Sfoglia per Autore
Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor
file con accesso da definire2000 Baraldi, Pier Giovanni; Zaid, A. N.; Lampronti, Ilaria; Fruttarolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Leung, E.; Romagnoli, Romeo
Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders.
file con accesso da definire2001 Baraldi, Pier Giovanni; Balboni, Gianfranco; Pavani, Maria Giovanna; Spalluto, Giampiero; AGHAZADEH TABRIZI, Mojgan; DE CLERCQ, Erik; Balzarini, Jan; Bando, Toshikazu; Sugiyama, Hiroshi; Romagnoli, Romeo
Synthesis, biological activity and molecular modeling studies of 1,2,3,4-tetrahydroisoquinoline derivatives as conformationally constrained analogues of KN62, a potent antagonist of the P2X(7)-receptor containing a tyrosine moiety
file con accesso da definire2002 Baraldi, Pier Giovanni; Makaeva, R; Pavani, Maria Giovanna; Nunez, Md; Spalluto, G; Moro, S; Falzoni, S; DI VIRGILIO, Francesco; Romagnoli, Romeo
Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: Synthesis and antitumour activity
file con accesso da definire2002 Baraldi, Pier Giovanni; Romagnoli, Romeo; Pavani, Maria Giovanna; Nunez, Md; Bingham, Jp; Hartley, Ja
Design, synthesis and in vitro cytotoxicity of a cis-dichloroplatinum(II) complex linked to the minor groove binder stallimycin
file con accesso da definire2003 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Nunez, Md; Makaeva, R; Gambari, Roberto; LA COLLA, P; Romagnoli, Romeo
DNA minor-groove binders. Design, synthesis, and biological evaluation of ligands structurally related to CC-1065, distamycin, and anthramycin
file con accesso da definire2003 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Fruttarolo, Francesca; Avitabile, B; Bovero, Andrea; Pavani, Maria Giovanna; NUNEZ CARRETERO, Md; Romagnoli, Romeo
DNA minor groove binders as potential antitumor and antimicrobial agents
file con accesso da definire2004 Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Romagnoli, Romeo
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; Preti, Delia; Pavani, Maria Giovanna; Bovero, Andrea; Iaconinoto, Antonietta; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; DI VIRGILIO, Francesco; Romagnoli, Romeo
Allosteric modulators for the A1-adenosine receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; MOORMAN ALLAN, R.; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Romagnoli, Romeo
Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A(1) receptor
file con accesso da definire2004 Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Shryock, Jc; Moorman, Ar; Iannotta, Valeria; Borea, Pier Andrea; Romagnoli, Romeo
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain
file con accesso da definire2005 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaconinoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Synthesis and biological characterization of [H-3] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)(4-chlorophenyl)-methan one, the first radiolabelled adenosine A(1) allosteric enhancer
file con accesso da definire2006 Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Leung, E; Moorman, Ar; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Romagnoli, Romeo
Synthesis and biological evaluation of 2-amino-3-(3 ',4 ',5 '-trimethoxybenzoyl)-5-aryl thiophenes as a new class of potent antitubulin agents
file con accesso da definire2006 Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Fruttarolo, Francesca; Piccagli, Laura; Jung, Mk; Hamel, E; Borgatti, Monica; Gambari, Roberto
Synthesis and biological characterization of [3H] 2-amino 4,5,6,7-tetrahydrobenzo(b)thiophen-3-yl-4-chloro phenyl methanone, the first radiolabeled adenosine A1 allosteric enhancer
file con accesso da definire2006 Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Iaconinoto, M. A.; Carrios, Y. Pelegrina M. D.; Cara, C. C.; Bowerman, S.; Varani, Katia; Moorman, A. R.; Romagnoli, Romeo
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked heterocycles as template for the adenosine receptor antagonism: medicinal chemistry approach and SAR considerations.
file con accesso da definire2006 Baraldi, Pier Giovanni; Romagnoli, Romeo; El Kashef, H; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Pavani, Maria Giovanna; Zanella, Lorenzo; Fruttarolo, Francesca
Hybrid molecules based on distamycin A as potential antitumor agents
file con accesso da definire2006 Baraldi, Pier Giovanni; Zaid, An; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Iaconinoto, Antonietta; Pavani, Maria Giovanna; Carrion, Md; Cara, Cl; Romagnoli, Romeo
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors
file con accesso da definire2006 Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; Balzarini, J; Jordan, Ma; Hamel, E.
