DALPIAZ, Alessandro
DALPIAZ, Alessandro
Dipartimento di Scienze chimiche, farmaceutiche ed agrarie
1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors
file con accesso da definire1996 Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINEDA DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia
[3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets
file con accesso da definire1996 Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea
[3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets
file con accesso da definire1996 Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea
[3H] SCH 58261 labels adenosine A2A receptors in human lymphocyte membranes
file con accesso da definire1997 Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea
[3H] SCH 58261 labels adenosine A2A receptors in human lymphocyte membranes
file con accesso da definire1997 Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea
A concerted binding study using binding measurements, X-ray structural data and molecular modeling on the stereochemical features responsible for the affinity of 6-arylpyrrolo[2,1-d][1,5]benzothiazepines to mitochondrial benzodiazepine receptors
file con accesso da definire1995 Dalpiaz, Alessandro; Bertolasi, Valerio; Borea, Pier Andrea; Nacci, V; Fiorini, I; Campiani, G; Mennini, T; Manzoni, C; Novellino, E; Greco, G.
A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach.
file con accesso da definire2012 Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spalluto, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach
2016 Marchetti, Paolo; Pavan, Barbara; Simoni, Daniele; Baruchello, Riccardo; Rondanin, Riccardo; Mischiati, Carlo; Feriotto, Giordana; Ferraro, Luca Nicola; Hsu, Lih Ching; Lee, Ray M.; Dalpiaz, Alessandro
Adenosine A1 receptor: Analysis of the potential therapeutic effects obtained by its activation in the central nervous system
file con accesso da definire2002 Dalpiaz, Alessandro; Manfredini, Stefano
Adenosine analogs prodrugs: design, synthesis and chemico-physical characterization of N6-cyclopentyladenosine (CPA) derivatives
file con accesso da definire2000 Manfredini, Stefano; Baraldi, P. G.; Durini, E.; Bortolotti, F.; Scatturin, Angelo; Dalpiaz, Alessandro
Adenylyl cyclases as innovative therapeutic goals.
file con accesso da definire2009 Pavan, Barbara; Biondi, Carla; Dalpiaz, Alessandro
Agonist behaviour of periodate oxidized analogs at adenosine A1 receptors
file con accesso da definire1995 Dalpiaz, Alessandro; Varani, Katia; Borea, Pier Andrea; Martini, C.; Chiellini, G.; Lucacchini, A.
Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A 1 receptors of LUF5831, a novel nonadenosine-like agonist
file con accesso da definire2006 Heitman, L. H.; MULDER KRIEGER, T.; Spanjersberg, R. F.; VON FRIJTAG DRABBE KUNZEL, J. K.; Dalpiaz, Alessandro; Ijzerman, A. P.
An RPE cell line as a useful in vitro model for studying retinoic acid receptor beta: expression and affinity.
file con accesso da definire2008 Pavan, Barbara; Dalpiaz, Alessandro; Biondi, Carla; Nieddu, M.; De Luca, A.; Prasad, P. D.; Paganetto, Guglielmo; Favaloro, B.
Application of the “in-oil nanoprecipitation” method in the encapsulation of hydrophilic drugs in PLGA nanoparticles
2016 Dalpiaz, Alessandro; Sacchetti, Francesca; Baldisserotto, Anna; Pavan, Barbara; Maretti, Eleonora; Iannuccelli, Valentina; Leo, Eliana
Ascorbic acid prodrugs of nipecotic, kynurenic and diclophenamic acids: design, synthesis and activity
file con accesso da definire2002 Dalpiaz, Alessandro; Pavan, Barbara; Vertuani, G; Scaglianti, M; Avanzi, L; Biondi, C; Scatturin, Angelo; Ferraro, Luca Nicola; Tanganelli, S; Prasad, P; Manfredini, Stefano
Ascorbic and 6-Br-ascorbic acid conjugates as a tool to increase the therapeutic effects of potentially central active drugs
file con accesso da definire2005 Dalpiaz, Alessandro; Pavan, Barbara; Vertuani, Silvia; Vitali, F; Scaglianti, M; Bortolotti, Fabrizio; Biondi, Carla; Scatturin, Angelo; Tanganelli, Sergio; Ferraro, Luca Nicola; Marzola, Giuliano; Prasad, P; Manfredini, Stefano
Bile acids modulation of nanoparticle macrophage uptake
file con accesso da definire2018 Dalpiaz, Alessandro; Pavan, Barbara; Fogagnolo, Marco; Ferraro, Luca; Sacchetti, Francesca; Maretti, Eleonora; Iannuccelli, Valentina; Leo, Eliana
Bile salt-coating modulates the macrophage uptake of nanocores constituted by a zidovudine prodrug and enhances its nose-to-brain delivery
2019 Dalpiaz, A.; Fogagnolo, M.; Ferraro, L.; Beggiato, S.; Hanuskova, M.; Maretti, E.; Sacchetti, F.; Leo, E.; Pavan, B.
