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Synthesis and activity profiles of new dermorphin-(1-4) peptide analogues
file con accesso da definire1987 Marastoni, Mauro; Salvadori, Severo; Balboni, G.; Borea, Pier Andrea; Marzola, G.; Tomatis, Roberto
Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a.
file con accesso da definire2011 Simoni, Daniele; Rondanin, Riccardo; Marchetti, Paolo; Rullo, Cinzia; Baruchello, Riccardo; Grisolia, Giuseppina; G., Barbato; R., Giovannini; C., Marchioro; A. M., Capelli; C., Virginio; A., Bozzoli; Borea, Pier Andrea; Merighi, Stefania; D., Donati
Synthesis and biological characterization of [H-3] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)(4-chlorophenyl)-methan one, the first radiolabelled adenosine A(1) allosteric enhancer
file con accesso da definire2006 Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Leung, E; Moorman, Ar; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Romagnoli, Romeo
Synthesis and biological effects of novel 2-amino-3-(4-chlorobenzoyl)-4- substituted thiophenes as allosteric enhancers of the A1 adenosine receptor
file con accesso da definire2013 Romagnoli, Romeo; Baraldi, Pier Giovanni; Maria Dora, Carrion; Carlota Lopez, Cara; Maria Kimatrai, Salvador; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Allan R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A(1) adenosine receptor
file con accesso da definire2003 Baraldi, P. G.; Romagnoli, R.; Pavani, M. G.; Del Carmen Nunez, M.; Tabrizi, M. A.; Shryock, J. C.; Leung, E.; Moorman, A. R.; Uluoglu, C.; Iannotta, V.; Merighi, S.; Borea, P. A.
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[(4- arylpiperazin-1-yl)methyl]-5-substituted-thiophenes. Effect of the 5-modification on allosteric enhancer activity at the A1 adenosine receptor
file con accesso da definire2012 Romagnoli, Romeo; Baraldi, Pier Giovanni; M. D., Carrion; C., Lopez Cara; O., Cruz Lopez; M. K., Salvador; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Moorman, A. l. R.; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N- (substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor
file con accesso da definire2008 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Cruz Lopez, O; Iaconinoto, Antonietta; Preti, Delia; Shryock, Jc; Moorman, Ar; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect study
2015 Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez Cara, Carlota; Cruz Lopez, Olga; Moorman, Allan R; Massink, Arnault; Ijzerman, Adriaan P; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain
file con accesso da definire2005 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaconinoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and activity profiles of new dermorphin-(1-4) peptide analogues | 1987 | Marastoni, Mauro; Salvadori, Severo; Balboni, G.; Borea, Pier Andrea; Marzola, G.; Tomatis, Roberto | file con accesso da definire |
Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a. | 2011 | Simoni, Daniele; Rondanin, Riccardo; Marchetti, Paolo; Rullo, Cinzia; Baruchello, Riccardo; Griso...lia, Giuseppina; G., Barbato; R., Giovannini; C., Marchioro; A. M., Capelli; C., Virginio; A., Bozzoli; Borea, Pier Andrea; Merighi, Stefania; D., Donati | file con accesso da definire |
Synthesis and biological characterization of [H-3] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)(4-chlorophenyl)-methan one, the first radiolabelled adenosine A(1) allosteric enhancer | 2006 | Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Leung, E; Moorman, Ar; Varani, Katia; Vincenzi, F...abrizio; Borea, Pier Andrea; Romagnoli, Romeo | file con accesso da definire |
Synthesis and biological effects of novel 2-amino-3-(4-chlorobenzoyl)-4- substituted thiophenes as allosteric enhancers of the A1 adenosine receptor | 2013 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Maria Dora, Carrion; Carlota Lopez, Cara; Maria Kimatra...i, Salvador; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Allan R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A(1) adenosine receptor | 2003 | Baraldi, P. G.; Romagnoli, R.; Pavani, M. G.; Del Carmen Nunez, M.; Tabrizi, M. A.; Shryock, J. C....; Leung, E.; Moorman, A. R.; Uluoglu, C.; Iannotta, V.; Merighi, S.; Borea, P. A. | file con accesso da definire |
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[(4- arylpiperazin-1-yl)methyl]-5-substituted-thiophenes. Effect of the 5-modification on allosteric enhancer activity at the A1 adenosine receptor | 2012 | Romagnoli, Romeo; Baraldi, Pier Giovanni; M. D., Carrion; C., Lopez Cara; O., Cruz Lopez; M. K., ...Salvador; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Moorman, A. l. R.; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N- (substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor | 2008 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Cruz Lopez, O; Iaconinoto, Anton...ietta; Preti, Delia; Shryock, Jc; Moorman, Ar; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect study | 2015 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez Cara, Carlota; Cruz Lopez, Olga; Moorman, Allan R...; Massink, Arnault; Ijzerman, Adriaan P; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | |
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain | 2005 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaco...ninoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli..., Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Legenda icone
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Opzioni
Scopri
Tipologia
- 03 Contributo in rivista (Pubblic... 372
- 03 Contributo in rivista (Pubblic... 372
Data di pubblicazione
- 2020 - 2023 22
- 2010 - 2019 85
- 2000 - 2009 120
- 1990 - 1999 77
- 1980 - 1989 59
- 1977 - 1979 9
Editore
- Blackwell Munksgaard:PO Box 2148,... 17
- Elsevier BV:PO Box 211, 1000 AE A... 17
- Elsevier Science Limited:Oxford F... 17
- American Chemical Society:1155 Si... 8
- Editio Cantor Verlag GmbH ECV:Bae... 7
- Attuale:ELSEVIER SCIENCE SA, PO B... 5
- Marcel Dekker Incorporated:270 Ma... 5
- Springer Verlag Germany:Tiergarte... 5
- Nature Publishing Group:Brunel Ro... 3
- American Society for Pharmacology... 2
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 48
- BIOCHEMICAL PHARMACOLOGY 20
- BRITISH JOURNAL OF PHARMACOLOGY 18
- EUROPEAN JOURNAL OF MEDICINAL CHE... 13
- JOURNAL OF CHROMATOGRAPHY A 13
- ARZNEIMITTEL-FORSCHUNG 10
- DRUG DEVELOPMENT RESEARCH 8
- EUROPEAN JOURNAL OF PHARMACOLOGY 8
- IL FARMACO 8
- ACTA CRYSTALLOGRAPHICA. SECTION B... 7
Keyword
- adenosine receptors 48
- Adenosine receptors 22
- binding experiments 20
- A 17
- Adenosine 16
- 3 15
- adenosine 15
- 1 13
- Inflammation 12
- A2A antagonists 7
Lingua
- eng 369
- ita 2
- fre 1
Accesso al fulltext
- no fulltext 307
- open 28
- partially open 20
- reserved 17