Sfoglia per Autore
A glance at adenosine receptors: Novel target for antitumor therapy
file con accesso da definire2003 Merighi, Stefania; Mirandola, P.; Varani, Katia; Gessi, Stefania; Leung, E.; Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Borea, Pier Andrea
New strategies for the synthesis of A(3) adenosine receptor antagonists
file con accesso da definire2003 Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Varani, Katia; Borea, Pier Andrea; Moorman, Ar
Recent developments in the field of A(2A) and A(3) adenosine receptor antagonists
file con accesso da definire2003 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Bovero, Andrea; Avitabile, B; Preti, Delia; Fruttarolo, Francesca; Romagnoli, Romeo; Varani, Katia; Borea, Pier Andrea
Biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptors
file con accesso da definire2003 Avitabile, Arianna; Baraldi, Pier Giovanni; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Leung, E.; Iannotta, Valeria; Merighi, Stefania; Gessi, Stefania; Varani, Katia; Pancaldi, Cecilia; Cattabriga, Elena; Borea, Pier Andrea
Synthesis, radiolabeling, and preliminary biological evaluation of [H-3]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl )-piperazine, a potent antagonist radioligand for the P2X(7) receptor
file con accesso da definire2004 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Mg; AGHAZADEH TABRIZI, Mojgan; Moorman, Ar; DI VIRGILIO, F; Cattabriga, Elena; Pancaldi, Cecilia; Gessi, Stefania; Borea, Pier Andrea
Allosteric modulators for the A1-adenosine receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; MOORMAN ALLAN, R.; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Romagnoli, Romeo
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; Preti, Delia; Pavani, Maria Giovanna; Bovero, Andrea; Iaconinoto, Antonietta; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; DI VIRGILIO, Francesco; Romagnoli, Romeo
Blockade of adenosine A(2A) receptors antagonizes parkinsonian tremor in the rat tacrine model by an action on specific striatal regions
file con accesso da definire2004 Simola, N; Fenu, S; Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Morelli, M.
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists
file con accesso da definire2004 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea
Design, synthesis and growth inhibition activity of bis-epoxyethyl derivatives of stallimycin modified on the amidino moiety
2004 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, M. G.; Fruttarolo, F.; Preti, Delia; Bovero, A.; AGHAZADEH TABRIZI, Mojgan; Bianchi, Nicoletta; Gambari, Roberto
[H-3]-MRE 2029-F20, a selective antagonist radioligand for the human A(2B) adenosine receptors
file con accesso da definire2004 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists
file con accesso da definire2004 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Romagnoli, Romeo; Fruttarolo, Francesca; Zaid, Na; Moorman, Ar; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and polypyrrole minor groove binders
file con accesso da definire2004 Baraldi, Pier Giovanni; Nunez, Md; AGHAZADEH TABRIZI, Mojgan; DE CLERCQ, E; Balzarini, J; Bermejo, J; Estevez, F; Romagnoli, Romeo
DNA minor groove binders as potential antitumor and antimicrobial agents
file con accesso da definire2004 Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Romagnoli, Romeo
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2.
file con accesso da definire2005 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Romagnoli, Romeo; Fruttarolo, Francesca; Pavani, G.; Iaconinoto, M. A.; Varani, Katia; Borea, Pier Andrea
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A(3) adenosine receptor antagonists
file con accesso da definire2005 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; Zaid, Na; Moorman, Ar; Varani, Katia; Borea, Pier Andrea
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2.
