Sfoglia per Autore
A new synthetic approach to 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidyl]-3-ethyl-1,3-dihydro-benzimidazol-2-one (J-113397), the first non-peptide ORL-1 receptor antagonist
file con accesso da definire2001 DE RISI, Carmela; Pollini, Gian Piero; Trapella, Claudio; Peretto, I.; Ronzoni, S.; Giardina, G. A. M.
A Convenient Route to Enantiomerically Pure 2-Substituted Methyl Glycerate Derivatives
file con accesso da definire2003 Ley, S. V.; Trapella, Claudio; Michel, P.
Identificazione di un antagonista del recettore NOP a struttura 1,2,3,6-tetraidropiridinica.
file con accesso da definire2004 Trapella, Claudio; Guerrini, Remo; Calo', Girolamo; Regoli, Domenico; Salvadori, Severo
Pharmacological profile of nociceptin/orphanin FQ receptors regulating 5-hydroxytryptamine release in the mouse neocortex
file con accesso da definire2004 Mela, Flora; Marti, Matteo; Ulazzi, L; Vaccari, E; Zucchini, Silvia; Trapella, Claudio; Salvadori, Severo; Beani, Lorenzo; Bianchi, Clementina; Morari, Michele
Nonpeptide/peptide chimeric ligands for the nociceptin/orphanin FQ receptor: design, synthesis and in vitro pharmacological activity
file con accesso da definire2004 Guerrini, Remo; Carra', G; Calo', Girolamo; Trapella, Claudio; Marzola, Erika; Rizzi, D; Regoli, D; Salvadori, Severo
HIV protease inhibitors: synthesis and activity of N-aryl-N '-hydroxyalkyl hydrazide pseudopeptides
file con accesso da definire2005 Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Mcdonald, J; Bortolotti, Fabrizio; Tomatis, Roberto
N- and C-terminal modifications of nociceptin/orphanin FQ generate highly potent NOP receptor ligands
2005 Guerrini, Remo; Calo', Girolamo; Lambert, Dg; Carra', Giacomo; Arduin, Marika; Barnes, Ta; Mcdonald, J; Rizzi, Daniela; Trapella, Claudio; Marzola, Erika; Rowbotham, Dj; Regoli, Domenico; Salvadori, Severo
Tryptophan replacement in the nociceptin/orphanin FQ receptor ligand Ac-RYYRWK-NH2
2005 Carra', Giacomo; Calo', Girolamo; Spagnolo, Barbara; Guerrini, Remo; Arduin, Marika; Marzola, Erika; Trapella, Claudio; Regoli, Domenico; Salvadori, Severo
New 2 ',6 '-dimethyl-L-tyrosine (Dmt) opioid peptidomimetics based on the Aba-Gly scaffold. Development of unique mu-opioid receptor ligands
file con accesso da definire2006 Ballet, S; Salvadori, Severo; Trapella, Claudio; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh; Negri, L; Giannini, E; Lattanzi, R; Tourwe, D; Balboni, G.
6-N,N-dimethylamino-2,3-naphthalimide: A new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides
file con accesso da definire2006 Vazquez, Me; Blanco, Jb; Salvadori, Severo; Trapella, Claudio; Argazzi, Roberto; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh; Negri, L; Giannini, E; Lattanzi, R; Colucci, M; Balboni, G.
Structure-activity studies on neuropeptide S - Identification of the amino acid residues crucial for receptor activation
file con accesso da definire2006 Roth, Al; Marzola, Erika; Rizzi, Anna; Arduin, Marika; Trapella, Claudio; Corti, C; Vergura, Raffaella; Martinelli, P; Salvadori, Severo; Regoli, Domenico; Corsi, M; Cavanni, P; Calo', Girolamo; Guerrini, Remo
Identification of an achiral analogue of J-113397 as potent nociceptin/orphanin FQ receptor antagonist
2006 Trapella, Claudio; Guerrini, Remo; Piccagli, Laura; Calo', Girolamo; Carra', Giacomo; Spagnolo, Barbara; Rubini, S; Fanton, Giulia; Hebbes, C; Mcdonald, J; Lambert, Dg; Regoli, Domenico; Salvadori, Severo
Anxiolytic and antidepressant-like activities of UFP-512, a novel selective delta opiold receptor agonist
file con accesso da definire2006 Vergura, Raffaella; Balboni, G; Spagnolo, Barbara; Gavioli, Elaine Cristina; Lambert, Dg; Mcdonald, J; Trapella, Claudio; Regoli, Domenico; Salvadori, Severo; Calo', Girolamo
Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore
file con accesso da definire2006 Balboni, G; Onnis, V; Congiu, C; Zotti, M; Sasaki, Y; Ambo, A; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh; Trapella, Claudio; Salvadori, Severo
P3 and P4 position analysis of vinyl ester pseudopeptide proteasome inhibitors
file con accesso da definire2006 Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto
New opioid designed multiple ligand from Dmt-Tic and morphinan pharmacophores
file con accesso da definire2006 Neumeyer, Jl; Peng, Xm; Knapp, Bi; Bidlack, Jm; Lazarus, Lh; Salvadori, Severo; Trapella, Claudio; Balboni, G.
