Sfoglia per Autore
Binding affinity of adenosine receptor agonists and antagonists at human cloned A3 adenosine receptors
file con accesso da definire1997 Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Borea, Pier Andrea
Synthesis, binding and thermodynamic studies of new highly selective A2A adenosine receptor antagonists
file con accesso da definire1997 Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, Giampiero; Ongini, E.; Dionisotti, S.; Varani, Katia; Gessi, Stefania; Borea, Pier Andrea
A new synthetic approach to indazole synthesis
file con accesso da definire1997 Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G.; Romagnoli, Romeo; Braccioli, G.; Zaid, A. N.; Delasinfantas, M. J. P.
Synthesis, cytotoxicity, antitumor activity and sequence selective binding of two pyrazole analogs structurally related to the antitumor agents U-71,184 and adozelesin
file con accesso da definire1997 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G; Gambari, Roberto; Bianchi, Nicoletta; Passadore, M; Ambrosino, P; Mongelli, N; Cozzi, P; Geroni, C.
Synthesis, solvolytic stability and cytotoxicity of a modified derivative of CPzI, a pyrazole analog of the alkylation subunit of the antitumor agent CC-1065: Effect of the nitrogen substitution on the functional reactivity
file con accesso da definire1997 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Zaid, An; Capolongo, L; Cozzi, P; Geroni, C; Mongelli, N.
Synthesis, cytotoxicity and antitumor activity of some new simplified pyrazole analogs of the antitumor agent CC-1065. Effect of an hydrophobic group on antitumor activity
file con accesso da definire1997 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Zaid, An; Cozzi, P; Geroni, C; Mongelli, N.
Second generation of A2A adenosine receptor antagonist: synthesis and biological evaluation
file con accesso da definire1998 Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, Giampiero; Ongini, E.; Varani, Katia; Borea, Pier Andrea
Ethyl (R,S)-5-acetyl-4,5-dihydro-3-isoxazoleacetate
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero
Heterocyclic analogs of DNA minor groove alkylating agents
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Zaid, An; Spalluto, G.
Ethyl-(R,S)-5-acetyl-4,5-dihydro-3-isoxazole acetate
file con accesso da definire1998 Baraldi, Pg; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.
Design, synthesis, and biological evaluation of a second generation of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as potent and selective A(2A) adenosine receptor antagonists
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G.; Bergonzoni, M.; Dionisotti, S.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
Synthesis and Biological Activity of a New Series of N6-Arylcarbamoyl, 2-(Ar)alkynyl-N6-arylcarbamoyl, and N6-Carboxamido Derivatives of Adenosine-5'-N-ethyluronamide as A1 and A3 Adenosine Receptor Agonists
1998 Baraldi, Pier Giovanni; Cacciari, Barbara; PINEDA DE INFANTAS MARIA, Jose; Romagnoli, Romeo; Spalluto, Giampiero; Volpini, Rosaria; Costanzi, Stefano; Vittori, Sauro; Cristalli, Gloria; Melman, Neli; Park, Kyungsun; Ji, Xiaoduo; JACOBSON KENNETH, A.
A2A-adenosine receptor reserve for coronary vasodilation
1998 SHRYOCK JOHN, C.; Snowdy, Stephen; Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, Giampiero; Monopoli, Angela; Ongini, Ennio; BAKER STEPHEN, P.; Belardinelli, Luiz
1-methyl-3-nitro-5-methoxycarbonyl pyrazole
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.
Design, synthesis and biological activity of a pyrrolo[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid
file con accesso da definire1998 Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Leoni, A; Romagnoli, Romeo; Spalluto, G; Mongelli, N; Howard, Pw; Thurston, De; Bianchi, Nicoletta; Gambari, Roberto
Binding affinity of adenosine receptor agonists and antagonists at human A3 adenosine receptors
file con accesso da definire1998 Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Gessi, Stefania; Borea, Pier Andrea
Binding affinity of adenosine receptor agonists and antagonists at human A3 adenosine receptors
file con accesso da definire1998 Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Gessi, Stefania; Borea, Pier Andrea
Binding affinity of adenosine receptor agonists and antagonists at human cloned A3 adenosine receptors
file con accesso da definire1998 Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Borea, Pier Andrea
Design, synthesis and biological properties of a new class of A2A adenosine receptor antagonists
file con accesso da definire1998 Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, G.; Bergonzoni, M.; Dionisotti, S.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
Selective binding to human genomic sequences of two synthetic analogues structurally related to U-71184 and adozelesin
file con accesso da definire1999 Bianchi, Nicoletta; Spalluto, G; Cacciari, Barbara; Romagnoli, Romeo; Feriotto, Giordana; Mischiati, Carlo; Rutigliano, C; Borsetti, E; Baraldi, Pier Giovanni; Gambari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Binding affinity of adenosine receptor agonists and antagonists at human cloned A3 adenosine receptors | 1997 | Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Borea, Pier... Andrea | file con accesso da definire |
