Sfoglia per Autore
Structure-activity studies on the nociceptin/orphanin FQ receptor antagonist 1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4'-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide.
file con accesso da definire2009 Trapella, Claudio; Fischetti, Carmela; Pela', Michela; Lazzari, Ilaria; Guerrini, Remo; Calo', Girolamo; Rizzi, Anna; Camarda, Valeria; Lambert, Dg; Mcdonald, J; Regoli, Domenico; Salvadori, Severo
1-Benzyl-N-[3-[spiroisobenzofuran-1(3H),4′-piperidin-1-yl]propyl]pyrrolidine-2-carboxamide (Compound 24) antagonizes NOP receptor-mediated potassium channel activation in rat periaqueductal gray slices
file con accesso da definire2009 Liao, Y. Y.; Trapella, Claudio; Chiou, L. C.
Synthesis and Biological Activity of Human Neuropeptide S Analogues Modified in Position 5: Identification of Potent and Pure Neuropeptide S Receptor Antagonists.
file con accesso da definire2009 Guerrini, Remo; Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Rizzi, Anna; Ruzza, Chiara; Fiorini, Stella; Marzola, Erika; R. K., Reinscheid; Regoli, Domenico; Salvadori, Severo
Influence of the Side Chain Next to C-Terminal Benzimidazole in Opioid Pseudopeptides Containing the Dmt-Tic Pharmacophore
file con accesso da definire2009 G., Balboni; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, Severo
First Application of the IART Approach with a new Re-188 Labeled Biotin-Derivative
2009 Duatti, Adriano; Pasquali, Micol; Trapella, Claudio; Guerrini, Remo; Boschi, Alessandra; Uccelli, Licia; E., Janevik Ivanovska
Further studies on the pharmacological features of the nociceptin/orphanin FQ receptor ligand ZP120
file con accesso da definire2009 Fischetti, Carmela; Rizzi, Anna; E. C., Gavioli; Marzola, Giuliano; Trapella, Claudio; Guerrini, Remo; J. S., Petersen; Calo', Girolamo
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Galpha(qi5).
file con accesso da definire2009 Camarda, Valeria; Fischetti, Carmela; N., Anzellotti; P., Molinari; C., Ambrosio; E., Kostenis; Regoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo
Structure-activity relationship study on Tyr9 of urotensin-II(4-11): identification of a partial agonist of the UT receptor.
file con accesso da definire2009 Batuwangala, Madura Suharshana; Camarda, Valeria; Mcdonald, J; Marzola, Erika; Lambert, Dg; Ng, Ll; Calo', Girolamo; Regoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo
Pharmacological profile and antiparkinsonian properties of the novel nociceptin/orphanin FQ receptor antagonist 1-[1-Cyclooctylmethyl-5-(1-hydroxy-1-methyl-ethyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-3-ethyl-1,3-dihydro-benzoimidazol-2-one (GF-4).
file con accesso da definire2010 Volta, Mattia; Marti, Matteo; Mcdonald, J.; Molinari, Stefano; Camarda, Valeria; Pelà, M.; Trapella, Claudio; Morari, Michele
Further studies on the pharmacological profile of the neuropeptide S receptor antagonist SHA 68.
file con accesso da definire2010 Ruzza, Chiara; Rizzi, Anna; Trapella, Claudio; Pela', Michela; Camarda, Valeria; Ruggieri, V.; Filaferro, M.; Cifani, C.; Reinscheid, R. K.; Vitale, G.; Ciccocioppo, R.; Salvadori, Severo; Guerrini, Remo; Calo', Girolamo
Might Re-188 be more effective for boosting therapy of breast cancer using the IART approach?
file con accesso da definire2010 Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Licia; Duatti, Adriano
Mastering chiral substituted 2-oxopiperazines
file con accesso da definire2010 DE RISI, Carmela; Pela', Michela; Pollini, Gian Piero; Trapella, Claudio; Zanirato, Vinicio
Modulation of Silent and Constitutively Active Nociceptin/Orphanin FQ Receptors by Potent Receptor Antagonists and Na+ Ions in Rat Sympathetic Neurons.
file con accesso da definire2010 Mahmoud, S.; Margas, W.; Trapella, Claudio; Calo', Girolamo; Ruiz Velasco, V.
Evolution of the bifunctional lead μ agonist/δ Antagonist containing the 2′,6′-dimethyl- l -tyrosine-1,2,3,4- tetrahydroisoquinoline-3-carboxylic acid (Dmt-Tic) opioid pharmacophore
file con accesso da definire2010 Balboni, G; Salvadori, Severo; Trapella, Claudio; Knapp, Bi; Bidlack, Jm; Lazarus, Lh; Peng, X; Neumeyer, J. L.