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors
file con accesso da definire2006 Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto
Endogenous nociceptin/orphanin FQ signalling produces opposite spinal antinociceptive and supraspinal pronociceptive effects in the mouse formalin test: Pharmacological and genetic evidences
file con accesso da definire2006 Rizzi, Anna; Nazzaro, Cristiano; Marzola, Giuliano; Zucchini, Silvia; Trapella, Claudio; Guerrini, Remo; Zeilhofer, Hu; Regoli, Domenico; Calo', Girolamo
Nocistatin inhibits 5-hydroxytryptamine release in the mouse neocortex via presynaptic G i/o protein linked pathways
file con accesso da definire2007 Fantin, Martina; Fischetti, Carmela; Trapella, Claudio; Morari, Michele
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl] methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vitro studies
file con accesso da definire2007 Spagnolo, Barbara; Carra', Giacomo; Fantin, Martina; Fischetti, Carmela; Hebbes, C; Mcdonald, J; Barnes, Ta; Rizzi, Anna; Trapella, Claudio; Fanton, Giulia; Morari, Michele; Lambert, Dg; Regoli, Domenico; Calo', Girolamo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A new synthetic approach to 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidyl]-3-ethyl-1,3-dihydro-benzimidazol-2-one (J-113397), the first non-peptide ORL-1 receptor antagonist | 2001 | DE RISI, Carmela; Pollini, Gian Piero; Trapella, Claudio; Peretto, I.; Ronzoni, S.; Giardina, G. ...A. M. | file con accesso da definire |
A Convenient Route to Enantiomerically Pure 2-Substituted Methyl Glycerate Derivatives | 2003 | Ley, S. V.; Trapella, Claudio; Michel, P. | file con accesso da definire |
Identificazione di un antagonista del recettore NOP a struttura 1,2,3,6-tetraidropiridinica. | 2004 | Trapella, Claudio; Guerrini, Remo; Calo', Girolamo; Regoli, Domenico; Salvadori, Severo | file con accesso da definire |
Pharmacological profile of nociceptin/orphanin FQ receptors regulating 5-hydroxytryptamine release in the mouse neocortex | 2004 | Mela, Flora; Marti, Matteo; Ulazzi, L; Vaccari, E; Zucchini, Silvia; Trapella, Claudio; Salvadori..., Severo; Beani, Lorenzo; Bianchi, Clementina; Morari, Michele | file con accesso da definire |
Nonpeptide/peptide chimeric ligands for the nociceptin/orphanin FQ receptor: design, synthesis and in vitro pharmacological activity | 2004 | Guerrini, Remo; Carra', G; Calo', Girolamo; Trapella, Claudio; Marzola, Erika; Rizzi, D; Regoli, ...D; Salvadori, Severo | file con accesso da definire |
HIV protease inhibitors: synthesis and activity of N-aryl-N '-hydroxyalkyl hydrazide pseudopeptides | 2005 | Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Mcdonald, J; Bortolotti, Fabrizio; Toma...tis, Roberto | file con accesso da definire |
N- and C-terminal modifications of nociceptin/orphanin FQ generate highly potent NOP receptor ligands | 2005 | Guerrini, Remo; Calo', Girolamo; Lambert, Dg; Carra', Giacomo; Arduin, Marika; Barnes, Ta; Mcdona...ld, J; Rizzi, Daniela; Trapella, Claudio; Marzola, Erika; Rowbotham, Dj; Regoli, Domenico; Salvadori, Severo | |
Tryptophan replacement in the nociceptin/orphanin FQ receptor ligand Ac-RYYRWK-NH2 | 2005 | Carra', Giacomo; Calo', Girolamo; Spagnolo, Barbara; Guerrini, Remo; Arduin, Marika; Marzola, Eri...ka; Trapella, Claudio; Regoli, Domenico; Salvadori, Severo | |
New 2 ',6 '-dimethyl-L-tyrosine (Dmt) opioid peptidomimetics based on the Aba-Gly scaffold. Development of unique mu-opioid receptor ligands | 2006 | Ballet, S; Salvadori, Severo; Trapella, Claudio; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh; Negri, L; G...iannini, E; Lattanzi, R; Tourwe, D; Balboni, G. | file con accesso da definire |
