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Synthesis and structure activity relationships of delthorphine analogues
file con accesso da definire1991 Salvadori, Severo; Marastoni, Mauro; Balboni, G.; Borea, Pier Andrea; Morari, Michele; Tomatis, Roberto
Synthesis by microwave irradiation and binding properties of novel 5-HT(1A) receptor ligands
file con accesso da definire2001 G., Caliendo; F., Fiorino; E., Perissutti; B., Severino; Gessi, Stefania; Cattabriga, Elena; Borea, Pier Andrea; V., Santagada
Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A(1) receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Shryock, Jc; Moorman, Ar; Iannotta, Valeria; Borea, Pier Andrea; Romagnoli, Romeo
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon
file con accesso da definire2007 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Ongini, E; EL KASHEF, H; Carrion, Md; Borea, Pier Andrea
Synthesis of imidazo[1,2-c]pyrazolo[4,3-e]pyrimidines and triazolo [5,1-i]purines: new potent A2 adenosine receptor antagonists
file con accesso da definire1993 Gatta, F.; DEL GIUDICE, M. R.; Borioni, A.; Borea, Pier Andrea; Dionisotti, S.; Ongini, Ennio
Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists
file con accesso da definire2002 Baraldi, Pier Giovanni; Cacciari, Barbara; Moro, S; Spalluto, G; Pastorin, G; DA ROS, T; Klotz, Kn; Varani, Katia; Gessi, Stefania; Borea, Pier Andrea
Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist
file con accesso da definire2002 Maconi, A; Pastorin, G; DA ROS, T; Spalluto, G; Gao, Zg; Jacobson, Ka; Baraldi, Pier Giovanni; Cacciari, Barbara; Varani, Katia; Moro, S; Borea, Pier Andrea
Synthesis, molecular modeling and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1 2,5]decanes and 2,7-diazatricyclo[4.4.0.0 3,8]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes
file con accesso da definire2000 Vianello, P.; Albinati, A.; Pinna, G.; Lavecchia, A.; Marinelli, L.; Borea, Pier Andrea; Gessi, Stefania; Fadda, P.; Tronci, S.; Cignarella, G.
Synthesis, radiolabeling, and preliminary biological evaluation of [H-3]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl )-piperazine, a potent antagonist radioligand for the P2X(7) receptor
file con accesso da definire2004 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Mg; AGHAZADEH TABRIZI, Mojgan; Moorman, Ar; DI VIRGILIO, F; Cattabriga, Elena; Pancaldi, Cecilia; Gessi, Stefania; Borea, Pier Andrea
Synthesis, structure-affinity relationships, and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists
file con accesso da definire2011 Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Squarcialupi, L; Filacchioni, G; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Ben, Dd; Lambertucci, C; Cristalli, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and structure activity relationships of delthorphine analogues | 1991 | Salvadori, Severo; Marastoni, Mauro; Balboni, G.; Borea, Pier Andrea; Morari, Michele; Tomatis, R...oberto | file con accesso da definire |
Synthesis by microwave irradiation and binding properties of novel 5-HT(1A) receptor ligands | 2001 | G., Caliendo; F., Fiorino; E., Perissutti; B., Severino; Gessi, Stefania; Cattabriga, Elena; Bore...a, Pier Andrea; V., Santagada | file con accesso da definire |
Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A(1) receptor | 2004 | Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Shryock, Jc; Moorman, Ar; Iannotta, Valeria; Bore...a, Pier Andrea; Romagnoli, Romeo | file con accesso da definire |
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon | 2007 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Ongini, E; EL KASHEF, H; Carrion, Md; Borea, Pier Andrea | file con accesso da definire |
Synthesis of imidazo[1,2-c]pyrazolo[4,3-e]pyrimidines and triazolo [5,1-i]purines: new potent A2 adenosine receptor antagonists | 1993 | Gatta, F.; DEL GIUDICE, M. R.; Borioni, A.; Borea, Pier Andrea; Dionisotti, S.; Ongini, Ennio | file con accesso da definire |
Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists | 2002 | Baraldi, Pier Giovanni; Cacciari, Barbara; Moro, S; Spalluto, G; Pastorin, G; DA ROS, T; Klotz, K...n; Varani, Katia; Gessi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist | 2002 | Maconi, A; Pastorin, G; DA ROS, T; Spalluto, G; Gao, Zg; Jacobson, Ka; Baraldi, Pier Giovanni; Ca...cciari, Barbara; Varani, Katia; Moro, S; Borea, Pier Andrea | file con accesso da definire |
Synthesis, molecular modeling and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1 2,5]decanes and 2,7-diazatricyclo[4.4.0.0 3,8]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes | 2000 | Vianello, P.; Albinati, A.; Pinna, G.; Lavecchia, A.; Marinelli, L.; Borea, Pier Andrea; Gessi, S...tefania; Fadda, P.; Tronci, S.; Cignarella, G. | file con accesso da definire |
Synthesis, radiolabeling, and preliminary biological evaluation of [H-3]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl]-4-(o-tolyl )-piperazine, a potent antagonist radioligand for the P2X(7) receptor | 2004 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Mg; AGHAZADEH TABRIZI, Mojgan; Moorman, Ar; DI ...VIRGILIO, F; Cattabriga, Elena; Pancaldi, Cecilia; Gessi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis, structure-affinity relationships, and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists | 2011 | Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Squarcialupi, L; Filacchioni, G; Varani, Katia; Vinc...enzi, Fabrizio; Borea, Pier Andrea; Ben, Dd; Lambertucci, C; Cristalli, G. | file con accesso da definire |
Legenda icone
- file ad accesso aperto
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile
Opzioni
Scopri
Tipologia
- 03 Contributo in rivista (Pubblic... 372
- 03 Contributo in rivista (Pubblic... 372
Data di pubblicazione
- 2020 - 2023 22
- 2010 - 2019 85
- 2000 - 2009 120
- 1990 - 1999 77
- 1980 - 1989 59
- 1977 - 1979 9
Editore
- Blackwell Munksgaard:PO Box 2148,... 17
- Elsevier BV:PO Box 211, 1000 AE A... 17
- Elsevier Science Limited:Oxford F... 17
- American Chemical Society:1155 Si... 8
- Editio Cantor Verlag GmbH ECV:Bae... 7
- Attuale:ELSEVIER SCIENCE SA, PO B... 5
- Marcel Dekker Incorporated:270 Ma... 5
- Springer Verlag Germany:Tiergarte... 5
- Nature Publishing Group:Brunel Ro... 3
- American Society for Pharmacology... 2
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 48
- BIOCHEMICAL PHARMACOLOGY 20
- BRITISH JOURNAL OF PHARMACOLOGY 18
- EUROPEAN JOURNAL OF MEDICINAL CHE... 13
- JOURNAL OF CHROMATOGRAPHY A 13
- ARZNEIMITTEL-FORSCHUNG 10
- DRUG DEVELOPMENT RESEARCH 8
- EUROPEAN JOURNAL OF PHARMACOLOGY 8
- IL FARMACO 8
- ACTA CRYSTALLOGRAPHICA. SECTION B... 7
Keyword
- adenosine receptors 48
- Adenosine receptors 22
- binding experiments 20
- A 17
- Adenosine 16
- 3 15
- adenosine 15
- 1 13
- Inflammation 12
- A2A antagonists 7
Lingua
- eng 369
- ita 2
- fre 1
Accesso al fulltext
- no fulltext 307
- open 28
- partially open 20
- reserved 17