Novel combretastatin analogues endowed with antitumor activity
file con accesso da definire2006 Simoni, Daniele; Romagnoli, Romeo; Baruchello, Riccardo; Rondanin, Riccardo; Rizzi, Michele; Pavani, Maria Giovanna; Alloatti, D; Giannini, G; Marcellini, M; Riccioni, T; Castorina, M; Guglielmi, Mb; Bucci, F; Carminati, P; Pisano, C.
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; DI CRISTINA, A; Balzarini, J; Hadfield, Ja; Brancale, A; Hamel, E.
Rational Design, Synthesis, and Evaluation of Key Analogues of CC-1065 and the Duocarmycins
file con accesso da definire2007 Tichenor, Ms; Macmillan, Ks; Stover, Js; Wolkenberg, Se; Pavani, Maria Giovanna; Zanella, Lorenzo; Zaid, An; Spalluto, G; Rayl, Tj; Hwang, I; Baraldi, Pier Giovanni; Boger, D. L.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor | 2000 | Baraldi, Pier Giovanni; Zaid, A. N.; Lampronti, Ilaria; Fruttarolo, Francesca; Pavani, Maria Giov...anna; AGHAZADEH TABRIZI, Mojgan; Shryock, J. C.; Leung, E.; Romagnoli, Romeo | file con accesso da definire |
Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders. | 2001 | Baraldi, Pier Giovanni; Balboni, Gianfranco; Pavani, Maria Giovanna; Spalluto, Giampiero; AGHAZAD...EH TABRIZI, Mojgan; DE CLERCQ, Erik; Balzarini, Jan; Bando, Toshikazu; Sugiyama, Hiroshi; Romagnoli, Romeo | file con accesso da definire |
Synthesis, biological activity and molecular modeling studies of 1,2,3,4-tetrahydroisoquinoline derivatives as conformationally constrained analogues of KN62, a potent antagonist of the P2X(7)-receptor containing a tyrosine moiety | 2002 | Baraldi, Pier Giovanni; Makaeva, R; Pavani, Maria Giovanna; Nunez, Md; Spalluto, G; Moro, S; Falz...oni, S; DI VIRGILIO, Francesco; Romagnoli, Romeo | file con accesso da definire |
Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: Synthesis and antitumour activity | 2002 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Pavani, Maria Giovanna; Nunez, Md; Bingham, Jp; Hartley..., Ja | file con accesso da definire |
Design, synthesis and in vitro cytotoxicity of a cis-dichloroplatinum(II) complex linked to the minor groove binder stallimycin | 2003 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Nunez, Md; Makaeva, R;... Gambari, Roberto; LA COLLA, P; Romagnoli, Romeo | file con accesso da definire |
DNA minor-groove binders. Design, synthesis, and biological evaluation of ligands structurally related to CC-1065, distamycin, and anthramycin | 2003 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Fruttarolo, Francesca; Avitabile..., B; Bovero, Andrea; Pavani, Maria Giovanna; NUNEZ CARRETERO, Md; Romagnoli, Romeo | file con accesso da definire |
DNA minor groove binders as potential antitumor and antimicrobial agents | 2004 | Baraldi, Pier Giovanni; Bovero, Andrea; Fruttarolo, Francesca; Preti, Delia; AGHAZADEH TABRIZI, M...ojgan; Pavani, Maria Giovanna; Romagnoli, Romeo | file con accesso da definire |
Structure-activity relationships around the KN-62, a potent antagonist of the P2X(7)receptor | 2004 | Baraldi, Pier Giovanni; Preti, Delia; Pavani, Maria Giovanna; Bovero, Andrea; Iaconinoto, Antonie...tta; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; DI VIRGILIO, Francesco; Romagnoli, Romeo | file con accesso da definire |
Allosteric modulators for the A1-adenosine receptor | 2004 | Baraldi, Pier Giovanni; MOORMAN ALLAN, R.; AGHAZADEH TABRIZI, Mojgan; Pavani, Maria Giovanna; Rom...agnoli, Romeo | file con accesso da definire |
Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A(1) receptor | 2004 | Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Shryock, Jc; Moorman, Ar; Iannotta, Valeria; Bore...a, Pier Andrea; Romagnoli, Romeo | file con accesso da definire |
Synthesis and biological evaluation of allosteric A(1)-adenosine receptor modulators structurally related to (2-amino-4,5,6,7-tetrahydro-benzo[b]thiophen-3-yl)-(4-chloro-phenyl)-mie thanone, a potent compound useful to reduce neuropathic pain | 2005 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Iaco...ninoto, Antonietta; Carrion, Md; Cara, Cl; Shryock, Jc; Leung, E; Moorman, Ar; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological characterization of [H-3] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)(4-chlorophenyl)-methan one, the first radiolabelled adenosine A(1) allosteric enhancer | 2006 | Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Leung, E; Moorman, Ar; Varani, Katia; Vincenzi, F...abrizio; Borea, Pier Andrea; Romagnoli, Romeo | file con accesso da definire |
Synthesis and biological evaluation of 2-amino-3-(3 ',4 ',5 '-trimethoxybenzoyl)-5-aryl thiophenes as a new class of potent antitubulin agents | 2006 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Pret...i, Delia; Fruttarolo, Francesca; Piccagli, Laura; Jung, Mk; Hamel, E; Borgatti, Monica; Gambari, Roberto | file con accesso da definire |
Synthesis and biological characterization of [3H] 2-amino 4,5,6,7-tetrahydrobenzo(b)thiophen-3-yl-4-chloro phenyl methanone, the first radiolabeled adenosine A1 allosteric enhancer | 2006 | Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Iaconinoto, M. A.; Carrios, Y. Pelegrina M. D.; C...ara, C. C.; Bowerman, S.; Varani, Katia; Moorman, A. R.; Romagnoli, Romeo | file con accesso da definire |
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked heterocycles as template for the adenosine receptor antagonism: medicinal chemistry approach and SAR considerations. | 2006 | Baraldi, Pier Giovanni; Romagnoli, Romeo; El Kashef, H; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; ...Pavani, Maria Giovanna; Zanella, Lorenzo; Fruttarolo, Francesca | file con accesso da definire |
Hybrid molecules based on distamycin A as potential antitumor agents | 2006 | Baraldi, Pier Giovanni; Zaid, An; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan;... Iaconinoto, Antonietta; Pavani, Maria Giovanna; Carrion, Md; Cara, Cl; Romagnoli, Romeo | file con accesso da definire |
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors | 2006 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, Md; Cara, Cl; Preti, Delia; Frutta...rolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; Balzarini, J; Jordan, Ma; Hamel, E. | file con accesso da definire |
Novel combretastatin analogues endowed with antitumor activity | 2006 | Simoni, Daniele; Romagnoli, Romeo; Baruchello, Riccardo; Rondanin, Riccardo; Rizzi, Michele; Pava...ni, Maria Giovanna; Alloatti, D; Giannini, G; Marcellini, M; Riccioni, T; Castorina, M; Guglielmi, Mb; Bucci, F; Carminati, P; Pisano, C. | file con accesso da definire |
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, France...sca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; DI CRISTINA, A; Balzarini, J; Hadfield, Ja; Brancale, A; Hamel, E. | file con accesso da definire |
Rational Design, Synthesis, and Evaluation of Key Analogues of CC-1065 and the Duocarmycins | 2007 | Tichenor, Ms; Macmillan, Ks; Stover, Js; Wolkenberg, Se; Pavani, Maria Giovanna; Zanella, Lorenzo...; Zaid, An; Spalluto, G; Rayl, Tj; Hwang, I; Baraldi, Pier Giovanni; Boger, D. L. | file con accesso da definire |
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