors and chronic caffeine intake in human neutrophils | 2005 | Varani, Katia; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Belardinelli, L.; Borea, P...ier Andrea | file con accesso da definire |
A2A adenosine receptors and chronic caffeine intake in human neutrophils | 2005 | Varani, Katia; Portaluppi, Francesco; Gessi, Stefania; Merighi, Stefania; Vincenzi, Fabrizio; Bel...ardinelli, L.; Borea, Pier Andrea | file con accesso da definire |