Binding thermodynamics and intrinsic activity of adenosine A1 receptor ligands
file con accesso da definire2000 Dalpiaz, Alessandro; Scatturin, Angelo; Varani, Katia; Pecoraro, R.; Pavan, Barbara; Borea, Pier Andrea
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors | 1996 | Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINED...A DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia | file con accesso da definire |
| [3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets | 1996 | Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea | file con accesso da definire |
| [3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets | 1996 | Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea | file con accesso da definire |
| [3H] SCH 58261 labels adenosine A2A receptors in human lymphocyte membranes | 1997 | Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea | file con accesso da definire |
| [3H] SCH 58261 labels adenosine A2A receptors in human lymphocyte membranes | 1997 | Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea | file con accesso da definire |
| A concerted binding study using binding measurements, X-ray structural data and molecular modeling on the stereochemical features responsible for the affinity of 6-arylpyrrolo[2,1-d][1,5]benzothiazepines to mitochondrial benzodiazepine receptors | 1995 | Dalpiaz, Alessandro; Bertolasi, Valerio; Borea, Pier Andrea; Nacci, V; Fiorini, I; Campiani, G; M...ennini, T; Manzoni, C; Novellino, E; Greco, G. | file con accesso da definire |
| A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach. | 2012 | Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spallut...o, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
| A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach | 2016 | Marchetti, Paolo; Pavan, Barbara; Simoni, Daniele; Baruchello, Riccardo; Rondanin, Riccardo; Misc...hiati, Carlo; Feriotto, Giordana; Ferraro, Luca Nicola; Hsu, Lih Ching; Lee, Ray M.; Dalpiaz, Alessandro | |
| Adenosine A1 receptor: Analysis of the potential therapeutic effects obtained by its activation in the central nervous system | 2002 | Dalpiaz, Alessandro; Manfredini, Stefano | file con accesso da definire |
| Adenosine analogs prodrugs: design, synthesis and chemico-physical characterization of N6-cyclopentyladenosine (CPA) derivatives | 2000 | Manfredini, Stefano; Baraldi, P. G.; Durini, E.; Bortolotti, F.; Scatturin, Angelo; Dalpiaz, Ales...sandro | file con accesso da definire |
| Adenylyl cyclases as innovative therapeutic goals. | 2009 | Pavan, Barbara; Biondi, Carla; Dalpiaz, Alessandro | file con accesso da definire |
| Agonist behaviour of periodate oxidized analogs at adenosine A1 receptors | 1995 | Dalpiaz, Alessandro; Varani, Katia; Borea, Pier Andrea; Martini, C.; Chiellini, G.; Lucacchini, A. | file con accesso da definire |
| Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A 1 receptors of LUF5831, a novel nonadenosine-like agonist | 2006 | Heitman, L. H.; MULDER KRIEGER, T.; Spanjersberg, R. F.; VON FRIJTAG DRABBE KUNZEL, J. K.; Dalpia...z, Alessandro; Ijzerman, A. P. | file con accesso da definire |
| An RPE cell line as a useful in vitro model for studying retinoic acid receptor beta: expression and affinity. | 2008 | Pavan, Barbara; Dalpiaz, Alessandro; Biondi, Carla; Nieddu, M.; De Luca, A.; Prasad, P. D.; Pagan...etto, Guglielmo; Favaloro, B. | file con accesso da definire |
| Application of the “in-oil nanoprecipitation” method in the encapsulation of hydrophilic drugs in PLGA nanoparticles | 2016 | Dalpiaz, Alessandro; Sacchetti, Francesca; Baldisserotto, Anna; Pavan, Barbara; Maretti, Eleonora...; Iannuccelli, Valentina; Leo, Eliana | |
| Ascorbic acid prodrugs of nipecotic, kynurenic and diclophenamic acids: design, synthesis and activity | 2002 | Dalpiaz, Alessandro; Pavan, Barbara; Vertuani, G; Scaglianti, M; Avanzi, L; Biondi, C; Scatturin,... Angelo; Ferraro, Luca Nicola; Tanganelli, S; Prasad, P; Manfredini, Stefano | file con accesso da definire |
| Ascorbic and 6-Br-ascorbic acid conjugates as a tool to increase the therapeutic effects of potentially central active drugs | 2005 | Dalpiaz, Alessandro; Pavan, Barbara; Vertuani, Silvia; Vitali, F; Scaglianti, M; Bortolotti, Fabr...izio; Biondi, Carla; Scatturin, Angelo; Tanganelli, Sergio; Ferraro, Luca Nicola; Marzola, Giuliano; Prasad, P; Manfredini, Stefano | file con accesso da definire |
| Bile acids modulation of nanoparticle macrophage uptake | 2018 | Dalpiaz, Alessandro; Pavan, Barbara; Fogagnolo, Marco; Ferraro, Luca; Sacchetti, Francesca; Maret...ti, Eleonora; Iannuccelli, Valentina; Leo, Eliana | file con accesso da definire |
| Bile salt-coating modulates the macrophage uptake of nanocores constituted by a zidovudine prodrug and enhances its nose-to-brain delivery | 2019 | Dalpiaz, A.; Fogagnolo, M.; Ferraro, L.; Beggiato, S.; Hanuskova, M.; Maretti, E.; Sacchetti, F.;... Leo, E.; Pavan, B. | |
| Binding thermodynamics and intrinsic activity of adenosine A1 receptor ligands | 2000 | Dalpiaz, Alessandro; Scatturin, Angelo; Varani, Katia; Pecoraro, R.; Pavan, Barbara; Borea, Pier ...Andrea | file con accesso da definire |