Sfoglia per Autore
Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent delta-opioid antagonist
2001 Lovekamp, T; Cooper, Ps; Hardison, J; Bryant, Sd; Guerrini, Remo; Balboni, Gianfranco; Salvadori, Severo; Lazarus, Lh
Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore
file con accesso da definire2002 Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Negri, L; Giannini, E; Jinsmaa, Y; Bryant, Sd; Lazarus, Lh
Evaluation of the Dmt-Tic pharmacophore: Conversion of a potent delta-opioid receptor antagonist into a potent delta agonist and ligands with mixed properties
2002 Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Bianchi, C; Rizzi, D; Bryant, Sd; Lazarus, Lh
Crystal structures of dipeptides containing the Dmt-Tic pharmacophore
file con accesso da definire2002 Bryant, Sd; George, C; FLIPPEN ANDERSON, Jl; Deschamps, Jr; Salvadori, Severo; Balboni, Gianfranco; Guerrini, Remo; Lazarus, Lh
Synthesis and opioid activity of N,N-dimethyl-Dmt-Tic-NH-CH(R)-R ' analogues: Acquisition of potent delta antagonism
file con accesso da definire2003 Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Negri, L; Giannini, E; Bryant, Sd; Jinsmaa, Y; Lazarus, Lh
Peptidic delta opioid receptor agonists produce antidepressant-like effects in the forced swim test amd regulate BDNF mRNA expression in rats.
file con accesso da definire2006 Torregrossa, M. M.; Jutkiewicz, E. M.; Mosberg, H. I.; Balboni, Gianfranco; Watson, S. J.; Woods, J. H.
In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist, correlation between desensitization and tolerance.
file con accesso da definire2007 Aguila, B; Coulbault, L; Boulouaerd, M; Leveille, F; Davis, A; Toth, G; Borsodi, A; Balboni, Gianfranco; Salvadori, Severo; Jauzac, P; Allouche, S.
Delta-, but not mu-, opioid receptor stabilize K+ homeostasis by reducing Ca2+ influx in the cortex during acute hypoxia.
file con accesso da definire2007 Chao, D; BAZZY ASAAD, A; Balboni, Gianfranco; Xia, Y.
Hydrogen sulfide induced disruption of Na+ homeostasis in the cortex
file con accesso da definire2012 Chao, D; He, X; Yang, Y; Balboni, Gianfranco; Salvadori, Severo; Kim, Dh; Xia, Y.
Critical role for prokineticin 2 in CNS autoimmunity
file con accesso da definire2015 Abou Hamdan, Mhamad; Costanza, Massimo; Fontana, Elena; Di Dario, Marco; Musio, Silvia; Congiu, Cenzo; Onnis, Valentina; Lattanzi, Roberta; Radaelli, Marta; Martinelli, Vittorio; Salvadori, Severo; Negri, Lucia; Poliani, Pietro Luigi; Farina, Cinthia; Balboni, Gianfranco; Steinman, Lawrence; Pedotti, Rosetta
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones
2016 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna; Manfredini, Stefano; Pacifico, Salvatore; Liekens, Sandra; Balzarini, Jan
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent delta-opioid antagonist | 2001 | Lovekamp, T; Cooper, Ps; Hardison, J; Bryant, Sd; Guerrini, Remo; Balboni, Gianfranco; Salvadori,... Severo; Lazarus, Lh | |
Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore | 2002 | Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Negri, L; Giannini, E; Jinsmaa, Y; Bryant..., Sd; Lazarus, Lh | file con accesso da definire |
Evaluation of the Dmt-Tic pharmacophore: Conversion of a potent delta-opioid receptor antagonist into a potent delta agonist and ligands with mixed properties | 2002 | Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Bianchi, C; Rizzi, D; Bryant, Sd; Lazarus..., Lh | |
Crystal structures of dipeptides containing the Dmt-Tic pharmacophore | 2002 | Bryant, Sd; George, C; FLIPPEN ANDERSON, Jl; Deschamps, Jr; Salvadori, Severo; Balboni, Gianfranc...o; Guerrini, Remo; Lazarus, Lh | file con accesso da definire |
Synthesis and opioid activity of N,N-dimethyl-Dmt-Tic-NH-CH(R)-R ' analogues: Acquisition of potent delta antagonism | 2003 | Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Negri, L; Giannini, E; Bryant, Sd; Jinsma...a, Y; Lazarus, Lh | file con accesso da definire |
Peptidic delta opioid receptor agonists produce antidepressant-like effects in the forced swim test amd regulate BDNF mRNA expression in rats. | 2006 | Torregrossa, M. M.; Jutkiewicz, E. M.; Mosberg, H. I.; Balboni, Gianfranco; Watson, S. J.; Woods,... J. H. | file con accesso da definire |
In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist, correlation between desensitization and tolerance. | 2007 | Aguila, B; Coulbault, L; Boulouaerd, M; Leveille, F; Davis, A; Toth, G; Borsodi, A; Balboni, Gian...franco; Salvadori, Severo; Jauzac, P; Allouche, S. | file con accesso da definire |
Delta-, but not mu-, opioid receptor stabilize K+ homeostasis by reducing Ca2+ influx in the cortex during acute hypoxia. | 2007 | Chao, D; BAZZY ASAAD, A; Balboni, Gianfranco; Xia, Y. | file con accesso da definire |
Hydrogen sulfide induced disruption of Na+ homeostasis in the cortex | 2012 | Chao, D; He, X; Yang, Y; Balboni, Gianfranco; Salvadori, Severo; Kim, Dh; Xia, Y. | file con accesso da definire |
Critical role for prokineticin 2 in CNS autoimmunity | 2015 | Abou Hamdan, Mhamad; Costanza, Massimo; Fontana, Elena; Di Dario, Marco; Musio, Silvia; Congiu, C...enzo; Onnis, Valentina; Lattanzi, Roberta; Radaelli, Marta; Martinelli, Vittorio; Salvadori, Severo; Negri, Lucia; Poliani, Pietro Luigi; Farina, Cinthia; Balboni, Gianfranco; Steinman, Lawrence; Pedotti, Rosetta | file con accesso da definire |
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones | 2016 | Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna...; Manfredini, Stefano; Pacifico, Salvatore; Liekens, Sandra; Balzarini, Jan |
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