file con accesso da definire2005 Baraldi, Pier Giovanni; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Bovero, Andrea; Preti, Delia; Fruttarolo, Francesca; Moorman, Ar; Borea, Pier Andrea
Recent improvements in the field of A(3) adenosine receptor ligands
file con accesso da definire2005 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Carrion, Md; Iaconinoto, Antonietta; Borea, Pier Andrea
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and alpha-bromoacryloyl moieties
file con accesso da definire2005 Romagnoli, Romeo; Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Bermejo, J; Estevez, F; Borgatti, Monica; Gambari, Roberto
Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates
file con accesso da definire2005 Romagnoli, Romeo; Baraldi, Pier Giovanni; Iaconinoto, Antonietta; Carrion, Md; AGHAZADEH TABRIZI, Mojgan; Gambari, Roberto; Borgatti, Monica; Heilmann, J.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A glance at adenosine receptors: Novel target for antitumor therapy | 2003 | Merighi, Stefania; Mirandola, P.; Varani, Katia; Gessi, Stefania; Leung, E.; Baraldi, Pier Giovan...ni; AGHAZADEH TABRIZI, Mojgan; Borea, Pier Andrea | file con accesso da definire |
New strategies for the synthesis of A(3) adenosine receptor antagonists | 2003 | Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; AGHAZADEH TABRIZ...I, Mojgan; Preti, Delia; Varani, Katia; Borea, Pier Andrea; Moorman, Ar | file con accesso da definire |
Recent developments in the field of A(2A) and A(3) adenosine receptor antagonists | 2003 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Bovero, Andrea; Avitabile, B; Preti, Delia; Fr...uttarolo, Francesca; Romagnoli, Romeo; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptors | 2003 | Avitabile, Arianna; Baraldi, Pier Giovanni; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Leung, E....; Iannotta, Valeria; Merighi, Stefania; Gessi, Stefania; Varani, Katia; Pancaldi, Cecilia; Cattabriga, Elena; Borea, Pier Andrea | file con accesso da definire |
Synthesis, radiolabeling, and preliminary biological evaluation of [H-3]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl )-piperazine, a potent antagonist radioligand for the P2X(7) receptor | 2004 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Mg; AGHAZADEH TABRIZI, Mojgan; Moorman, Ar; DI ...VIRGILIO, F; Cattabriga, Elena; Pancaldi, Cecilia; Gessi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Allosteric modulators for the A1-adenosine receptor | 2004 | Baraldi, Pier Giovanni; MOORMAN ALLAN, R.; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Rom...agnoli, Romeo | file con accesso da definire |
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor | 2004 | Baraldi, Pier Giovanni; Preti, Delia; Pavani, Maria Giovanna; Bovero, Andrea; Iaconinoto, Antonie...tta; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; DI VIRGILIO, Francesco; Romagnoli, Romeo | file con accesso da definire |
Blockade of adenosine A(2A) receptors antagonizes parkinsonian tremor in the rat tacrine model by an action on specific striatal regions | 2004 | Simola, N; Fenu, S; Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Morelli, M. | file con accesso da definire |
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists | 2004 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Design, synthesis and growth inhibition activity of bis-epoxyethyl derivatives of stallimycin modified on the amidino moiety | 2004 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, M. G.; Fruttarolo, F.; Preti, Delia; Bovero, A....; AGHAZADEH TABRIZI, Mojgan; Bianchi, Nicoletta; Gambari, Roberto | |
[H-3]-MRE 2029-F20, a selective antagonist radioligand for the human A(2B) adenosine receptors | 2004 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Fran...cesca; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists | 2004 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Romagnoli, Romeo...; Fruttarolo, Francesca; Zaid, Na; Moorman, Ar; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and polypyrrole minor groove binders | 2004 | Baraldi, Pier Giovanni; Nunez, Md; AGHAZADEH TABRIZI, Mojgan; DE CLERCQ, E; Balzarini, J; Bermejo..., J; Estevez, F; Romagnoli, Romeo | file con accesso da definire |
DNA minor groove binders as potential antitumor and antimicrobial agents | 2004 | Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Preti, Delia; AGHAZADEH TABRIZI, M...ojgan; Pavani, Maria Giovanna; Romagnoli, Romeo | file con accesso da definire |
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2. | 2005 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Romagnoli, Romeo...; Fruttarolo, Francesca; Pavani, G.; Iaconinoto, M. A.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A(3) adenosine receptor antagonists | 2005 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Fran...cesca; Romagnoli, Romeo; Zaid, Na; Moorman, Ar; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2. | 2005 | Baraldi, Pier Giovanni; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Bovero, Andrea; Preti, Delia...; Fruttarolo, Francesca; Moorman, Ar; Borea, Pier Andrea | file con accesso da definire |
Recent improvements in the field of A(3) adenosine receptor ligands | 2005 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Carrion, Md; Iaconinoto, Antonietta; Borea, Pier Andrea | file con accesso da definire |
Design, synthesis, and biological evaluation of hybrid molecules containing alpha-methylene-gamma-butyrolactones and alpha-bromoacryloyl moieties | 2005 | Romagnoli, Romeo; Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Bermejo, J; Estevez, F; Borg...atti, Monica; Gambari, Roberto | file con accesso da definire |
Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates | 2005 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Iaconinoto, Antonietta; Carrion, Md; AGHAZADEH TABRIZI,... Mojgan; Gambari, Roberto; Borgatti, Monica; Heilmann, J. | file con accesso da definire |
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