Synthesis and proteasome inhibition of N-allyl vinyl ester-based peptides
file con accesso da definire2010 Baldisserotto, Anna; Franceschini, Christian; Scalambra, Franco; Trapella, Claudio; Marastoni, Mauro; Sforza, Fabio; Gavioli, Riccardo; Tomatis, Roberto
The IART approach: new Re-188 nitrido biotinilated radiopharmaceuticals useful for cancer therapy
file con accesso da definire2011 Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Licia; S., Papi; M., Chinol; Giganti, Melchiore; Duatti, Adriano
Synthesis and separation of the enantiomers of the neuropeptide S receptor antagonist (9R/S)-3-oxo-1,1-diphenyl-tetrahydro-oxazolo[3,4-a]pyrazine-7-carboxylic acid 4-fluoro-benzylamide (SHA 68).
file con accesso da definire2011 Trapella, Claudio; Pela', Michela; DEL ZOPPO, Luisa; Calo', Girolamo; Camarda, Valeria; Ruzza, Chiara; Cavazzini, Alberto; Costa, Valentina; Bertolasi, Valerio; Reinscheid, R. K.; Salvadori, Severo; Guerrini, Remo
Dopamine-nociceptin/orphanin FQ interactions in the substantia nigra reticulata of hemiparkinsonian rats: Involvement of D2/D3 receptors and impact on nigro-thalamic neurons and motor activity
file con accesso da definire2011 Volta, Mattia; Viaro, Riccardo; Trapella, Claudio; Marti, Matteo; Morari, Michele
Synthesis of folic conjugated LR octapeptide
file con accesso da definire2012 Pela', Michela; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Gaetano, Marverti; Silvia, Pirondi; Rosaria, Luciani; Maria Paola, Costi
A linear allergic contact dermatitis to p-tert-butylphenol formaldehyde resin sectorially present in a neoprene orthopedic brace: role of spectroscopy
file con accesso da definire2012 Corazza, Monica; S., Zauli; Bernardi, Tatiana; Trapella, Claudio; Benetti, Simonetta; Virgili, Anna
Titolo | Data di pubblicazione | Autore(i) | File |
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Structure-activity studies on the nociceptin/orphanin FQ receptor antagonist 1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4'-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide. | 2009 | Trapella, Claudio; Fischetti, Carmela; Pela', Michela; Lazzari, Ilaria; Guerrini, Remo; Calo', Gi...rolamo; Rizzi, Anna; Camarda, Valeria; Lambert, Dg; Mcdonald, J; Regoli, Domenico; Salvadori, Severo | file con accesso da definire |
1-Benzyl-N-[3-[spiroisobenzofuran-1(3H),4′-piperidin-1-yl]propyl]pyrrolidine-2-carboxamide (Compound 24) antagonizes NOP receptor-mediated potassium channel activation in rat periaqueductal gray slices | 2009 | Liao, Y. Y.; Trapella, Claudio; Chiou, L. C. | file con accesso da definire |
Synthesis and Biological Activity of Human Neuropeptide S Analogues Modified in Position 5: Identification of Potent and Pure Neuropeptide S Receptor Antagonists. | 2009 | Guerrini, Remo; Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Rizzi, Anna; Ruzza, Chiara;... Fiorini, Stella; Marzola, Erika; R. K., Reinscheid; Regoli, Domenico; Salvadori, Severo | file con accesso da definire |
Influence of the Side Chain Next to C-Terminal Benzimidazole in Opioid Pseudopeptides Containing the Dmt-Tic Pharmacophore | 2009 | G., Balboni; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, ...Severo | file con accesso da definire |
First Application of the IART Approach with a new Re-188 Labeled Biotin-Derivative | 2009 | Duatti, Adriano; Pasquali, Micol; Trapella, Claudio; Guerrini, Remo; Boschi, Alessandra; Uccelli,... Licia; E., Janevik Ivanovska | |
Further studies on the pharmacological features of the nociceptin/orphanin FQ receptor ligand ZP120 | 2009 | Fischetti, Carmela; Rizzi, Anna; E. C., Gavioli; Marzola, Giuliano; Trapella, Claudio; Guerrini, ...Remo; J. S., Petersen; Calo', Girolamo | file con accesso da definire |
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Galpha(qi5). | 2009 | Camarda, Valeria; Fischetti, Carmela; N., Anzellotti; P., Molinari; C., Ambrosio; E., Kostenis; R...egoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo | file con accesso da definire |
