Sfoglia per Autore
Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore
file con accesso da definire2007 Balboni, G; Onnis, V; Congiu, C; Zotti, M; Sasaki, Y; Ambo, A; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh; Lazzari, Ilaria; Trapella, Claudio; Salvadori, Severo
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl] methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vitro studies
file con accesso da definire2007 Spagnolo, Barbara; Carra', Giacomo; Fantin, Martina; Fischetti, Carmela; Hebbes, C; Mcdonald, J; Barnes, Ta; Rizzi, Anna; Trapella, Claudio; Fanton, Giulia; Morari, Michele; Lambert, Dg; Regoli, Domenico; Calo', Girolamo
The nociceptin/orphanin FQ receptor antagonist J-113397 and L-DOPA additively attenuate experimental parkinsonism through overinhibition of the nigrothalamic pathway
file con accesso da definire2007 Marti, Matteo; Trapella, Claudio; Viaro, Riccardo; Morari, Michele
Nocistatin inhibits 5-hydroxytryptamine release in the mouse neocortex via presynaptic G i/o protein linked pathways
file con accesso da definire2007 Fantin, Martina; Fischetti, Carmela; Trapella, Claudio; Morari, Michele
Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with C alpha,alpha-dialkylated amino acids
2007 Arduin, Marika; Spagnolo, Barbara; Calo', Girolamo; Guerrini, Remo; Carra', Giacomo; Fischetti, Carmela; Trapella, Claudio; Marzola, Erika; Mcdonald, J; Lambert, Dg; Regoli, Domenico; Salvadori, Severo
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8 ,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vivo studies
file con accesso da definire2007 Rizzi, Anna; Gavioli, Elaine Cristina; Marzola, Giuliano; Spagnolo, Barbara; Zucchini, Silvia; Ciccocioppo, R; Trapella, Claudio; Regoli, Domenico; Calo', Girolamo
The novel nociceptin/orphanin FQ receptor antagonist Trap-101 alleviates experimental parkinsonism through inhibition of the nigro-thalamic pathway. Positive interaction with L-DOPA
file con accesso da definire2008 Marti, Matteo; Trapella, Claudio; Morari, Michele
Nociceptin/orphanin FQ receptor blockade attenuates MPTP-induced parkinsonism
file con accesso da definire2008 Viaro, Riccardo; Sanchez Pernaute, R.; Marti, Matteo; Trapella, Claudio; Isacson, O.; Morari, Michele
Role of benzimidazole (Bid) in the d-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH2-Bid (UFP-502)
file con accesso da definire2008 Salvadori, Severo; Fiorini, S.; Trapella, Claudio; Porreca, F.; Davis, P.; Sasaki, Y.; Ambo, A.; Marczak, E. D.; Lazarus, L. H.; Balboni, G.
Structure-activity study at positions 3 and 4 of human neuropeptide S.
file con accesso da definire2008 Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Guerrini, Remo; Rizzi, Anna; Ruzza, Chiara; Fiorini, Stella; Marzola, Erika; R. K., Reinscheid; Regoli, Domenico; Salvadori, Severo
Triazine Compounds as Antagonists at Bv8-Prokineticin Receptors
file con accesso da definire2008 Balboni, G.; Lazzari, I.; Trapella, Claudio; Negri, L.; Lattanzi, R.; Giannini, E.; Nicotra, A.; Melchiorri, P.; Visentin, S.; Nuccio, C. D.; Salvadori, Severo
C-terminal constrained phenylalanine as a pharmacophoric unit in peptide-based proteasome inhibitors
file con accesso da definire2008 Baldisserotto, Anna; Marastoni, Mauro; Lazzari, Ilaria; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto
Further studies on lead compounds containing the opioid pharmacophore Dmt-Tic.
