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Titolo Data di pubblicazione Autore(i) File
Structure-activity studies on the nociceptin/orphanin FQ receptor antagonist 1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4'-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide. 2009 Trapella, Claudio; Fischetti, Carmela; Pela', Michela; Lazzari, Ilaria; Guerrini, Remo; Calo', Gi...rolamo; Rizzi, Anna; Camarda, Valeria; Lambert, Dg; Mcdonald, J; Regoli, Domenico; Salvadori, Severo file con accesso da definire
1-Benzyl-N-[3-[spiroisobenzofuran-1(3H),4′-piperidin-1-yl]propyl]pyrrolidine-2-carboxamide (Compound 24) antagonizes NOP receptor-mediated potassium channel activation in rat periaqueductal gray slices 2009 Liao, Y. Y.; Trapella, Claudio; Chiou, L. C. file con accesso da definire
Synthesis and Biological Activity of Human Neuropeptide S Analogues Modified in Position 5: Identification of Potent and Pure Neuropeptide S Receptor Antagonists. 2009 Guerrini, Remo; Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Rizzi, Anna; Ruzza, Chiara;... Fiorini, Stella; Marzola, Erika; R. K., Reinscheid; Regoli, Domenico; Salvadori, Severo file con accesso da definire
Influence of the Side Chain Next to C-Terminal Benzimidazole in Opioid Pseudopeptides Containing the Dmt-Tic Pharmacophore 2009 G., Balboni; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, ...Severo file con accesso da definire
First Application of the IART Approach with a new Re-188 Labeled Biotin-Derivative 2009 Duatti, Adriano; Pasquali, Micol; Trapella, Claudio; Guerrini, Remo; Boschi, Alessandra; Uccelli,... Licia; E., Janevik Ivanovska
Further studies on the pharmacological features of the nociceptin/orphanin FQ receptor ligand ZP120 2009 Fischetti, Carmela; Rizzi, Anna; E. C., Gavioli; Marzola, Giuliano; Trapella, Claudio; Guerrini, ...Remo; J. S., Petersen; Calo', Girolamo file con accesso da definire
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Galpha(qi5). 2009 Camarda, Valeria; Fischetti, Carmela; N., Anzellotti; P., Molinari; C., Ambrosio; E., Kostenis; R...egoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo file con accesso da definire
Structure-activity relationship study on Tyr9 of urotensin-II(4-11): identification of a partial agonist of the UT receptor. 2009 Batuwangala, Madura Suharshana; Camarda, Valeria; Mcdonald, J; Marzola, Erika; Lambert, Dg; Ng, L...l; Calo', Girolamo; Regoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo file con accesso da definire
Pharmacological profile and antiparkinsonian properties of the novel nociceptin/orphanin FQ receptor antagonist 1-[1-Cyclooctylmethyl-5-(1-hydroxy-1-methyl-ethyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-3-ethyl-1,3-dihydro-benzoimidazol-2-one (GF-4). 2010 Volta, Mattia; Marti, Matteo; Mcdonald, J.; Molinari, Stefano; Camarda, Valeria; Pelà, M.; Trapel...la, Claudio; Morari, Michele file con accesso da definire
Further studies on the pharmacological profile of the neuropeptide S receptor antagonist SHA 68. 2010 Ruzza, Chiara; Rizzi, Anna; Trapella, Claudio; Pela', Michela; Camarda, Valeria; Ruggieri, V.; Fi...laferro, M.; Cifani, C.; Reinscheid, R. K.; Vitale, G.; Ciccocioppo, R.; Salvadori, Severo; Guerrini, Remo; Calo', Girolamo file con accesso da definire
Might Re-188 be more effective for boosting therapy of breast cancer using the IART approach? 2010 Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Lic...ia; Duatti, Adriano file con accesso da definire
Mastering chiral substituted 2-oxopiperazines 2010 DE RISI, Carmela; Pela', Michela; Pollini, Gian Piero; Trapella, Claudio; Zanirato, Vinicio file con accesso da definire
Modulation of Silent and Constitutively Active Nociceptin/Orphanin FQ Receptors by Potent Receptor Antagonists and Na+ Ions in Rat Sympathetic Neurons. 2010 Mahmoud, S.; Margas, W.; Trapella, Claudio; Calo', Girolamo; Ruiz Velasco, V. file con accesso da definire
Evolution of the bifunctional lead μ agonist/δ Antagonist containing the 2′,6′-dimethyl- l -tyrosine-1,2,3,4- tetrahydroisoquinoline-3-carboxylic acid (Dmt-Tic) opioid pharmacophore 2010 Balboni, G; Salvadori, Severo; Trapella, Claudio; Knapp, Bi; Bidlack, Jm; Lazarus, Lh; Peng, X; N...eumeyer, J. L. file con accesso da definire
Synthesis and proteasome inhibition of N-allyl vinyl ester-based peptides 2010 Baldisserotto, Anna; Franceschini, Christian; Scalambra, Franco; Trapella, Claudio; Marastoni, Ma...uro; Sforza, Fabio; Gavioli, Riccardo; Tomatis, Roberto file con accesso da definire
The IART approach: new Re-188 nitrido biotinilated radiopharmaceuticals useful for cancer therapy 2011 Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Lic...ia; S., Papi; M., Chinol; Giganti, Melchiore; Duatti, Adriano file con accesso da definire
Synthesis and separation of the enantiomers of the neuropeptide S receptor antagonist (9R/S)-3-oxo-1,1-diphenyl-tetrahydro-oxazolo[3,4-a]pyrazine-7-carboxylic acid 4-fluoro-benzylamide (SHA 68). 2011 Trapella, Claudio; Pela', Michela; DEL ZOPPO, Luisa; Calo', Girolamo; Camarda, Valeria; Ruzza, Ch...iara; Cavazzini, Alberto; Costa, Valentina; Bertolasi, Valerio; Reinscheid, R. K.; Salvadori, Severo; Guerrini, Remo file con accesso da definire
Dopamine-nociceptin/orphanin FQ interactions in the substantia nigra reticulata of hemiparkinsonian rats: Involvement of D2/D3 receptors and impact on nigro-thalamic neurons and motor activity 2011 Volta, Mattia; Viaro, Riccardo; Trapella, Claudio; Marti, Matteo; Morari, Michele file con accesso da definire
Synthesis of folic conjugated LR octapeptide 2012 Pela', Michela; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Gaetano, Marverti; Silvia, ...Pirondi; Rosaria, Luciani; Maria Paola, Costi file con accesso da definire
A linear allergic contact dermatitis to p-tert-butylphenol formaldehyde resin sectorially present in a neoprene orthopedic brace: role of spectroscopy 2012 Corazza, Monica; S., Zauli; Bernardi, Tatiana; Trapella, Claudio; Benetti, Simonetta; Virgili, Anna file con accesso da definire
Mostrati risultati da 41 a 60 di 156
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