Structure-activity relationship study on Tyr9 of urotensin-II(4-11): identification of a partial agonist of the UT receptor. | 2009 | Batuwangala, Madura Suharshana; Camarda, Valeria; Mcdonald, J; Marzola, Erika; Lambert, Dg; Ng, L...l; Calo', Girolamo; Regoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo | file con accesso da definire |
Pharmacological profile and antiparkinsonian properties of the novel nociceptin/orphanin FQ receptor antagonist 1-[1-Cyclooctylmethyl-5-(1-hydroxy-1-methyl-ethyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-3-ethyl-1,3-dihydro-benzoimidazol-2-one (GF-4). | 2010 | Volta, Mattia; Marti, Matteo; Mcdonald, J.; Molinari, Stefano; Camarda, Valeria; Pelà, M.; Trapel...la, Claudio; Morari, Michele | file con accesso da definire |
Further studies on the pharmacological profile of the neuropeptide S receptor antagonist SHA 68. | 2010 | Ruzza, Chiara; Rizzi, Anna; Trapella, Claudio; Pela', Michela; Camarda, Valeria; Ruggieri, V.; Fi...laferro, M.; Cifani, C.; Reinscheid, R. K.; Vitale, G.; Ciccocioppo, R.; Salvadori, Severo; Guerrini, Remo; Calo', Girolamo | file con accesso da definire |
Might Re-188 be more effective for boosting therapy of breast cancer using the IART approach? | 2010 | Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Lic...ia; Duatti, Adriano | file con accesso da definire |
Mastering chiral substituted 2-oxopiperazines | 2010 | DE RISI, Carmela; Pela', Michela; Pollini, Gian Piero; Trapella, Claudio; Zanirato, Vinicio | file con accesso da definire |
Modulation of Silent and Constitutively Active Nociceptin/Orphanin FQ Receptors by Potent Receptor Antagonists and Na+ Ions in Rat Sympathetic Neurons. | 2010 | Mahmoud, S.; Margas, W.; Trapella, Claudio; Calo', Girolamo; Ruiz Velasco, V. | file con accesso da definire |
Evolution of the bifunctional lead μ agonist/δ Antagonist containing the 2′,6′-dimethyl- l -tyrosine-1,2,3,4- tetrahydroisoquinoline-3-carboxylic acid (Dmt-Tic) opioid pharmacophore | 2010 | Balboni, G; Salvadori, Severo; Trapella, Claudio; Knapp, Bi; Bidlack, Jm; Lazarus, Lh; Peng, X; N...eumeyer, J. L. | file con accesso da definire |
Synthesis and proteasome inhibition of N-allyl vinyl ester-based peptides | 2010 | Baldisserotto, Anna; Franceschini, Christian; Scalambra, Franco; Trapella, Claudio; Marastoni, Ma...uro; Sforza, Fabio; Gavioli, Riccardo; Tomatis, Roberto | file con accesso da definire |
The IART approach: new Re-188 nitrido biotinilated radiopharmaceuticals useful for cancer therapy | 2011 | Boschi, Alessandra; Pasquali, Micol; E., Janevik; Guerrini, Remo; Trapella, Claudio; Uccelli, Lic...ia; S., Papi; M., Chinol; Giganti, Melchiore; Duatti, Adriano | file con accesso da definire |
Synthesis and separation of the enantiomers of the neuropeptide S receptor antagonist (9R/S)-3-oxo-1,1-diphenyl-tetrahydro-oxazolo[3,4-a]pyrazine-7-carboxylic acid 4-fluoro-benzylamide (SHA 68). | 2011 | Trapella, Claudio; Pela', Michela; DEL ZOPPO, Luisa; Calo', Girolamo; Camarda, Valeria; Ruzza, Ch...iara; Cavazzini, Alberto; Costa, Valentina; Bertolasi, Valerio; Reinscheid, R. K.; Salvadori, Severo; Guerrini, Remo | file con accesso da definire |
Dopamine-nociceptin/orphanin FQ interactions in the substantia nigra reticulata of hemiparkinsonian rats: Involvement of D2/D3 receptors and impact on nigro-thalamic neurons and motor activity | 2011 | Volta, Mattia; Viaro, Riccardo; Trapella, Claudio; Marti, Matteo; Morari, Michele | file con accesso da definire |
Synthesis of folic conjugated LR octapeptide | 2012 | Pela', Michela; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Gaetano, Marverti; Silvia, ...Pirondi; Rosaria, Luciani; Maria Paola, Costi | file con accesso da definire |
A linear allergic contact dermatitis to p-tert-butylphenol formaldehyde resin sectorially present in a neoprene orthopedic brace: role of spectroscopy | 2012 | Corazza, Monica; S., Zauli; Bernardi, Tatiana; Trapella, Claudio; Benetti, Simonetta; Virgili, Anna | file con accesso da definire |
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