Sfoglia per Autore
Conjugation of Dopamine and an A2A Adenosine Receptor Antagonist: a possible approach for the treatment of Parkinson’s Disease.
file con accesso da definire2012 Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; F., Bortolotti; G., Spalluto; S., Federico; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Effect of pulsed electromagnetic field exposure on adenosine receptors in rat brain
file con accesso da definire2012 Varani, Katia; Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Fini, Milena; Setti, Stefania; Cadossi, Ruggero; Borea, Pier Andrea
A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach.
file con accesso da definire2012 Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spalluto, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
Dopamine conjugation with A2A Antagonist: enhancement of drug effect and its controlled release in brain homogenates
file con accesso da definire2012 Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; F., Bortolotti; G., Spalluto; S., Federico; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor
file con accesso da definire2012 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez, O.; Kimatrai Salvador, M.; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Moorman, A. R.; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea
Electromagnetic fields (EMFs) and adenosine receptors modulate prostaglandin E(2) and cytokine release in human osteoarthritic synovial fibroblasts
2012 Ongaro, Alessia; Varani, Katia; Masieri, Federica Francesca; Pellati, Agnese; Massari, Leo; Cadossi, R.; Vincenzi, Fabrizio; Borea, Pier Andrea; Fini, M.; Caruso, Angelo; DE MATTEI, Monica
The Anti-Tumor Effect of A(3) Adenosine Receptors Is Potentiated by Pulsed Electromagnetic Fields in Cultured Neural Cancer Cells
file con accesso da definire2012 Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Gessi, Stefania; Merighi, Stefania; Setti, S.; Cadossi, R.; Borea, Pier Andrea; Varani, Katia
2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation
file con accesso da definire2013 Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S.
A(2A) adenosine receptors are differentially modulated by pharmacological treatments in rheumatoid arthritis patients and their stimulation ameliorates adjuvant-induced arthritis in rats
file con accesso da definire2013 Vincenzi, Fabrizio; Padovan, Melissa; Targa, Martina; Corciulo, Carmen; Giacuzzo, Sarah; Merighi, Stefania; Gessi, Stefania; Govoni, Marcello; Borea, Pa; Varani, Katia
Functional tissue engineering in articular cartilage repair: is there a role for electromagnetic biophysical stimulation?
2013 Fini, Milena; Pagani, Stefania; Giavaresi, Gianluca; DE MATTEI, Monica; Ongaro, Alessia; Varani, Katia; Vincenzi, Fabrizio; Massari, Leo; Cadossi, Matteo
Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists
file con accesso da definire2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
A(2A) adenosine receptors are up-regulated in lymphocytes from amyotrophic lateral sclerosis patients
file con accesso da definire2013 Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Casetta, Ilaria; Gentile, Mauro; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea; P., Popoli; Varani, Katia
Multiple sclerosis lymphocytes upregulate A(2A) adenosine receptors that are antiinflammatory when stimulated
file con accesso da definire2013 Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Merighi, Stefania; Gessi, Stefania; Casetta, Ilaria; Gentile, Mauro; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea; Varani, Katia
Antinociceptive effects of the selective CB2 agonist MT178 in inflammatory and chronic rodent pain models.
file con accesso da definire2013 Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; AGHAZADEH TABRIZI, Mojgan; Merighi, Stefania; Gessi, Stefania; Saponaro, Giulia; Baraldi, Pier Giovanni; Borea, Pier Andrea; Varani, Katia
Pulsed Electromagnetic Fields Increased the Anti-Inflammatory Effect of A2A and A3 Adenosine Receptors in Human T/C-28a2 Chondrocytes and hFOB 1.19 Osteoblasts.
file con accesso da definire2013 Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Gessi, Stefania; Merighi, Stefania; S., Setti; R., Cadossi; Goldring, M. B.; Borea, Pier Andrea; Varani, Katia
Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists.
file con accesso da definire2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; Moorman, Ar; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Tintori, C; Tuccinardi, T; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
The stimulation of A3 adenosine receptors reduces bone-residing breast cancer in a rat preclinical model
file con accesso da definire2013 Varani, Katia; Vincenzi, Fabrizio; Targa, Martina; Paradiso, Beatrice; Parrilli, A.; Fini, M.; Lanza, Giovanni; Borea, Pier Andrea
Pyrazolo[1,5-c]quinazoline derivatives and their simplified analogues as adenosine receptor antagonists; synthesis, structure-affinity relationships and molecular modeling studies
file con accesso da definire2013 D., Catarzi; V., Colotta; F., Varano; D., Poli; L., Squarcialupi; G., Filacchioni; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; D., Dal Ben; C., Lambertucci; G., Cristalli
Adenosine and adenosine receptors in rheumatoid arthritis
file con accesso da definire2013 Padovan, Melissa; Vincenzi, Fabrizio; Govoni, Marcello; Bortoluzzi, Alessandra; Borea, Pier Andrea; Varani, Katia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Conjugation of Dopamine and an A2A Adenosine Receptor Antagonist: a possible approach for the treatment of Parkinson’s Disease. | 2012 | Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; F., Bortolotti; G., Spalluto;... S., Federico; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Effect of pulsed electromagnetic field exposure on adenosine receptors in rat brain | 2012 | Varani, Katia; Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Fini, Milena; Setti, Stefani...a; Cadossi, Ruggero; Borea, Pier Andrea | file con accesso da definire |
A Novel Conjugated Agent between Dopamine and an A(2A) Adenosine Receptor Antagonist as a Potential Anti-Parkinson Multitarget Approach. | 2012 | Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; Bortolotti, Fabrizio; Spallut...o, G.; Federico, S.; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
Dopamine conjugation with A2A Antagonist: enhancement of drug effect and its controlled release in brain homogenates | 2012 | Dalpiaz, Alessandro; Cacciari, Barbara; Vicentini, Chiara Beatrice; F., Bortolotti; G., Spalluto;... S., Federico; Pavan, Barbara; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor | 2012 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez, O.; Kimatra...i Salvador, M.; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Moorman, A. R.; Vincenzi, Fabrizio; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Electromagnetic fields (EMFs) and adenosine receptors modulate prostaglandin E(2) and cytokine release in human osteoarthritic synovial fibroblasts | 2012 | Ongaro, Alessia; Varani, Katia; Masieri, Federica Francesca; Pellati, Agnese; Massari, Leo; Cados...si, R.; Vincenzi, Fabrizio; Borea, Pier Andrea; Fini, M.; Caruso, Angelo; DE MATTEI, Monica | |
The Anti-Tumor Effect of A(3) Adenosine Receptors Is Potentiated by Pulsed Electromagnetic Fields in Cultured Neural Cancer Cells | 2012 | Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Gessi, Stefania; Merighi, Stefania; Setti, ...S.; Cadossi, R.; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation | 2013 | Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo,... Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S. | file con accesso da definire |
A(2A) adenosine receptors are differentially modulated by pharmacological treatments in rheumatoid arthritis patients and their stimulation ameliorates adjuvant-induced arthritis in rats | 2013 | Vincenzi, Fabrizio; Padovan, Melissa; Targa, Martina; Corciulo, Carmen; Giacuzzo, Sarah; Merighi,... Stefania; Gessi, Stefania; Govoni, Marcello; Borea, Pa; Varani, Katia | file con accesso da definire |
Functional tissue engineering in articular cartilage repair: is there a role for electromagnetic biophysical stimulation? | 2013 | Fini, Milena; Pagani, Stefania; Giavaresi, Gianluca; DE MATTEI, Monica; Ongaro, Alessia; Varani, ...Katia; Vincenzi, Fabrizio; Massari, Leo; Cadossi, Matteo | |
Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists | 2013 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, R...omeo; Preti, Delia; Baraldi, Stefania; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
A(2A) adenosine receptors are up-regulated in lymphocytes from amyotrophic lateral sclerosis patients | 2013 | Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Casetta, Ilaria; Gentile, Mauro; Granieri, ...Enrico Gavino Giuseppe; Borea, Pier Andrea; P., Popoli; Varani, Katia | file con accesso da definire |
Multiple sclerosis lymphocytes upregulate A(2A) adenosine receptors that are antiinflammatory when stimulated | 2013 | Vincenzi, Fabrizio; Corciulo, Carmen; Targa, Martina; Merighi, Stefania; Gessi, Stefania; Casetta..., Ilaria; Gentile, Mauro; Granieri, Enrico Gavino Giuseppe; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Antinociceptive effects of the selective CB2 agonist MT178 in inflammatory and chronic rodent pain models. | 2013 | Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; AGHAZADEH TABRIZI, Mojgan; Merighi, Stefani...a; Gessi, Stefania; Saponaro, Giulia; Baraldi, Pier Giovanni; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Pulsed Electromagnetic Fields Increased the Anti-Inflammatory Effect of A2A and A3 Adenosine Receptors in Human T/C-28a2 Chondrocytes and hFOB 1.19 Osteoblasts. | 2013 | Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; Gessi, Stefania; Merighi, Stefania; S., Set...ti; R., Cadossi; Goldring, M. B.; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists. | 2013 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; Moorman, Ar; Romagnoli, Rome...o; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Tintori, C; Tuccinardi, T; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
The stimulation of A3 adenosine receptors reduces bone-residing breast cancer in a rat preclinical model | 2013 | Varani, Katia; Vincenzi, Fabrizio; Targa, Martina; Paradiso, Beatrice; Parrilli, A.; Fini, M.; La...nza, Giovanni; Borea, Pier Andrea | file con accesso da definire |
Pyrazolo[1,5-c]quinazoline derivatives and their simplified analogues as adenosine receptor antagonists; synthesis, structure-affinity relationships and molecular modeling studies | 2013 | D., Catarzi; V., Colotta; F., Varano; D., Poli; L., Squarcialupi; G., Filacchioni; Varani, Katia;... Vincenzi, Fabrizio; Borea, Pier Andrea; D., Dal Ben; C., Lambertucci; G., Cristalli | file con accesso da definire |
Adenosine and adenosine receptors in rheumatoid arthritis | 2013 | Padovan, Melissa; Vincenzi, Fabrizio; Govoni, Marcello; Bortoluzzi, Alessandra; Borea, Pier Andre...a; Varani, Katia | file con accesso da definire |
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