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STEREOCHEMISTRY OF BENZODIAZEPINE-RECEPTOR LIGANDS .2. STRUCTURES OF 2 2-ARYLPYRAZOLO[4,3-C]QUINOLIN-3-ONES - CGS8216, C16H11N3O, AND CGS9896, C16H10CLN3O
file con accesso da definire1985 Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea
Strategies for Drug Delivery into the Brain: A Review on Adenosine Receptors Modulation for Central Nervous System Diseases Therapy
file con accesso da definire2023 Fernandez, M; Nigro, M; Travagli, A; Pasquini, S; Vincenzi, F; Varani, K; Borea, Pa; Merighi, S; Gessi, S
Structural features controlling the binding of beta-carbolines to the benzodiazepine receptor
file con accesso da definire2004 Ferretti, Valeria; Gilli, Paola; Borea, Pier Andrea
Structure activity relationship for dermophin related tetrapeptides
file con accesso da definire1984 Sarto, Gianpietro; Borea, Pier Andrea; Salvadori, Severo; Tomatis, Roberto
Structure of 2-[7-chloro-2(3H)-oxo-5-phenyl-1H-1,4-benzodiazepin-1-yl]ethyl hydrogen succinate N4-oxide, C21H19ClN2O6
1984 Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea
Structure of 7-chloro-2-(3H)-oxo-5-phenyl-1H-1,4-benzodiazepine-1-yl-ethyl idrogen succinate N4-oxide, C21H19C1N206
file con accesso da definire1984 Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea
Structure of 7-chloro-2-methylamino-5-phenyl-3H-1,4-benzodiazepin-4-oxide (chlordiazepoxide)
file con accesso da definire1982 Bertolasi, Valerio; Sacerdoti, Michele; Gilli, Gastone; Borea, Pier Andrea
Structure of methyl beta-carboline-3-carboxylate (betaCCM). Stereochemistry of benzodiazepine receptor ligands I.
file con accesso da definire1984 Bertolasi, Valerio; Ferretti, Valeria; Gilli, Gastone; Borea, Pier Andrea
Structure-activity relationship studies and pharmacological characterization of N5-heteroarylalkyl-substituted-2-(2-furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine-based derivatives as inverse agonists at human A2Aadenosine receptor
2018 Varano, Flavia; Catarzi, Daniela; Vincenzi, Fabrizio; Falsini, Matteo; Pasquini, Silvia; Borea, Pier Andrea; Colotta, Vittoria; Varani, Katia
Structure-activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A(3) adenosine receptor antagonists.
file con accesso da definire2008 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Botta, M; Bernardini, C; Tafi, A; Tuccinardi, T; Martinelli, A; Varani, Katia; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
STEREOCHEMISTRY OF BENZODIAZEPINE-RECEPTOR LIGANDS .2. STRUCTURES OF 2 2-ARYLPYRAZOLO[4,3-C]QUINOLIN-3-ONES - CGS8216, C16H11N3O, AND CGS9896, C16H10CLN3O | 1985 | Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea | file con accesso da definire |
Strategies for Drug Delivery into the Brain: A Review on Adenosine Receptors Modulation for Central Nervous System Diseases Therapy | 2023 | Fernandez, M; Nigro, M; Travagli, A; Pasquini, S; Vincenzi, F; Varani, K; Borea, Pa; Merighi, S; ...Gessi, S | file con accesso da definire |
Structural features controlling the binding of beta-carbolines to the benzodiazepine receptor | 2004 | Ferretti, Valeria; Gilli, Paola; Borea, Pier Andrea | file con accesso da definire |
Structure activity relationship for dermophin related tetrapeptides | 1984 | Sarto, Gianpietro; Borea, Pier Andrea; Salvadori, Severo; Tomatis, Roberto | file con accesso da definire |
Structure of 2-[7-chloro-2(3H)-oxo-5-phenyl-1H-1,4-benzodiazepin-1-yl]ethyl hydrogen succinate N4-oxide, C21H19ClN2O6 | 1984 | Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea | |
Structure of 7-chloro-2-(3H)-oxo-5-phenyl-1H-1,4-benzodiazepine-1-yl-ethyl idrogen succinate N4-oxide, C21H19C1N206 | 1984 | Ferretti, Valeria; Bertolasi, Valerio; Gilli, Gastone; Borea, Pier Andrea | file con accesso da definire |
Structure of 7-chloro-2-methylamino-5-phenyl-3H-1,4-benzodiazepin-4-oxide (chlordiazepoxide) | 1982 | Bertolasi, Valerio; Sacerdoti, Michele; Gilli, Gastone; Borea, Pier Andrea | file con accesso da definire |
Structure of methyl beta-carboline-3-carboxylate (betaCCM). Stereochemistry of benzodiazepine receptor ligands I. | 1984 | Bertolasi, Valerio; Ferretti, Valeria; Gilli, Gastone; Borea, Pier Andrea | file con accesso da definire |
Structure-activity relationship studies and pharmacological characterization of N5-heteroarylalkyl-substituted-2-(2-furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine-based derivatives as inverse agonists at human A2Aadenosine receptor | 2018 | Varano, Flavia; Catarzi, Daniela; Vincenzi, Fabrizio; Falsini, Matteo; Pasquini, Silvia; Borea, P...ier Andrea; Colotta, Vittoria; Varani, Katia | |
Structure-activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A(3) adenosine receptor antagonists. | 2008 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Botta, M; Bernardini, C; Tafi, A; Tuccinardi, T; Martinelli, A; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Legenda icone
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Opzioni
Scopri
Tipologia
- 03 Contributo in rivista (Pubblic... 372
- 03 Contributo in rivista (Pubblic... 372
Data di pubblicazione
- 2020 - 2023 22
- 2010 - 2019 85
- 2000 - 2009 120
- 1990 - 1999 77
- 1980 - 1989 59
- 1977 - 1979 9
Editore
- Blackwell Munksgaard:PO Box 2148,... 17
- Elsevier BV:PO Box 211, 1000 AE A... 17
- Elsevier Science Limited:Oxford F... 17
- American Chemical Society:1155 Si... 8
- Editio Cantor Verlag GmbH ECV:Bae... 7
- Attuale:ELSEVIER SCIENCE SA, PO B... 5
- Marcel Dekker Incorporated:270 Ma... 5
- Springer Verlag Germany:Tiergarte... 5
- Nature Publishing Group:Brunel Ro... 3
- American Society for Pharmacology... 2
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 48
- BIOCHEMICAL PHARMACOLOGY 20
- BRITISH JOURNAL OF PHARMACOLOGY 18
- EUROPEAN JOURNAL OF MEDICINAL CHE... 13
- JOURNAL OF CHROMATOGRAPHY A 13
- ARZNEIMITTEL-FORSCHUNG 10
- DRUG DEVELOPMENT RESEARCH 8
- EUROPEAN JOURNAL OF PHARMACOLOGY 8
- IL FARMACO 8
- ACTA CRYSTALLOGRAPHICA. SECTION B... 7
Keyword
- adenosine receptors 48
- Adenosine receptors 22
- binding experiments 20
- A 17
- Adenosine 16
- 3 15
- adenosine 15
- 1 13
- Inflammation 12
- A2A antagonists 7
Lingua
- eng 369
- ita 2
- fre 1
Accesso al fulltext
- no fulltext 307
- open 28
- partially open 20
- reserved 17