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Titolo Data di pubblicazione Autore(i) File
Synthesis, metabolic stability and chemotactic activity of peptide T and its analogues 1990 Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Spisani, Susanna; Gavioli, Riccardo; Tr...aniello, Maria Serena; Tomatis, Roberto file con accesso da definire
A CYCLIC PEPTIDE T ANALOGUE WITH HIGH CHEMOTACTIC ACTIVITY 1992 Marastoni, Mauro; Salvadori, Severo; Balboni, Gianfranco; Scaranari, V.; Spisani, Susanna; Reali,... Eva; Giuliani, Anna Lisa; Tomatis, Roberto file con accesso da definire
Conformational analysis of potent and very selective delta opioid dipeptide antagonists 1995 Amodeo, P; Balboni, Gianfranco; Crescenzi, O; Guerrini, Remo; Picone, D; Salvadori, Severo; Tancr...edi, T; Temussi, Pa file con accesso da definire
Acid catalysis in the formation of dioxopiperazines from peptides containing tetrahydroisoquinoline‐3‐carboxylic acid at position 2 1995 Capasso, S; Sica, F; Mazzarella, L; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo file con accesso da definire
DMT-TIC-OH, a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse 1996 Capasso, A; Guerrini, Remo; Balboni, Gianfranco; Sorrentino, L; Temussi, P; Lazarus, Lh; Bryant, ...Sd; Salvadori, Severo file con accesso da definire
Design and solution structure of a partially rigid opioid antagonist lacking the basic center - Models of antagonism 1997 Crescenzi, O; Fraternali, F; Picone, D; Tancredi, T; Balboni, Gianfranco; Guerrini, Remo; Lazarus..., Lh; Salvadori, Severo; Temussi, Pa file con accesso da definire
Opioid diketopiperazines: Synthesis and activity of a prototypic class of opioid antagonists 1997 Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Bryant, Sd; Bianchi, C; Attil...a, M; Lazarus, Lh file con accesso da definire
Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary δ opioid antagonist activity 1997 Salvadori, Severo; Balboni, Gianfranco; Guerrini, Remo; Tomatis, R; Bianchi, C; Bryant, Sd; Coope...r, Ps; Lazarus, Lh file con accesso da definire
Opioid diketopiperazines: Refinement of the delta opioid antagonist pharmacophore 1997 Bryant, Sd; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo; Tomatis, R; Lazarus, Lh file con accesso da definire
Design of μ selective opioid dipeptide antagonists 1997 Capasso, A; Amodeo, P; Balboni, Gianfranco; Guerrini, Remo; Lazarus, Lh; Temussi, Pa; Salvadori, ...Severo file con accesso da definire
Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides 1997 Tomatis, R; Marastoni, Mauro; Balboni, Gianfranco; Guerrini, Remo; Capasso, A; Sorrentino, L; San...tagada, V; Caliendo, G; Lazarus, Lh; Salvadori, Severo file con accesso da definire
Design of d-opioid peptide antagonists for emerging drug applications 1998 L. H., Lazarus; S. n. D., Bryant; P. S., Cooper; Guerrini, Remo; Balboni, Gianfranco; Salvadori, ...Severo file con accesso da definire
Tritiation of delta opioid-receptor selective antagonist dipeptide ligands with extraordinary affinity containing 2 ', 6 ' dimethyltyrosine 1999 Kertesz, I; Toth, G; Balboni, Gianfranco; Guerrini, Remo; Salvadori, Severo file con accesso da definire
Further Studies on the Dmt-Tic Pharmacophore: Hydrophobic Substituents at the C-Terminus Endow delta Antagonists To Manifest mu Agonism or mu Antagonism 1999 Salvadori, Severo; Guerrini, Remo; Balboni, Gianfranco; C., Bianchi; S. D., Bryant; P. S., Cooper...; L. H., Lazarus file con accesso da definire
Synthesis, in vitro antiproliferative activity, and DNA-binding properties of hybrid molecules containing pyrrolo[2,1-c][1,4] benzodiazepine and minor-groove-binding oligopyrrole carriers 1999 Baraldi, Pier Giovanni; Balboni, Gianfranco; Cacciari, Barbara; A., Guiotto; Manfredini, Stefano;... Romagnoli, Romeo; Spalluto, Giampiero; D. E., Thurston; P. W., Howard; Bianchi, Nicoletta; Rutigliano, Cristina; Mischiati, Carlo; Gambari, Roberto file con accesso da definire
Inverse agonism by Dmt-Tic analogues and H5 378, a naltrindole analogue 2000 Labarre, M; Butterworth, J; ST ONGE, S; Payza, K; Schmidhammer, H; Salvadori, Severo; Balboni, Gi...anfranco; Guerrini, Remo; Bryant, Sd; Lazarus, Lh file con accesso da definire
Characterization of N,N(Me)(2)-Dmt-Tic-OH, a delta selective opioid dipeptide antagonist 2000 Monory, K; Bryant, Sd; Kertesz, I; Balboni, Gianfranco; Guerrini, Remo; Toth, G; Salvadori, Sever...o; Lazarus, Lh; Borsodi, A. file con accesso da definire
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues 2000 Santagada, V; Balboni, Gianfranco; Caliendo, G; Guerrini, Remo; Salvadori, Severo; Bianchi, C; Br...yant, Sd; Lazarus, Lh file con accesso da definire
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei 2000 Balboni, Gianfranco; Salvadori, Severo; Guerrini, Remo; Bianchi, C; Santagada, V; Calliendo, G; B...ryant, Sd; Lazarus, Lh
Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders. 2001 Baraldi, Pier Giovanni; Balboni, Gianfranco; Pavani, Maria Giovanna; Spalluto, Giampiero; AGHAZAD...EH TABRIZI, Mojgan; DE CLERCQ, Erik; Balzarini, Jan; Bando, Toshikazu; Sugiyama, Hiroshi; Romagnoli, Romeo file con accesso da definire
Mostrati risultati da 1 a 20 di 31
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