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3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
5'-Phosphoramidates and 5'-diphosphates of 2'-O-allyl-β-D- arabinofuranosyl-uracil, -cytosine, and -adenine: Inhibition of ribonucleotide reductase
file con accesso da definire1999 Manfredini, Stefano; Baraldi, Pier Giovanni; Durini, Elisa; Vertuani, Silvia; Balzarini, Jan; DE CLERCQ, Erik; Karlsson, Anna; Buzzoni, Valentina; Thelander, Lars
5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists.
file con accesso da definire2006 Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G.
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility
file con accesso da definire2002 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation
2012 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1
file con accesso da definire2000 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Leoni, A; Bianchi, Nicoletta; Feriotto, Giordana; Rutigliano, C; Mischiati, Carlo; Gambari, Roberto
[3H]-MRE 2029-F20, a novel selective antagonist radioligand, for the pharmacological and biochemical characterization of A2B receptors.
file con accesso da definire2006 Gessi, Stefania; Varani, Katia; Merighi, Stefania; Cattabriga, Elena; Szabadkai, Y.; Rizzuto, Rosario; Klotz, K. N.; Leung, E.; Maclennan, S.; Baraldi, Pier Giovanni; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Bra...ncale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro | |
5'-Phosphoramidates and 5'-diphosphates of 2'-O-allyl-β-D- arabinofuranosyl-uracil, -cytosine, and -adenine: Inhibition of ribonucleotide reductase | 1999 | Manfredini, Stefano; Baraldi, Pier Giovanni; Durini, Elisa; Vertuani, Silvia; Balzarini, Jan; DE ...CLERCQ, Erik; Karlsson, Anna; Buzzoni, Valentina; Thelander, Lars | file con accesso da definire |
5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists. | 2006 | Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier ...Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G. | file con accesso da definire |
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility. | 2001 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility | 2002 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, ...E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility. | 2001 | Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation | 2012 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, S...tefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia | |
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding to transcription factor Sp1 | 2000 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Leoni, A; B...ianchi, Nicoletta; Feriotto, Giordana; Rutigliano, C; Mischiati, Carlo; Gambari, Roberto | file con accesso da definire |
[3H]-MRE 2029-F20, a novel selective antagonist radioligand, for the pharmacological and biochemical characterization of A2B receptors. | 2006 | Gessi, Stefania; Varani, Katia; Merighi, Stefania; Cattabriga, Elena; Szabadkai, Y.; Rizzuto, Ros...ario; Klotz, K. N.; Leung, E.; Maclennan, S.; Baraldi, Pier Giovanni; Borea, Pier Andrea | file con accesso da definire |
Legenda icone
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Opzioni
Scopri
Tipologia
- 03 Contributo in rivista (Pubblic... 356
- 03 Contributo in rivista (Pubblic... 356
- 04 Atto di Convegno (Proceedings) 67
- 04 Atto di Convegno (Proceedings)... 60
- 06 Brevetto 39
- 06 Brevetto::06.1 Brevetto 39
- 04 Atto di Convegno (Proceedings)... 7
- 02 Contributo in volume 4
- 02 Contributo in volume::02.1 Con... 4
Data di pubblicazione
- 2010 - 2019 73
- 2000 - 2009 238
- 1990 - 1999 94
- 1980 - 1989 51
- 1976 - 1979 10
Editore
- - 21
- American Chemical Society:1155 Si... 9
- -- 4
- Elsevier Science Limited:Oxford F... 4
- Società Italiana di Farmacologia 3
- Bentham Science Publishers BV:PO ... 2
- Georg Thieme Verlag Stuttgart:Pos... 2
- Purine 2
- Purines 2
- Springer 2
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 71
- BIOORGANIC & MEDICINAL CHEMISTRY ... 26
- SYNTHESIS 21
- IL FARMACO 15
- EUROPEAN JOURNAL OF MEDICINAL CHE... 14
- DRUG DEVELOPMENT RESEARCH 13
- PURINERGIC SIGNALLING 13
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- TETRAHEDRON LETTERS 10
- BIOORGANIC & MEDICINAL CHEMISTRY 9
Serie
- HANDBOOK OF EXPERIMENTAL PHARMACO... 2
- PHARMACOCHEMISTRY LIBRARY 1
- THE RECEPTORS 1
Keyword
- adenosine receptors 36
- A 17
- Apoptosis 17
- Adenosine 13
- 3 12
- Adenosine receptors 10
- 1 9
- Humans 7
- Animals 6
- Pharmacology 6
Lingua
- eng 459
- ita 6
- spa 1
Accesso al fulltext
- no fulltext 424
- reserved 22
- partially open 16
- open 4