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Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor
file con accesso da definire2012 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez, O.; Kimatrai Salvador, M.; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Moorman, A. R.; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea
Structure-activity studies of the Phe(4) residue of nociceptin(1-13)-NH2: Identification of highly potent agonists of the nociceptin/orphanin FQ receptor
file con accesso da definire2001 Guerrini, Remo; Calo', Girolamo; Bigoni, R; Rizzi, D; Rizzi, Anna; Zucchini, M; Varani, Katia; Hashiba, E; Lambert, Dg; Toth, G; Borea, Pier Andrea; Salvadori, Severo; Regoli, Domenico
STRUCTURE-ACTIVITY-RELATIONSHIPS IN HISTAMINE H-1 RECEPTOR ANTAGONISTS
file con accesso da definire1981 Bertolasi, Valerio; Borea, Pier Andrea; Gilli, Gastone; Sacerdoti, Michele
Structure-affinity relationships of a unique nicotinic ligand: N1-dimethyl-N4-phenylpiperazinium iodide (DMPP)
file con accesso da definire2001 Romanelli, M. N.; Manetti, D.; Scapecchi, S.; Borea, Pier Andrea; Dei, S.; Bartolini, A.; Ghelardini, C.; Gualtieri, F.; Guandalini, L.; Varani, Katia
Structuries of two 2-azylpyrazolo(4,3-c)quinolin-3-ones: CGS 8216, C16H11N30, and CGS 9896, C16H10ClN30, stereochemistry of benzodiazepine receptor ligands II.
file con accesso da definire1985 Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea
Study of lipophilic character of serotoninergic ligands
file con accesso da definire1996 Biagi, G. L.; Barbaro, A. M.; Sapone, A.; Borea, Pier Andrea; Varani, Katia; Recanatini, M.
Study of the lipophilic character of a series of β-carbolines
file con accesso da definire1989 Biagi, G. L.; Pietrogrande, Maria Chiara; Barbaro, A. M.; Guerra, M. C.; Borea, Pier Andrea; CANTELLI FORTI, G.
Study of the lipophylic character of xanthine and adenosine derivatives. II Relationships between logk', Rm and log P values
file con accesso da definire1990 Biagi, G. L.; Guerra, M. C.; Barbaro, A. M.; Barbieri, S.; Recanatini, M.; Borea, Pier Andrea
Study of the molecular factors determining specific binding to central adenosine A1 receptors by principal component analysis.
file con accesso da definire1990 Borea, Pier Andrea; Varani, Katia; V., Malaguti; Guerra, Laura; Pietrogrande, Maria Chiara; Gilli, Paola
Synthesis and activity of dermorphine growth hormone releasing factor hybrid peptides
file con accesso da definire1989 Marastoni, Mauro; Salvadori, Severo; Balboni, G.; Borea, Pier Andrea; Tomatis, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor | 2012 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez, O.; Kimatra...i Salvador, M.; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Moorman, A. R.; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Structure-activity studies of the Phe(4) residue of nociceptin(1-13)-NH2: Identification of highly potent agonists of the nociceptin/orphanin FQ receptor | 2001 | Guerrini, Remo; Calo', Girolamo; Bigoni, R; Rizzi, D; Rizzi, Anna; Zucchini, M; Varani, Katia; Ha...shiba, E; Lambert, Dg; Toth, G; Borea, Pier Andrea; Salvadori, Severo; Regoli, Domenico | file con accesso da definire |
STRUCTURE-ACTIVITY-RELATIONSHIPS IN HISTAMINE H-1 RECEPTOR ANTAGONISTS | 1981 | Bertolasi, Valerio; Borea, Pier Andrea; Gilli, Gastone; Sacerdoti, Michele | file con accesso da definire |
Structure-affinity relationships of a unique nicotinic ligand: N1-dimethyl-N4-phenylpiperazinium iodide (DMPP) | 2001 | Romanelli, M. N.; Manetti, D.; Scapecchi, S.; Borea, Pier Andrea; Dei, S.; Bartolini, A.; Ghelard...ini, C.; Gualtieri, F.; Guandalini, L.; Varani, Katia | file con accesso da definire |
Structuries of two 2-azylpyrazolo(4,3-c)quinolin-3-ones: CGS 8216, C16H11N30, and CGS 9896, C16H10ClN30, stereochemistry of benzodiazepine receptor ligands II. | 1985 | Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea | file con accesso da definire |
Study of lipophilic character of serotoninergic ligands | 1996 | Biagi, G. L.; Barbaro, A. M.; Sapone, A.; Borea, Pier Andrea; Varani, Katia; Recanatini, M. | file con accesso da definire |
Study of the lipophilic character of a series of β-carbolines | 1989 | Biagi, G. L.; Pietrogrande, Maria Chiara; Barbaro, A. M.; Guerra, M. C.; Borea, Pier Andrea; CANT...ELLI FORTI, G. | file con accesso da definire |
Study of the lipophylic character of xanthine and adenosine derivatives. II Relationships between logk', Rm and log P values | 1990 | Biagi, G. L.; Guerra, M. C.; Barbaro, A. M.; Barbieri, S.; Recanatini, M.; Borea, Pier Andrea | file con accesso da definire |
Study of the molecular factors determining specific binding to central adenosine A1 receptors by principal component analysis. | 1990 | Borea, Pier Andrea; Varani, Katia; V., Malaguti; Guerra, Laura; Pietrogrande, Maria Chiara; Gilli..., Paola | file con accesso da definire |
Synthesis and activity of dermorphine growth hormone releasing factor hybrid peptides | 1989 | Marastoni, Mauro; Salvadori, Severo; Balboni, G.; Borea, Pier Andrea; Tomatis, Roberto | file con accesso da definire |
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Opzioni
Scopri
Tipologia
- 03 Contributo in rivista (Pubblic... 372
- 03 Contributo in rivista (Pubblic... 372
Data di pubblicazione
- 2020 - 2023 22
- 2010 - 2019 85
- 2000 - 2009 120
- 1990 - 1999 77
- 1980 - 1989 59
- 1977 - 1979 9
Editore
- Blackwell Munksgaard:PO Box 2148,... 17
- Elsevier BV:PO Box 211, 1000 AE A... 17
- Elsevier Science Limited:Oxford F... 17
- American Chemical Society:1155 Si... 8
- Editio Cantor Verlag GmbH ECV:Bae... 7
- Attuale:ELSEVIER SCIENCE SA, PO B... 5
- Marcel Dekker Incorporated:270 Ma... 5
- Springer Verlag Germany:Tiergarte... 5
- Nature Publishing Group:Brunel Ro... 3
- American Society for Pharmacology... 2
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 48
- BIOCHEMICAL PHARMACOLOGY 20
- BRITISH JOURNAL OF PHARMACOLOGY 18
- EUROPEAN JOURNAL OF MEDICINAL CHE... 13
- JOURNAL OF CHROMATOGRAPHY A 13
- ARZNEIMITTEL-FORSCHUNG 10
- DRUG DEVELOPMENT RESEARCH 8
- EUROPEAN JOURNAL OF PHARMACOLOGY 8
- IL FARMACO 8
- ACTA CRYSTALLOGRAPHICA. SECTION B... 7
Keyword
- adenosine receptors 48
- Adenosine receptors 22
- binding experiments 20
- A 17
- Adenosine 16
- 3 15
- adenosine 15
- 1 13
- Inflammation 12
- A2A antagonists 7
Lingua
- eng 369
- ita 2
- fre 1
Accesso al fulltext
- no fulltext 307
- open 28
- partially open 20
- reserved 17