Sfoglia per Titolo
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect study
2015 Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez Cara, Carlota; Cruz Lopez, Olga; Moorman, Allan R; Massink, Arnault; Ijzerman, Adriaan P; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological evaluation of a novel 99m Tc -Nitrido Labeled Substance P Derivative
file con accesso da definire2012 Pasquali, Micol; Uccelli, Licia; Boschi, Alessandra; DI DOMENICO, Giovanni; Pupillo, Gaia; Giganti, Melchiore; Guerrini, Remo; E., Janevik; K., Smilkov; Duatti, Adriano
Synthesis and biological evaluation of a series of 2-(3,4,5-trimethoxybenzoyl)-indol-3-yl acetic acid derivatives as potential agents against human leukemia K562 cells
file con accesso da definire2008 Romagnoli, Romeo; Baraldi, Pier Giovanni; Cruz Lopez, O.; Carrion, M. D.; Lopez Cara, C.; Balzarini, J.; Fabbri, Enrica; Gambari, Roberto
Synthesis and Biological Evaluation of a Series of Substituted Pyrazolo[3,4-d]-1,2,3-triazoles and Pyrazolo[3,4-d]oxazoles
file con accesso da definire1998 Vicentini, Chiara Beatrice; Manfredini, Stefano; Manfrini, M; Bazzanini, R; Musiu, C; Putzolu, M; Perra, G; Marongiu, M. E.
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain
file con accesso da definire2005 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaconinoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Synthesis and biological evaluation of allosteric A1 adenosine receptor modulators structurally related to 2-amino 4,5,6,7-tetrahydrobenzo(b) thiophen-3-yl-4-chloro phenyl methanone a potent compound useful to reduce neurophatic pain
file con accesso da definire2006 Romagnoli, Romeo; Iaconinoto, M. A.; Carrion, M. D.; Cara, C. L.; Shryock, J. C.; Leung, E.; Moorman, A. R.; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea
Synthesis and biological evaluation of alpha-bromoacryloylamido indolyl pyridinyl propenones as potent apoptotic inducers in human leukaemia cells
2018 Romagnoli, Romeo; Prencipe, Filippo; Lopez-Cara, Luisa Carlota; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco
Synthesis and Biological Evaluation of Diastereoisomerically Pure N,O-Nucleosides
file con accesso da definire2010 B., Russo; Bortolini, Olga; A., De Nino; A., Garofalo; A., Melicchio; L., Maiuolo
Synthesis and biological evaluation of diastereoisomerically pure N,O-nucleosides
2010 Bortolini, Olga; DE NINO, A.; Eliseo, T.; Gavioli, Riccardo; Maiuolo, L.; Russo, B.; Sforza, Fabio
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity
2016 Di Capua, A; Sticozzi, Claudia; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, Giuseppe; Giorgi, Giulia; Giordani, Alice; Poce, G; Biava, M; Anzini, M.
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
2022 Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Synthesis and biological evaluation of new 8-heterocyclic xanthine derivative as highly potent and selective human A2B adenosine receptor antagonist
file con accesso da definire2006 Baraldi, Pier Giovanni; Tabrizi, M. A.; Preti, Delia; Bovero, A.; Romagnoli, Romeo; Fruttarolo, Francesca; Zaid, N. A.; Moorman, A. R.; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues. J.Pept.Sci, 18, 418-426, 2012.
