Sfoglia per Autore
Preparation of fused purine derivatives as adenosine A3 receptor modulators.
file con accesso da definire2006 Baraldi, Pier Giovanni; Borea, Pier Andrea; Preti, Delia; AGHAZADEH TABRIZI, Mojgan
Recent developments in the field of A2B and A3 adenosine receptors antagonists
file con accesso da definire2006 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Zaid, N. A.; Moorman, A. R.; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea
New 2-arylpyrazolo[4,3-c]quinoline derivates as potent and selective human A3 adenosine receptor antagonists
file con accesso da definire2006 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; Hussein, E. K.; Moormann, A. R.; Varani, Katia; Borea, Pier Andrea
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked heterocycles as template for the adenosine receptor antagonism: medicinal chemistry approach and SAR considerations.
file con accesso da definire2006 Baraldi, Pier Giovanni; Romagnoli, Romeo; El Kashef, H; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Pavani, Maria Giovanna; Zanella, Lorenzo; Fruttarolo, Francesca
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor
file con accesso da definire2006 Romagnoli, Romeo; Baraldi, Pier Giovanni; Moorman, Ar; Iaconinoto, Antonietta; Carrion, Md; Cara, Cl; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Fruttarolo, Francesca; Baker, Sp; Varani, Katia; Borea, Pier Andrea
Pyrazolo [4,3-e][1,2,4]triazolo[1,5-c]pyrimidine template: Organic and medicinal chemistry approach
file con accesso da definire2006 Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; EL KASHEF, H; Preti, Delia; Bovero, Andrea; Fruttarolo, Francesca; Gordaliza, M; Borea, Pier Andrea
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors
file con accesso da definire2006 Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; Balzarini, J; Jordan, Ma; Hamel, E.
Hybrid molecules based on distamycin A as potential antitumor agents
file con accesso da definire2006 Baraldi, Pier Giovanni; Zaid, An; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Iaconinoto, Antonietta; Pavani, Maria Giovanna; Carrion, Md; Cara, Cl; Romagnoli, Romeo
Ligands for A(2B) adenosine receptor subtype
file con accesso da definire2006 Baraldi, Pier Giovanni; Romagnoli, Romeo; Preti, Delia; Fruttarolo, Francesca; Carrion, Md; AGHAZADEH TABRIZI, Mojgan
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea
Preparation of adenosine a2b receptor agonists for use as prodrugs treating diseases in mammals
file con accesso da definire2007 Baraldi, Pier Giovanni; Borea, Pier Andrea; Moorman, Ar; Preti, Delia
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; DI CRISTINA, A; Balzarini, J; Hadfield, Ja; Brancale, A; Hamel, E.
Hybrid molecules containing benzo[4,5]imidazo[1,2-d][1,2,4]thiadiazole and alpha-bromoacryloyl moieties as potent apoptosis inducers on human myeloid leukaemia cells
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; CRUZ LOPEZ, O; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Hellmann, J; Bermejo, J; Estevez, F.
Hybrid molecules between distamycin A and active moieties of antitumor agents
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo
N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Saponaro, Giulia; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea
Microwave-assisted synthesis of substituted 2,4-diarylthiazoles and their evaluation as anticancer agents
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez, Olga Cruz; Carrion, Maria Dora; Cara, Carlota Lopez; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Balzarini, J. a. n.
Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxyphenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez, O; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Balzarini, J; Hamel, E.
