Sfoglia per Autore
Synthesis, metabolic stability and chemotactic activity of peptide T and its analogues
file con accesso da definire1990 Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Spisani, Susanna; Gavioli, Riccardo; Traniello, Maria Serena; Tomatis, Roberto
A CYCLIC PEPTIDE T ANALOGUE WITH HIGH CHEMOTACTIC ACTIVITY
file con accesso da definire1992 Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Scaranari, V.; Spisani, Susanna; Reali, Eva; Giuliani, Anna Lisa; Tomatis, Roberto
Conformational analysis of potent and very selective delta opioid dipeptide antagonists
file con accesso da definire1995 Amodeo, P; Balboni, Gianfranco; Crescenzi, O; Guerrini, Remo; Picone, D; Salvadori, Severo; Tancredi, T; Temussi, Pa
Acid catalysis in the formation of dioxopiperazines from peptides containing tetrahydroisoquinoline‐3‐carboxylic acid at position 2
file con accesso da definire1995 Capasso, S; Sica, F; Mazzarella, L; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo
DMT-TIC-OH, a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse
file con accesso da definire1996 Capasso, A; Guerrini, Remo; Balboni, Gianfranco; Sorrentino, L; Temussi, P; Lazarus, Lh; Bryant, Sd; Salvadori, Severo
Opioid diketopiperazines: Refinement of the delta opioid antagonist pharmacophore
file con accesso da definire1997 Bryant, Sd; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Lazarus, Lh
Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary δ opioid antagonist activity
file con accesso da definire1997 Salvadori, Severo; Balboni, Gianfranco; Guerrini, Remo; Tomatis, R; Bianchi, C; Bryant, Sd; Cooper, Ps; Lazarus, Lh
Design and solution structure of a partially rigid opioid antagonist lacking the basic center - Models of antagonism
file con accesso da definire1997 Crescenzi, O; Fraternali, F; Picone, D; Tancredi, T; Balboni, Gianfranco; Guerrini, Remo; Lazarus, Lh; Salvadori, Severo; Temussi, Pa
Design of μ selective opioid dipeptide antagonists
file con accesso da definire1997 Capasso, A; Amodeo, P; Balboni, Gianfranco; Guerrini, Remo; Lazarus, Lh; Temussi, Pa; Salvadori, Severo
Opioid diketopiperazines: Synthesis and activity of a prototypic class of opioid antagonists
file con accesso da definire1997 Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Bryant, Sd; Bianchi, C; Attila, M; Lazarus, Lh
Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides
file con accesso da definire1997 Tomatis, R; Marastoni, Mauro; Balboni, Gianfranco; Guerrini, Remo; Capasso, A; Sorrentino, L; Santagada, V; Caliendo, G; Lazarus, Lh; Salvadori, Severo
Design of d-opioid peptide antagonists for emerging drug applications
file con accesso da definire1998 L. H., Lazarus; S. n. D., Bryant; P. S., Cooper; Guerrini, Remo; Balboni, Gianfranco; Salvadori, Severo
Tritiation of delta opioid-receptor selective antagonist dipeptide ligands with extraordinary affinity containing 2 ', 6 ' dimethyltyrosine
file con accesso da definire1999 Kertesz, I; Toth, G; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo
Further Studies on the Dmt-Tic Pharmacophore: Hydrophobic Substituents at the C-Terminus Endow delta Antagonists To Manifest mu Agonism or mu Antagonism
file con accesso da definire1999 Salvadori, Severo; Guerrini, Remo; Balboni, Gianfranco; C., Bianchi; S. D., Bryant; P. S., Cooper; L. H., Lazarus
Synthesis, in vitro antiproliferative activity, and DNA-binding properties of hybrid molecules containing pyrrolo[2,1-c][1,4] benzodiazepine and minor-groove-binding oligopyrrole carriers
file con accesso da definire1999 Baraldi, Pier Giovanni; Balboni, Gianfranco; Cacciari, Barbara; A., Guiotto; Manfredini, Stefano; Romagnoli, Romeo; Spalluto, Giampiero; D. E., Thurston; P. W., Howard; Bianchi, Nicoletta; Rutigliano, Cristina; Mischiati, Carlo; Gambari, Roberto
Characterization of N,N(Me)(2)-Dmt-Tic-OH, a delta selective opioid dipeptide antagonist
file con accesso da definire2000 Monory, K; Bryant, Sd; Kertesz, I; Balboni, Gianfranco; Guerrini, Remo; Toth, G; Salvadori, Severo; Lazarus, Lh; Borsodi, A.
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei
2000 Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Bianchi, C; Santagada, V; Calliendo, G; Bryant, Sd; Lazarus, Lh
Inverse agonism by Dmt-Tic analogues and H5 378, a naltrindole analogue
file con accesso da definire2000 Labarre, M; Butterworth, J; ST ONGE, S; Payza, K; Schmidhammer, H; Salvadori, Severo; Balboni, Gianfranco; Guerrini, Remo; Bryant, Sd; Lazarus, Lh
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues
file con accesso da definire2000 Santagada, V; Balboni, Gianfranco; Caliendo, G; Guerrini, Remo; Salvadori, Severo; Bianchi, C; Bryant, Sd; Lazarus, Lh
Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders.
