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In vitro pharmacological characterization of a novel unbiased NOP receptor-selective nonpeptide agonist AT-403
file con accesso da definire2017 Ferrari, Federica; Malfacini, Davide; Journigan, Blair V.; Bird, Mark F.; Trapella, Claudio; Guerrini, Remo; Lambert, David G.; Calo', Girolamo; Zaveri, Nurulain T.
Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt(1)]N/OFQ(1-13)
file con accesso da definire2017 Cerlesi, Maria Camilla; Ding, Huiping; Bird, Mark F; Kiguchi, Norikazu; Ferrari, Federica; Malfacini, Davide; Rizzi, Anna; Ruzza, Chiara; Lambert, David G; Ko, Mei Chuan; Calo', Girolamo; Guerrini, Remo
NOP receptor pharmacological profile – A dynamic mass redistribution study
2018 Malfacini, Davide; Simon, Katharina; Trapella, Claudio; Guerrini, Remo; Zaveri, Nurulain T.; Kostenis, Evi; Calo, Girolamo
Rational design of a heterotrimeric G protein subunit with artificial inhibitor sensitivity
file con accesso da definire2019 Malfacini, D.; Patt, J.; Annala, S.; Harpsoe, K.; Eryilmaz, F.; Reher, R.; Crusemann, M.; Hanke, W.; Zhang, H.; Tietze, D.; Gloriam, D. E.; Brauner-Osborne, H.; Stromgaard, K.; Konig, G. M.; Inoue, A.; Gomeza, J.; Kostenis, E.
Pharmacological Assays for Investigating the NOP Receptor
2019 Malfacini, Davide; Calo', Girolamo
Functional Selectivity Does Not Predict Antinociceptive/Locomotor Impairing Potencies of NOP Receptor Agonists
2021 Azevedo Neto, J.; Ruzza, C.; Sturaro, C.; Malfacini, D.; Pacifico, S.; Zaveri, N. T.; Calo, G.
Pharmacological characterization of naloxegol: In vitro and in vivo studies
2021 Costanzini, A.; Ruzza, C.; Neto, J. A.; Sturaro, C.; Malfacini, D.; Sternini, C.; De Giorgio, R.; Calo, G.
Pharmacology of Kappa Opioid Receptors: Novel Assays and Ligands
2022 Sturaro, Chiara; Malfacini, Davide; Argentieri, Michela; Djeujo, Francine M; Marzola, Erika; Albanese, Valentina; Ruzza, Chiara; Guerrini, Remo; Calo', Girolamo; Molinari, Paola
In vitro and in vivo pharmaco-dynamic study of the novel fentanyl derivatives: Acrylfentanyl, Ocfentanyl and Furanylfentanyl
2022 Bilel, Sabrine; Azevedo Neto, Joaquim; Arfè, Raffaella; Tirri, Micaela; Gaudio, Rosa Maria; Fantinati, Anna; Bernardi, Tatiana; Boccuto, Federica; Marchetti, Beatrice; Corli, Giorgia; Serpelloni, Giovanni; De-Giorgio, Fabio; Malfacini, Davide; Trapella, Claudio; Calo', Girolamo; Marti, Matteo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
In vitro pharmacological characterization of a novel unbiased NOP receptor-selective nonpeptide agonist AT-403 | 2017 | Ferrari, Federica; Malfacini, Davide; Journigan, Blair V.; Bird, Mark F.; Trapella, Claudio; Guer...rini, Remo; Lambert, David G.; Calo', Girolamo; Zaveri, Nurulain T. | file con accesso da definire |
Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt(1)]N/OFQ(1-13) | 2017 | Cerlesi, Maria Camilla; Ding, Huiping; Bird, Mark F; Kiguchi, Norikazu; Ferrari, Federica; Malfac...ini, Davide; Rizzi, Anna; Ruzza, Chiara; Lambert, David G; Ko, Mei Chuan; Calo', Girolamo; Guerrini, Remo | file con accesso da definire |
NOP receptor pharmacological profile – A dynamic mass redistribution study | 2018 | Malfacini, Davide; Simon, Katharina; Trapella, Claudio; Guerrini, Remo; Zaveri, Nurulain T.; Kost...enis, Evi; Calo, Girolamo | |
Rational design of a heterotrimeric G protein subunit with artificial inhibitor sensitivity | 2019 | Malfacini, D.; Patt, J.; Annala, S.; Harpsoe, K.; Eryilmaz, F.; Reher, R.; Crusemann, M.; Hanke, ...W.; Zhang, H.; Tietze, D.; Gloriam, D. E.; Brauner-Osborne, H.; Stromgaard, K.; Konig, G. M.; Inoue, A.; Gomeza, J.; Kostenis, E. | file con accesso da definire |
Pharmacological Assays for Investigating the NOP Receptor | 2019 | Malfacini, Davide; Calo', Girolamo | |
Functional Selectivity Does Not Predict Antinociceptive/Locomotor Impairing Potencies of NOP Receptor Agonists | 2021 | Azevedo Neto, J.; Ruzza, C.; Sturaro, C.; Malfacini, D.; Pacifico, S.; Zaveri, N. T.; Calo, G. | |
Pharmacological characterization of naloxegol: In vitro and in vivo studies | 2021 | Costanzini, A.; Ruzza, C.; Neto, J. A.; Sturaro, C.; Malfacini, D.; Sternini, C.; De Giorgio, R.;... Calo, G. | |
Pharmacology of Kappa Opioid Receptors: Novel Assays and Ligands | 2022 | Sturaro, Chiara; Malfacini, Davide; Argentieri, Michela; Djeujo, Francine M; Marzola, Erika; Alba...nese, Valentina; Ruzza, Chiara; Guerrini, Remo; Calo', Girolamo; Molinari, Paola | |
In vitro and in vivo pharmaco-dynamic study of the novel fentanyl derivatives: Acrylfentanyl, Ocfentanyl and Furanylfentanyl | 2022 | Bilel, Sabrine; Azevedo Neto, Joaquim; Arfè, Raffaella; Tirri, Micaela; Gaudio, Rosa Maria; Fanti...nati, Anna; Bernardi, Tatiana; Boccuto, Federica; Marchetti, Beatrice; Corli, Giorgia; Serpelloni, Giovanni; De-Giorgio, Fabio; Malfacini, Davide; Trapella, Claudio; Calo', Girolamo; Marti, Matteo |
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