6-N,N-dimethylamino-2,3-naphthalimide: A new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides | 2006 | Vazquez, Me; Blanco, Jb; Salvadori, Severo; Trapella, Claudio; Argazzi, Roberto; Bryant, Sd; Jins...maa, Y; Lazarus, Lh; Negri, L; Giannini, E; Lattanzi, R; Colucci, M; Balboni, G. | file con accesso da definire |
Structure-activity studies on neuropeptide S - Identification of the amino acid residues crucial for receptor activation | 2006 | Roth, Al; Marzola, Erika; Rizzi, Anna; Arduin, Marika; Trapella, Claudio; Corti, C; Vergura, Raff...aella; Martinelli, P; Salvadori, Severo; Regoli, Domenico; Corsi, M; Cavanni, P; Calo', Girolamo; Guerrini, Remo | file con accesso da definire |
Identification of an achiral analogue of J-113397 as potent nociceptin/orphanin FQ receptor antagonist | 2006 | Trapella, Claudio; Guerrini, Remo; Piccagli, Laura; Calo', Girolamo; Carra', Giacomo; Spagnolo, B...arbara; Rubini, S; Fanton, Giulia; Hebbes, C; Mcdonald, J; Lambert, Dg; Regoli, Domenico; Salvadori, Severo | |
Anxiolytic and antidepressant-like activities of UFP-512, a novel selective delta opiold receptor agonist | 2006 | Vergura, Raffaella; Balboni, G; Spagnolo, Barbara; Gavioli, Elaine Cristina; Lambert, Dg; Mcdonal...d, J; Trapella, Claudio; Regoli, Domenico; Salvadori, Severo; Calo', Girolamo | file con accesso da definire |
Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore | 2006 | Balboni, G; Onnis, V; Congiu, C; Zotti, M; Sasaki, Y; Ambo, A; Bryant, Sd; Jinsmaa, Y; Lazarus, L...h; Trapella, Claudio; Salvadori, Severo | file con accesso da definire |
P3 and P4 position analysis of vinyl ester pseudopeptide proteasome inhibitors | 2006 | Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto | file con accesso da definire |
New opioid designed multiple ligand from Dmt-Tic and morphinan pharmacophores | 2006 | Neumeyer, Jl; Peng, Xm; Knapp, Bi; Bidlack, Jm; Lazarus, Lh; Salvadori, Severo; Trapella, Claudio...; Balboni, G. | file con accesso da definire |
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors | 2006 | Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto | file con accesso da definire |
Endogenous nociceptin/orphanin FQ signalling produces opposite spinal antinociceptive and supraspinal pronociceptive effects in the mouse formalin test: Pharmacological and genetic evidences | 2006 | Rizzi, Anna; Nazzaro, Cristiano; Marzola, Giuliano; Zucchini, Silvia; Trapella, Claudio; Guerrini..., Remo; Zeilhofer, Hu; Regoli, Domenico; Calo', Girolamo | file con accesso da definire |
Nocistatin inhibits 5-hydroxytryptamine release in the mouse neocortex via presynaptic G i/o protein linked pathways | 2007 | Fantin, Martina; Fischetti, Carmela; Trapella, Claudio; Morari, Michele | file con accesso da definire |
Pharmacological characterization of the nociceptin/orphanin FQ receptor antagonist SB-612111 [(-)-cis-1-methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl] methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol]: In vitro studies | 2007 | Spagnolo, Barbara; Carra', Giacomo; Fantin, Martina; Fischetti, Carmela; Hebbes, C; Mcdonald, J; ...Barnes, Ta; Rizzi, Anna; Trapella, Claudio; Fanton, Giulia; Morari, Michele; Lambert, Dg; Regoli, Domenico; Calo', Girolamo | file con accesso da definire |
Legenda icone
- file ad accesso aperto
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile