MALFACINI, Davide

MALFACINI, Davide  

Dipartimento di Scienze mediche  

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Risultati 1 - 20 di 29 (tempo di esecuzione: 0.061 secondi).
Titolo Data di pubblicazione Autore(i) File
1,4-Dioxolane-triazaspirodecanone derivatives as nociceptin/orphanin FQ receptor ligands 2014 S., Corrado; C., Sorbi; A., Tait; U. M., Battisti; Camarda, Valeria; Malfacini, Davide; Calo', Gi...rolamo; L., Brasili file con accesso da definire
[D-Pen(p-tBuBzl)5]NPS, a novel ligand for the neuropeptide S receptor: structure activity and pharmacological studies 2014 Ruzza, Chiara; L., del Zoppo; Malfacini, Davide; Pela', Michela; Trapella, Claudio; P., Grieco; S...alvadori, Severo; Calo', Girolamo; Guerrini, Remo file con accesso da definire
A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ. 2014 Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pela', Michela; Molinari, Stefano; Cerlesi, Ma...ria Camilla; Malfacini, Davide; Rizzi, Anna; Salvadori, Severo; Calo', Girolamo file con accesso da definire
Acute and chronic antiparkinsonian effects of the novel nociceptin/orphanin FQ receptor antagonist NiK-21273 in comparison with SB-612111 2013 Marti, Matteo; Mela, Flora; Budri, Mirco; Volta, Mattia; Malfacini, Davide; Molinari, Stefano; N.... T., Zaveri; S., Ronzoni; P., Petrillo; Calo', Girolamo; Morari, Michele file con accesso da definire
Beta-arrestin 2 rather than G protein efficacy determines the anxiolytic- versus antidepressant-like effects of nociceptin/orphanin FQ receptor ligands 2016 Asth, L; Ruzza, Chiara; Malfacini, Davide; Medeiros, I; Guerrini, Remo; Zaveri, N. T; Gavioli, E.... C; Calo', Girolamo
Characterisation of the novel mixed Mu-NOP peptide ligand dermorphin-N/OFQ (DeNo) 2016 Bird, Mark F.; Camilla Cerlesi, Maria; Brown, Mark; Malfacini, Davide; Vezzi, Vanessa; Molinari, ...Paola; Micheli, Laura; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Guerrini, Remo; Calo', Girolamo; Lambert, David G.
Exploring pharmacological activities and signaling of morphinans substituted in position 6 as potent agonists interacting with the μ opioid receptor 2014 Tanila Ben, Haddou; Malfacini, Davide; Calo', Girolamo; Mario D., Aceto; Louis S., Harris; John R...., Traynor; Andrew, Coop; Helmut, Schmidhammer; Mariana, Spetea file con accesso da definire
Functional Selectivity Does Not Predict Antinociceptive/Locomotor Impairing Potencies of NOP Receptor Agonists 2021 Azevedo Neto, J.; Ruzza, C.; Sturaro, C.; Malfacini, D.; Pacifico, S.; Zaveri, N. T.; Calo, G.
In vitro and in vivo pharmaco-dynamic study of the novel fentanyl derivatives: Acrylfentanyl, Ocfentanyl and Furanylfentanyl 2022 Bilel, Sabrine; Azevedo Neto, Joaquim; Arfè, Raffaella; Tirri, Micaela; Gaudio, Rosa Maria; Fanti...nati, Anna; Bernardi, Tatiana; Boccuto, Federica; Marchetti, Beatrice; Corli, Giorgia; Serpelloni, Giovanni; De-Giorgio, Fabio; Malfacini, Davide; Trapella, Claudio; Calo', Girolamo; Marti, Matteo file con accesso da definire
In vitro and in vivo pharmacological characterization of a neuropeptide S tetrabranched derivative 2015 Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Pulga, Alice; Pacifico, Salvatore; Salvadori, Seve...ro; Trapella, Claudio; Reinscheid, Rainer K; Calo', Girolamo; Guerrini, Remo file con accesso da definire
In vitro and in vivo pharmacological characterization of nociceptin/orphanin FQ tetrabranched derivatives 2014 Rizzi, Anna; Malfacini, Davide; Cerlesi, Maria Camilla; Ruzza, Chiara; Marzola, Erika; M. F., Bir...d; D. J., Rowbotham; Salvadori, Severo; Guerrini, Remo; D. G., Lambert; Calo', Girolamo file con accesso da definire
In vitro and in vivo pharmacological characterization of Pronetupitant, a prodrug of the neurokinin 1 receptor antagonist Netupitant 2015 Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Molinari, Stefano; Giuliano, Claudio; Lovati, Eman...uela; Pietra, Claudio; Calo', Girolamo file con accesso da definire
In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations 2016 Ferrari, Federica; Cerlesi, Maria Camilla; Malfacini, Davide; Asth, Laila; Gavioli, Elaine C; Jou...rnigan, Blair V; Kamakolanu, Uma Gayathri; Meyer, Michael E; Yasuda, Dennis; Polgar, Willma E; Rizzi, Anna; Guerrini, Remo; Ruzza, Chiara; Zaveri, Nurulain T; Calo', Girolamo file con accesso da definire
In vitro pharmacological characterization of a novel unbiased NOP receptor-selective nonpeptide agonist AT-403 2017 Ferrari, Federica; Malfacini, Davide; Journigan, Blair V.; Bird, Mark F.; Trapella, Claudio; Guer...rini, Remo; Lambert, David G.; Calo', Girolamo; Zaveri, Nurulain T. file con accesso da definire
NOP receptor pharmacological profile – A dynamic mass redistribution study 2018 Malfacini, Davide; Simon, Katharina; Trapella, Claudio; Guerrini, Remo; Zaveri, Nurulain T.; Kost...enis, Evi; Calo, Girolamo
Novel ligands and assays for nociceptin/orphanin FQ and classical opioid receptors 2015 Malfacini, Davide
Pharmacological Assays for Investigating the NOP Receptor 2019 Malfacini, Davide; Calo', Girolamo
Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist 2016 Rizzi, Anna; Cerlesi, Maria Camilla; Ruzza, Chiara; Malfacini, Davide; Ferrari, Federica; Bianco,... Sara; Costa, Tommaso; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo file con accesso da definire
Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues 2014 Renata, Perlikowska; Malfacini, Davide; Cerlesi, Maria Camilla; Calo', Girolamo; Justyna, Piekiel...na; Léonore, Floriot; Tiphaine, Henry; Jean Claude do, Rego; Csaba, Tömböly; Alicja, Kluczyk; Anna, Janecka file con accesso da definire
Pharmacological characterization of naloxegol: In vitro and in vivo studies 2021 Costanzini, A.; Ruzza, C.; Neto, J. A.; Sturaro, C.; Malfacini, D.; Sternini, C.; De Giorgio, R.;... Calo, G.