beta-Enaminoketoesters, obtained by metal-catalyzed reaction between alkyl acetoacetates and alkyl cyanoformates, are useful starting materials for rapid access to beta-acetyl-dehydroaspartic acid derivatives which could be transformed into (+/-)-2-azetidinones bearing a 1-hydroxy-ethyl substituent through suitable reductive processes.

A new simple route for the synthesis of (+/-)-2-azetidinones starting from beta-enaminoketoesters

DE RISI, Carmela;POLLINI, Gian Piero;VERONESE, Augusto;BERTOLASI, Valerio
1999

Abstract

beta-Enaminoketoesters, obtained by metal-catalyzed reaction between alkyl acetoacetates and alkyl cyanoformates, are useful starting materials for rapid access to beta-acetyl-dehydroaspartic acid derivatives which could be transformed into (+/-)-2-azetidinones bearing a 1-hydroxy-ethyl substituent through suitable reductive processes.
1999
DE RISI, Carmela; Pollini, Gian Piero; Veronese, Augusto; Bertolasi, Valerio
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Utilizza questo identificativo per citare o creare un link a questo documento: https://hdl.handle.net/11392/1198168
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