Novel 8-heterocyclyl xanthine derivatives in drug development - An update
file con accesso da definire2007 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon
file con accesso da definire2007 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Ongini, E; EL KASHEF, H; Carrion, Md; Borea, Pier Andrea
From tyrosine to glycine: Synthesis and biological activity of potent antagonists of the purinergic P2X(7) receptor
file con accesso da definire2007 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; CRUZ LOPEZ, O; AGHAZADEH TABRIZI, Mojgan; Moorman, Ar; Gessi, Stefania; Fogli, Eleonora; Sacchetto, Valeria; Borea, Pier Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Preparation of fused purine derivatives as adenosine A3 receptor modulators. | 2006 | Baraldi, Pier Giovanni; Borea, Pier Andrea; Preti, Delia; AGHAZADEH TABRIZI, Mojgan | file con accesso da definire |
Recent developments in the field of A2B and A3 adenosine receptors antagonists | 2006 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli..., Romeo; Zaid, N. A.; Moorman, A. R.; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
New 2-arylpyrazolo[4,3-c]quinoline derivates as potent and selective human A3 adenosine receptor antagonists | 2006 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Fran...cesca; Romagnoli, Romeo; Hussein, E. K.; Moormann, A. R.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and linked heterocycles as template for the adenosine receptor antagonism: medicinal chemistry approach and SAR considerations. | 2006 | Baraldi, Pier Giovanni; Romagnoli, Romeo; El Kashef, H; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; ...Pavani, Maria Giovanna; Zanella, Lorenzo; Fruttarolo, Francesca | file con accesso da definire |
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor | 2006 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Moorman, Ar; Iaconinoto, Antonietta; Carrion, Md; Cara,... Cl; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Fruttarolo, Francesca; Baker, Sp; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Pyrazolo [4,3-e][1,2,4]triazolo[1,5-c]pyrimidine template: Organic and medicinal chemistry approach | 2006 | Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; EL KASHEF, H; Preti, Delia; ...Bovero, Andrea; Fruttarolo, Francesca; Gordaliza, M; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of 2-(3 ',4 ',5 '-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors | 2006 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, Md; Cara, Cl; Preti, Delia; Frutta...rolo, Francesca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; Balzarini, J; Jordan, Ma; Hamel, E. | file con accesso da definire |
Hybrid molecules based on distamycin A as potential antitumor agents | 2006 | Baraldi, Pier Giovanni; Zaid, An; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan;... Iaconinoto, Antonietta; Pavani, Maria Giovanna; Carrion, Md; Cara, Cl; Romagnoli, Romeo | file con accesso da definire |
Ligands for A(2B) adenosine receptor subtype | 2006 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Preti, Delia; Fruttarolo, Francesca; Carrion, Md; AGHAZ...ADEH TABRIZI, Mojgan | file con accesso da definire |
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli..., Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Preparation of adenosine a2b receptor agonists for use as prodrugs treating diseases in mammals | 2007 | Baraldi, Pier Giovanni; Borea, Pier Andrea; Moorman, Ar; Preti, Delia | file con accesso da definire |
Synthesis and biological evaluation of 2-and 3-aminobenzo[b]thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; Fruttarolo, France...sca; Pavani, Maria Giovanna; AGHAZADEH TABRIZI, Mojgan; Tolomeo, M; Grimaudo, S; DI CRISTINA, A; Balzarini, J; Hadfield, Ja; Brancale, A; Hamel, E. | file con accesso da definire |
Hybrid molecules containing benzo[4,5]imidazo[1,2-d][1,2,4]thiadiazole and alpha-bromoacryloyl moieties as potent apoptosis inducers on human myeloid leukaemia cells | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; CRUZ LOPEZ, O; Preti, Delia; AGHAZADEH TAB...RIZI, Mojgan; Fruttarolo, Francesca; Hellmann, J; Bermejo, J; Estevez, F. | file con accesso da definire |
Hybrid molecules between distamycin A and active moieties of antitumor agents | 2007 | Baraldi, Pier Giovanni; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli..., Romeo | file con accesso da definire |
N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Saponaro,... Giulia; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Microwave-assisted synthesis of substituted 2,4-diarylthiazoles and their evaluation as anticancer agents | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Lopez, Olga Cruz; Carrion, Maria Dora; Cara, Carlota Lo...pez; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Balzarini, J. a. n. | file con accesso da definire |
Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxyphenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Remusat, V; Carrion, M. D.; Lopez Cara, C.; Cruz Lopez,... O; Preti, Delia; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Balzarini, J; Hamel, E. | file con accesso da definire |
Novel 8-heterocyclyl xanthine derivatives in drug development - An update | 2007 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia | file con accesso da definire |
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines structurally related to zaleplon | 2007 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Ongini, E; EL KASHEF, H; Carrion, Md; Borea, Pier Andrea | file con accesso da definire |
From tyrosine to glycine: Synthesis and biological activity of potent antagonists of the purinergic P2X(7) receptor | 2007 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Md; Cara, Cl; Preti, Delia; CRUZ LOPEZ, O; AGH...AZADEH TABRIZI, Mojgan; Moorman, Ar; Gessi, Stefania; Fogli, Eleonora; Sacchetto, Valeria; Borea, Pier Andrea | file con accesso da definire |
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