file con accesso da definire2008 G., Balboni; Fiorini, Stella; Baldisserotto, Anna; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, Severo
Recent advances in the stereoselective synthesis of trans-3,4- disubstituted-piperidines: applications to (-)paroxetine
file con accesso da definire2008 DE RISI, Carmela; Fanton, Giulia; G. P., Pollini; Trapella, Claudio; Valente, Filippo; Zanirato, Vinicio
Anxiolytic- and antidepressant-like activities of H-Dmt-Tic-NH-CH(CH2-COOH)-Bid (UFP-512), a novel selective delta opioid receptor agonist
file con accesso da definire2008 Vergura, Raffaella; G., Balboni; Spagnolo, Barbara; Gavioli, Elaine Cristina; D. G., Lambert; J., Mcdonald; Trapella, Claudio; L. H., Lazarus; Regoli, Domenico; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo
Structure-activity relationship study of position 4 in the urotensin-II receptor ligand U-II(4-11)
file con accesso da definire2008 Marzola, Erika; Camarda, Valeria; Batuwangala, Madura Suharshana; Lamberti, Dg; Calo', Girolamo; Guerrini, Remo; Trapella, Claudio; Regoli, Domenico; Tomatis, Roberto; Salvadori, Severo
Synthesis and biological activity of human neuropeptide S analogues modified in position 2
file con accesso da definire2008 Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Guerrini, Remo; Rizzi, Anna; Ruzza, Chiara; Fiorini, Stella; Marzola, Erika; Reinscheid, R. K.; Regoli, Domenico; Salvadori, Severo
First Application of the IART Approach with a new Re-188 Labeled Biotin-Derivative
2009 Duatti, Adriano; Pasquali, Micol; Trapella, Claudio; Guerrini, Remo; Boschi, Alessandra; Uccelli, Licia; E., Janevik Ivanovska
Influence of the Side Chain Next to C-Terminal Benzimidazole in Opioid Pseudopeptides Containing the Dmt-Tic Pharmacophore
file con accesso da definire2009 G., Balboni; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, Severo
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Galpha(qi5).
file con accesso da definire2009 Camarda, Valeria; Fischetti, Carmela; N., Anzellotti; P., Molinari; C., Ambrosio; E., Kostenis; Regoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore | 2007 | Balboni, G; Onnis, V; Congiu, C; Zotti, M; Sasaki, Y; Ambo, A; Bryant, Sd; Jinsmaa, Y; Lazarus, L...h; Lazzari, Ilaria; Trapella, Claudio; Salvadori, Severo | file con accesso da definire |
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl] methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vitro studies | 2007 | Spagnolo, Barbara; Carra', Giacomo; Fantin, Martina; Fischetti, Carmela; Hebbes, C; Mcdonald, J; ...Barnes, Ta; Rizzi, Anna; Trapella, Claudio; Fanton, Giulia; Morari, Michele; Lambert, Dg; Regoli, Domenico; Calo', Girolamo | file con accesso da definire |
The nociceptin/orphanin FQ receptor antagonist J-113397 and L-DOPA additively attenuate experimental parkinsonism through overinhibition of the nigrothalamic pathway | 2007 | Marti, Matteo; Trapella, Claudio; Viaro, Riccardo; Morari, Michele | file con accesso da definire |
Nocistatin inhibits 5-hydroxytryptamine release in the mouse neocortex via presynaptic G i/o protein linked pathways | 2007 | Fantin, Martina; Fischetti, Carmela; Trapella, Claudio; Morari, Michele | file con accesso da definire |
Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with C alpha,alpha-dialkylated amino acids | 2007 | Arduin, Marika; Spagnolo, Barbara; Calo', Girolamo; Guerrini, Remo; Carra', Giacomo; Fischetti, C...armela; Trapella, Claudio; Marzola, Erika; Mcdonald, J; Lambert, Dg; Regoli, Domenico; Salvadori, Severo | |
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8 ,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vivo studies | 2007 | Rizzi, Anna; Gavioli, Elaine Cristina; Marzola, Giuliano; Spagnolo, Barbara; Zucchini, Silvia; Ci...ccocioppo, R; Trapella, Claudio; Regoli, Domenico; Calo', Girolamo | file con accesso da definire |