Synthesis, binding and thermodynamic studies of new highly selective A2A adenosine receptor antagonists | 1997 | Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, Giampiero; Ongini, E.; Dionisotti, S.; Varan...i, Katia; Gessi, Stefania; Borea, Pier Andrea | file con accesso da definire |
A new synthetic approach to indazole synthesis | 1997 | Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G.; Romagnoli, Romeo; Braccioli, G.; Zaid, A.... N.; Delasinfantas, M. J. P. | file con accesso da definire |
Synthesis, cytotoxicity, antitumor activity and sequence selective binding of two pyrazole analogs structurally related to the antitumor agents U-71,184 and adozelesin | 1997 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G; Gambari, Roberto; Bianc...hi, Nicoletta; Passadore, M; Ambrosino, P; Mongelli, N; Cozzi, P; Geroni, C. | file con accesso da definire |
Synthesis, solvolytic stability and cytotoxicity of a modified derivative of CPzI, a pyrazole analog of the alkylation subunit of the antitumor agent CC-1065: Effect of the nitrogen substitution on the functional reactivity | 1997 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Zaid, An; C...apolongo, L; Cozzi, P; Geroni, C; Mongelli, N. | file con accesso da definire |
Synthesis, cytotoxicity and antitumor activity of some new simplified pyrazole analogs of the antitumor agent CC-1065. Effect of an hydrophobic group on antitumor activity | 1997 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Spalluto, G; Zaid, An; C...ozzi, P; Geroni, C; Mongelli, N. | file con accesso da definire |
Second generation of A2A adenosine receptor antagonist: synthesis and biological evaluation | 1998 | Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, Giampiero; Ongini, E.; Varani, Katia; Borea,... Pier Andrea | file con accesso da definire |
Ethyl (R,S)-5-acetyl-4,5-dihydro-3-isoxazoleacetate | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero | file con accesso da definire |
Heterocyclic analogs of DNA minor groove alkylating agents | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Romagnoli, Romeo; Zaid, An; Spalluto, G. | file con accesso da definire |
Ethyl-(R,S)-5-acetyl-4,5-dihydro-3-isoxazole acetate | 1998 | Baraldi, Pg; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G. | file con accesso da definire |
Design, synthesis, and biological evaluation of a second generation of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as potent and selective A(2A) adenosine receptor antagonists | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, G.; Bergonzoni, M.; Dionisotti, S.; Ongini, ...E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and Biological Activity of a New Series of N6-Arylcarbamoyl, 2-(Ar)alkynyl-N6-arylcarbamoyl, and N6-Carboxamido Derivatives of Adenosine-5'-N-ethyluronamide as A1 and A3 Adenosine Receptor Agonists | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; PINEDA DE INFANTAS MARIA, Jose; Romagnoli, Romeo; Spal...luto, Giampiero; Volpini, Rosaria; Costanzi, Stefano; Vittori, Sauro; Cristalli, Gloria; Melman, Neli; Park, Kyungsun; Ji, Xiaoduo; JACOBSON KENNETH, A. | |
A2A-adenosine receptor reserve for coronary vasodilation | 1998 | SHRYOCK JOHN, C.; Snowdy, Stephen; Baraldi, Pier Giovanni; Cacciari, Barbara; Spalluto, Giampiero...; Monopoli, Angela; Ongini, Ennio; BAKER STEPHEN, P.; Belardinelli, Luiz | |
1-methyl-3-nitro-5-methoxycarbonyl pyrazole | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G. | file con accesso da definire |
Design, synthesis and biological activity of a pyrrolo[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid | 1998 | Baraldi, Pier Giovanni; Cacciari, Barbara; Guiotto, A; Leoni, A; Romagnoli, Romeo; Spalluto, G; M...ongelli, N; Howard, Pw; Thurston, De; Bianchi, Nicoletta; Gambari, Roberto | file con accesso da definire |
Binding affinity of adenosine receptor agonists and antagonists at human A3 adenosine receptors | 1998 | Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Gessi, Stef...ania; Borea, Pier Andrea | file con accesso da definire |
Binding affinity of adenosine receptor agonists and antagonists at human A3 adenosine receptors | 1998 | Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Gessi, Stef...ania; Borea, Pier Andrea | file con accesso da definire |
Binding affinity of adenosine receptor agonists and antagonists at human cloned A3 adenosine receptors | 1998 | Varani, Katia; Cacciari, Barbara; Baraldi, Pier Giovanni; Dionisotti, S.; Ongini, E.; Borea, Pier... Andrea | file con accesso da definire |
Design, synthesis and biological properties of a new class of A2A adenosine receptor antagonists | 1998 | Cacciari, Barbara; Baraldi, Pier Giovanni; Spalluto, G.; Bergonzoni, M.; Dionisotti, S.; Ongini, ...E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Selective binding to human genomic sequences of two synthetic analogues structurally related to U-71184 and adozelesin | 1999 | Bianchi, Nicoletta; Spalluto, G; Cacciari, Barbara; Romagnoli, Romeo; Feriotto, Giordana; Mischia...ti, Carlo; Rutigliano, C; Borsetti, E; Baraldi, Pier Giovanni; Gambari, Roberto | file con accesso da definire |
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