file con accesso da definire2012 Mollica, A.; Feliciani, F.; Stefanucci, A.; Costante, R.; Lucente, G.; Pinnen, F.; Notaristefano, D.; Spisani, Susanna
Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
2020 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors
file con accesso da definire2006 Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea
Synthesis and Biological Evaluation of Novel 2-Amino-3-Aroyl-4-Neopentyl-5-Substituted Thiophene Derivatives as Allosteric Enhancers of the A1 Adenosine Receptor
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Kimatrai Salvador, M.; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Moorman, A. R.; Vincenzi, Fabrizio; Borea, A. P.; Varani, Katia
Synthesis and Biological Evaluation of Novel 2-Aroyl Benzofuran-Based Hydroxamic Acids as Antimicrotubule Agents
file con accesso da definire2024 Mariotto, Elena; Canton, Martina; Marchioro, Chiara; Brancale, Andrea; Hamel, Ernest; Varani, Katia; Vincenzi, Fabrizio; De Ventura, Tiziano; Padroni, Chiara; Viola, Giampietro; Romagnoli, Romeo
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; A. P., Ijzerman; A., Massink; O., Cruz Lopez; L. C., Lopez Cara; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; A. R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists
file con accesso da definire2004 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect study | 2015 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez Cara, Carlota; Cruz Lopez, Olga; Moorman, Allan R...; Massink, Arnault; Ijzerman, Adriaan P; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | |
Synthesis and biological evaluation of a novel 99m Tc -Nitrido Labeled Substance P Derivative | 2012 | Pasquali, Micol; Uccelli, Licia; Boschi, Alessandra; DI DOMENICO, Giovanni; Pupillo, Gaia; Gigant...i, Melchiore; Guerrini, Remo; E., Janevik; K., Smilkov; Duatti, Adriano | file con accesso da definire |
Synthesis and biological evaluation of a series of 2-(3,4,5-trimethoxybenzoyl)-indol-3-yl acetic acid derivatives as potential agents against human leukemia K562 cells | 2008 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Cruz Lopez, O.; Carrion, M. D.; Lopez Cara, C.; Balzari...ni, J.; Fabbri, Enrica; Gambari, Roberto | file con accesso da definire |
Synthesis and Biological Evaluation of a Series of Substituted Pyrazolo[3,4-d]-1,2,3-triazoles and Pyrazolo[3,4-d]oxazoles | 1998 | Vicentini, Chiara Beatrice; Manfredini, Stefano; Manfrini, M; Bazzanini, R; Musiu, C; Putzolu, M;... Perra, G; Marongiu, M. E. | file con accesso da definire |
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain | 2005 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaco...ninoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of allosteric A1 adenosine receptor modulators structurally related to 2-amino 4,5,6,7-tetrahydrobenzo(b) thiophen-3-yl-4-chloro phenyl methanone a potent compound useful to reduce neurophatic pain | 2006 | Romagnoli, Romeo; Iaconinoto, M. A.; Carrion, M. D.; Cara, C. L.; Shryock, J. C.; Leung, E.; Moor...man, A. R.; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of alpha-bromoacryloylamido indolyl pyridinyl propenones as potent apoptotic inducers in human leukaemia cells | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Lopez-Cara, Luisa Carlota; Oliva, Paola; Baraldi, Stefania; ...Baraldi, Pier Giovanni; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco | |
Synthesis and Biological Evaluation of Diastereoisomerically Pure N,O-Nucleosides | 2010 | B., Russo; Bortolini, Olga; A., De Nino; A., Garofalo; A., Melicchio; L., Maiuolo | file con accesso da definire |
Synthesis and biological evaluation of diastereoisomerically pure N,O-nucleosides | 2010 | Bortolini, Olga; DE NINO, A.; Eliseo, T.; Gavioli, Riccardo; Maiuolo, L.; Russo, B.; Sforza, Fabio | |
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity | 2016 | Di Capua, A; Sticozzi, Claudia; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, ...S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, Giuseppe; Giorgi, Giulia; Giordani, Alice; Poce, G; Biava, M; Anzini, M. | |
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents | 2022 | Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale..., Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta | |
Synthesis and biological evaluation of new 8-heterocyclic xanthine derivative as highly potent and selective human A2B adenosine receptor antagonist | 2006 | Baraldi, Pier Giovanni; Tabrizi, M. A.; Preti, Delia; Bovero, A.; Romagnoli, Romeo; Fruttarolo, F...rancesca; Zaid, N. A.; Moorman, A. R.; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues. J.Pept.Sci, 18, 418-426, 2012. | 2012 | Mollica, A.; Feliciani, F.; Stefanucci, A.; Costante, R.; Lucente, G.; Pinnen, F.; Notaristefano,... D.; Spisani, Susanna | file con accesso da definire |
Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold | 2020 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sa...ndra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto | |
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors | 2006 | Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto | file con accesso da definire |
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli..., Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and Biological Evaluation of Novel 2-Amino-3-Aroyl-4-Neopentyl-5-Substituted Thiophene Derivatives as Allosteric Enhancers of the A1 Adenosine Receptor | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Kimatra...i Salvador, M.; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Moorman, A. R.; Vincenzi, Fabrizio; Borea, A. P.; Varani, Katia | file con accesso da definire |
Synthesis and Biological Evaluation of Novel 2-Aroyl Benzofuran-Based Hydroxamic Acids as Antimicrotubule Agents | 2024 | Mariotto, Elena; Canton, Martina; Marchioro, Chiara; Brancale, Andrea; Hamel, Ernest; Varani, Kat...ia; Vincenzi, Fabrizio; De Ventura, Tiziano; Padroni, Chiara; Viola, Giampietro; Romagnoli, Romeo | file con accesso da definire |
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; A. P., Ijzerman; A., Massink; O., Cruz Lopez; L. C., Lo...pez Cara; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; A. R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists | 2004 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
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