The novel nociceptin/orphanin FQ receptor antagonist Trap-101 alleviates experimental parkinsonism through inhibition of the nigro-thalamic pathway. Positive interaction with L-DOPA | 2008 | Marti, Matteo; Trapella, Claudio; Morari, Michele | file con accesso da definire |
Nociceptin/orphanin FQ receptor blockade attenuates MPTP-induced parkinsonism | 2008 | Viaro, Riccardo; Sanchez Pernaute, R.; Marti, Matteo; Trapella, Claudio; Isacson, O.; Morari, Mic...hele | file con accesso da definire |
Role of benzimidazole (Bid) in the d-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH2-Bid (UFP-502) | 2008 | Salvadori, Severo; Fiorini, S.; Trapella, Claudio; Porreca, F.; Davis, P.; Sasaki, Y.; Ambo, A.; ...Marczak, E. D.; Lazarus, L. H.; Balboni, G. | file con accesso da definire |
Structure-activity study at positions 3 and 4 of human neuropeptide S. | 2008 | Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Guerrini, Remo; Rizzi, Anna; Ruzza, Chiara;... Fiorini, Stella; Marzola, Erika; R. K., Reinscheid; Regoli, Domenico; Salvadori, Severo | file con accesso da definire |
Triazine Compounds as Antagonists at Bv8-Prokineticin Receptors | 2008 | Balboni, G.; Lazzari, I.; Trapella, Claudio; Negri, L.; Lattanzi, R.; Giannini, E.; Nicotra, A.; ...Melchiorri, P.; Visentin, S.; Nuccio, C. D.; Salvadori, Severo | file con accesso da definire |
C-terminal constrained phenylalanine as a pharmacophoric unit in peptide-based proteasome inhibitors | 2008 | Baldisserotto, Anna; Marastoni, Mauro; Lazzari, Ilaria; Trapella, Claudio; Gavioli, Riccardo; Tom...atis, Roberto | file con accesso da definire |
Further studies on lead compounds containing the opioid pharmacophore Dmt-Tic. | 2008 | G., Balboni; Fiorini, Stella; Baldisserotto, Anna; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D...., Marczak; L. H., Lazarus; Salvadori, Severo | file con accesso da definire |
Recent advances in the stereoselective synthesis of trans-3,4- disubstituted-piperidines: applications to (-)paroxetine | 2008 | DE RISI, Carmela; Fanton, Giulia; G. P., Pollini; Trapella, Claudio; Valente, Filippo; Zanirato, ...Vinicio | file con accesso da definire |
Anxiolytic- and antidepressant-like activities of H-Dmt-Tic-NH-CH(CH2-COOH)-Bid (UFP-512), a novel selective delta opioid receptor agonist | 2008 | Vergura, Raffaella; G., Balboni; Spagnolo, Barbara; Gavioli, Elaine Cristina; D. G., Lambert; J.,... Mcdonald; Trapella, Claudio; L. H., Lazarus; Regoli, Domenico; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo | file con accesso da definire |
Structure-activity relationship study of position 4 in the urotensin-II receptor ligand U-II(4-11) | 2008 | Marzola, Erika; Camarda, Valeria; Batuwangala, Madura Suharshana; Lamberti, Dg; Calo', Girolamo; ...Guerrini, Remo; Trapella, Claudio; Regoli, Domenico; Tomatis, Roberto; Salvadori, Severo | file con accesso da definire |
Synthesis and biological activity of human neuropeptide S analogues modified in position 2 | 2008 | Camarda, Valeria; Trapella, Claudio; Calo', Girolamo; Guerrini, Remo; Rizzi, Anna; Ruzza, Chiara;... Fiorini, Stella; Marzola, Erika; Reinscheid, R. K.; Regoli, Domenico; Salvadori, Severo | file con accesso da definire |
First Application of the IART Approach with a new Re-188 Labeled Biotin-Derivative | 2009 | Duatti, Adriano; Pasquali, Micol; Trapella, Claudio; Guerrini, Remo; Boschi, Alessandra; Uccelli,... Licia; E., Janevik Ivanovska | |
Influence of the Side Chain Next to C-Terminal Benzimidazole in Opioid Pseudopeptides Containing the Dmt-Tic Pharmacophore | 2009 | G., Balboni; Trapella, Claudio; Y., Sasaki; A., Ambo; E. D., Marczak; L. H., Lazarus; Salvadori, ...Severo | file con accesso da definire |
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Galpha(qi5). | 2009 | Camarda, Valeria; Fischetti, Carmela; N., Anzellotti; P., Molinari; C., Ambrosio; E., Kostenis; R...egoli, Domenico; Trapella, Claudio; Guerrini, Remo; Salvadori, Severo; Calo', Girolamo | file con accesso da definire |
Legenda icone
- file ad accesso aperto
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile