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Mostrati risultati da 21 a 40 di 58
Titolo Data di pubblicazione Autore(i) File
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism 2017 Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, M...aria Camilla; Trapella, Claudio; Calo', Girolamo
Expeditious Synthesis and Biological Characterization of Enantio-Enriched (-)-Nutlin-3 2017 Fantinati, Anna; Bianco, Sara; Cristofori, Virginia; Cavazzini, Alberto; Catani, Martina; Zanirat...o, Vinicio; Pacifico, Salvatore; Rimondi, Erika; Milani, Daniela; Voltan, Rebecca; Secchiero, Paola; Trapella, Claudio
Conveying a newly designed hydrophilic anti-human thymidylate synthase peptide to cisplatin resistant cancer cells: are pH-sensitive liposomes more effective than conventional ones? 2017 Sacchetti, Francesca; D'Arca, Domenico; Genovese, Filippo; Pacifico, Salvatore; Maretti, E; Hanus...kova, M; Iannuccelli, V; Costi, Mp; Leo, E. file con accesso da definire
Activation of nociceptin/orphanin FQ receptors inhibits contextual fear memory reconsolidation 2017 Rekik, Khaoula; Faria Da Silva, Raquel; Colom, Morgane; Pacifico, Salvatore; Zaveri, Nurulain T; ...Calo', Girolamo; Rampon, Claire; Frances, Bernard; Mouledous, Lionel file con accesso da definire
Fluorometric detection of protein-ligand engagement: The case of phosphodiesterase5 2018 Di Rocco, G; Martinelli, I; Pacifico, S; Guerrini, R; Cichero, E; Fossa, P; Franchini, S; Cardare...lli, S; Giorgi, M; Sola, M; Ponterini, G.
Discovery of Novel 1,3,8-Triazaspiro[4.5]decane Derivatives That Target the c Subunit of F1/FO-Adenosine Triphosphate (ATP) Synthase for the Treatment of Reperfusion Damage in Myocardial Infarction 2018 Morciano, Giampaolo; Preti, Delia; Pedriali, Gaia; Aquila, Giorgio; Missiroli, Sonia; Fantinati, ...Anna; Caroccia, Natascia; Pacifico, Salvatore; Bonora, Massimo; Talarico, Anna; Morganti, Claudia; Rizzo, Paola; Ferrari, Roberto; Wieckowski, Mariusz R.; Campo, Gianluca; Giorgi, Carlotta; Trapella, Claudio; Pinton, Paolo
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth 2018 Saxena, P; Severi, L; Santucci, M; Taddia, L; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C;... Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp
Peptide welding technology – A simple strategy for generating innovative ligands for G protein coupled receptors 2018 Calo, Girolamo; Rizzi, Anna; Ruzza, Chiara; Ferrari, Federica; Pacifico, Salvatore; Gavioli, Elai...ne C.; Salvadori, Severo; Guerrini, Remo
Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones 2019 Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacif...ico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Modulation of the NOP receptor signaling affects resilience to acute stress 2019 D Holanda, Victor A; Pacifico, Salvatore; AZEVEDO NETO, Joaquim Gonalves; Finetti, Luca; Lobão-So...ares, Bruno; Calo', Girolamo; Gavioli, Elaine Cristina; Ruzza, Chiara
Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors 2019 Pacifico, Salvatore; Ferretti, Valeria; Albanese, Valentina; Fantinati, Anna; Gallerani, Eleonora...; Nicoli, Francesco; Gavioli, Riccardo; Zamberlan, Francesco; Preti, Delia; Marastoni, Mauro
Probing the Effect of Sildenafil on Progesterone and Testosterone Production by an Intracellular FRET/BRET Combined Approach 2019 Casarini, L; Riccetti, L; Limoncella, S; Lazzaretti, C; Barbagallo, F; Pacifico, S; Guerrini, R; ...Tagliavini, S; Trenti, T; Simoni, M; Sola, M; Di Rocco, G
Tetrabranched Hetero-Conjugated Peptides as Bifunctional Agonists of the NOP and Mu Opioid Receptors 2019 Pacifico, S.; Albanese, V.; Illuminati, Davide; Fantinati, A.; Marzola, E.; Ferrari, F.; Neto, J.... A.; Sturaro, Chiara; Ruzza, C.; Calo, G.; Preti, D.; Guerrini, R.
Cyclic peptides acting as allosteric inhibitors of human thymidylate synthase and cancer cell growth 2019 Pacifico, S.; Santucci, M.; Luciani, R.; Saxena, P.; Linciano, P.; Ponterini, G.; Lauriola, A.; D...'Arca, D.; Marverti, G.; Guerrini, R.; Costi, M. P.
Synthesis of folic acid functionalized gold nanoclusters for targeting folate receptor-positive cells 2019 Liu, Z.; Turyanska, L.; Zamberlan, F.; Pacifico, S.; Bradshaw, T. D.; Moro, F.; Fay, M. W.; Willi...ams, H. E. L.; Thomas, N. R.
A Peptidic Thymidylate-Synthase Inhibitor Loaded on Pegylated Liposomes Enhances the Antitumour Effect of Chemotherapy Drugs in Human Ovarian Cancer Cells 2020 Marverti, Gaetano; Gozzi, Gaia; Maretti, Eleonora; Lauriola, Angela; Severi, Leda; Sacchetti, Fra...ncesca; Losi, Lorena; Pacifico, Salvatore; Ferrari, Stefania; Ponterini, Glauco; Leo, Eliana; Costi, Maria Paola; D'Arca, Domenico
The Tat Protein of HIV-1 Prevents the Loss of HSV-Specific Memory Adaptive Responses and Favors the Control of Viral Reactivation 2020 Nicoli, Francesco; Gallerani, Eleonora; Sicurella, Mariaconcetta; Pacifico, Salvatore; Cafaro, Au...relio; Ensoli, Barbara; Marconi, Peggy; Caputo, Antonella; Gavioli, Riccardo
Increased blood BACE1 activity as a potential common pathogenic factor of vascular dementia and late onset Alzheimer's disease 2020 Zuliani, G.; Trentini, A.; Rosta, V.; Guerrini, R.; Pacifico, S.; Bonazzi, S.; Guiotto, A.; Passa...ro, A.; Seripa, D.; Valacchi, G.; Cervellati, C.
Effects of non-peptide nociceptin/orphanin FQ receptor ligands on methylphenidate-induced hyperactivity in mice: Implications for bipolar disorders 2020 Asth, Laila; Tiago, Pamella R. F.; Costa, Layse R. F.; Holanda, Victor A. D.; Pacifico, Salvatore...; Zaveri, Nurulain T.; Calo', Girolamo; Ruzza, Chiara; Gavioli, Elaine C.
Serum beta-secretase 1 (BACE1) activity as candidate biomarker for late-onset Alzheimer’s disease 2020 Cervellati, C.; Trentini, A.; Rosta, V.; Passaro, A.; Bosi, C.; Sanz, J. M.; Bonazzi, S.; Pacific...o, S.; Seripa, D.; Valacchi, G.; Guerini, R.; Zuliani, G.
Mostrati risultati da 21 a 40 di 58
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