file con accesso da definire2001 Baraldi, Pier Giovanni; Balboni, Gianfranco; Pavani, Maria Giovanna; Spalluto, Giampiero; AGHAZADEH TABRIZI, Mojgan; DE CLERCQ, Erik; Balzarini, Jan; Bando, Toshikazu; Sugiyama, Hiroshi; Romagnoli, Romeo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, metabolic stability and chemotactic activity of peptide T and its analogues | 1990 | Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Spisani, Susanna; Gavioli, Riccardo; Tr...aniello, Maria Serena; Tomatis, Roberto | file con accesso da definire |
A CYCLIC PEPTIDE T ANALOGUE WITH HIGH CHEMOTACTIC ACTIVITY | 1992 | Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Scaranari, V.; Spisani, Susanna; Reali,... Eva; Giuliani, Anna Lisa; Tomatis, Roberto | file con accesso da definire |
Conformational analysis of potent and very selective delta opioid dipeptide antagonists | 1995 | Amodeo, P; Balboni, Gianfranco; Crescenzi, O; Guerrini, Remo; Picone, D; Salvadori, Severo; Tancr...edi, T; Temussi, Pa | file con accesso da definire |
Acid catalysis in the formation of dioxopiperazines from peptides containing tetrahydroisoquinoline‐3‐carboxylic acid at position 2 | 1995 | Capasso, S; Sica, F; Mazzarella, L; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo | file con accesso da definire |
DMT-TIC-OH, a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse | 1996 | Capasso, A; Guerrini, Remo; Balboni, Gianfranco; Sorrentino, L; Temussi, P; Lazarus, Lh; Bryant, ...Sd; Salvadori, Severo | file con accesso da definire |
Opioid diketopiperazines: Refinement of the delta opioid antagonist pharmacophore | 1997 | Bryant, Sd; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Lazarus, Lh | file con accesso da definire |
Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary δ opioid antagonist activity | 1997 | Salvadori, Severo; Balboni, Gianfranco; Guerrini, Remo; Tomatis, R; Bianchi, C; Bryant, Sd; Coope...r, Ps; Lazarus, Lh | file con accesso da definire |
Design and solution structure of a partially rigid opioid antagonist lacking the basic center - Models of antagonism | 1997 | Crescenzi, O; Fraternali, F; Picone, D; Tancredi, T; Balboni, Gianfranco; Guerrini, Remo; Lazarus..., Lh; Salvadori, Severo; Temussi, Pa | file con accesso da definire |
Design of μ selective opioid dipeptide antagonists | 1997 | Capasso, A; Amodeo, P; Balboni, Gianfranco; Guerrini, Remo; Lazarus, Lh; Temussi, Pa; Salvadori, ...Severo | file con accesso da definire |
Opioid diketopiperazines: Synthesis and activity of a prototypic class of opioid antagonists | 1997 | Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Bryant, Sd; Bianchi, C; Attil...a, M; Lazarus, Lh | file con accesso da definire |
Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides | 1997 | Tomatis, R; Marastoni, Mauro; Balboni, Gianfranco; Guerrini, Remo; Capasso, A; Sorrentino, L; San...tagada, V; Caliendo, G; Lazarus, Lh; Salvadori, Severo | file con accesso da definire |
Design of d-opioid peptide antagonists for emerging drug applications | 1998 | L. H., Lazarus; S. n. D., Bryant; P. S., Cooper; Guerrini, Remo; Balboni, Gianfranco; Salvadori, ...Severo | file con accesso da definire |
Tritiation of delta opioid-receptor selective antagonist dipeptide ligands with extraordinary affinity containing 2 ', 6 ' dimethyltyrosine | 1999 | Kertesz, I; Toth, G; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo | file con accesso da definire |
Further Studies on the Dmt-Tic Pharmacophore: Hydrophobic Substituents at the C-Terminus Endow delta Antagonists To Manifest mu Agonism or mu Antagonism | 1999 | Salvadori, Severo; Guerrini, Remo; Balboni, Gianfranco; C., Bianchi; S. D., Bryant; P. S., Cooper...; L. H., Lazarus | file con accesso da definire |
Synthesis, in vitro antiproliferative activity, and DNA-binding properties of hybrid molecules containing pyrrolo[2,1-c][1,4] benzodiazepine and minor-groove-binding oligopyrrole carriers | 1999 | Baraldi, Pier Giovanni; Balboni, Gianfranco; Cacciari, Barbara; A., Guiotto; Manfredini, Stefano;... Romagnoli, Romeo; Spalluto, Giampiero; D. E., Thurston; P. W., Howard; Bianchi, Nicoletta; Rutigliano, Cristina; Mischiati, Carlo; Gambari, Roberto | file con accesso da definire |
Characterization of N,N(Me)(2)-Dmt-Tic-OH, a delta selective opioid dipeptide antagonist | 2000 | Monory, K; Bryant, Sd; Kertesz, I; Balboni, Gianfranco; Guerrini, Remo; Toth, G; Salvadori, Sever...o; Lazarus, Lh; Borsodi, A. | file con accesso da definire |
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei | 2000 | Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Bianchi, C; Santagada, V; Calliendo, G; B...ryant, Sd; Lazarus, Lh | |
Inverse agonism by Dmt-Tic analogues and H5 378, a naltrindole analogue | 2000 | Labarre, M; Butterworth, J; ST ONGE, S; Payza, K; Schmidhammer, H; Salvadori, Severo; Balboni, Gi...anfranco; Guerrini, Remo; Bryant, Sd; Lazarus, Lh | file con accesso da definire |
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues | 2000 | Santagada, V; Balboni, Gianfranco; Caliendo, G; Guerrini, Remo; Salvadori, Severo; Bianchi, C; Br...yant, Sd; Lazarus, Lh | file con accesso da definire |
Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders. | 2001 | Baraldi, Pier Giovanni; Balboni, Gianfranco; Pavani, Maria Giovanna; Spalluto, Giampiero; AGHAZAD...EH TABRIZI, Mojgan; DE CLERCQ, Erik; Balzarini, Jan; Bando, Toshikazu; Sugiyama, Hiroshi; Romagnoli, Romeo | file con accesso da definire |
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