Sfoglia per Autore
Acute and chronic antiparkinsonian effects of the novel nociceptin/orphanin FQ receptor antagonist NiK-21273 in comparison with SB-612111
file con accesso da definire2013 Marti, Matteo; Mela, Flora; Budri, Mirco; Volta, Mattia; Malfacini, Davide; Molinari, Stefano; N. T., Zaveri; S., Ronzoni; P., Petrillo; Calo', Girolamo; Morari, Michele
[D-Pen(p-tBuBzl)5]NPS, a novel ligand for the neuropeptide S receptor: structure activity and pharmacological studies
file con accesso da definire2014 Ruzza, Chiara; L., del Zoppo; Malfacini, Davide; Pela', Michela; Trapella, Claudio; P., Grieco; Salvadori, Severo; Calo', Girolamo; Guerrini, Remo
Pharmacological characterization of tachykinin tetrabranched derivatives
file con accesso da definire2014 Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Cerlesi, Maria Camilla; Ferrari, Federica; Marzola, Erika; Caterina, Ambrosio; Cristina, Gro; Salvadori, Severo; Tommaso, Costa; Calo', Girolamo; Guerrini, Remo
In vitro and in vivo pharmacological characterization of nociceptin/orphanin FQ tetrabranched derivatives
file con accesso da definire2014 Rizzi, Anna; Malfacini, Davide; Cerlesi, Maria Camilla; Ruzza, Chiara; Marzola, Erika; M. F., Bird; D. J., Rowbotham; Salvadori, Severo; Guerrini, Remo; D. G., Lambert; Calo', Girolamo
Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues
file con accesso da definire2014 Renata, Perlikowska; Malfacini, Davide; Cerlesi, Maria Camilla; Calo', Girolamo; Justyna, Piekielna; Léonore, Floriot; Tiphaine, Henry; Jean Claude do, Rego; Csaba, Tömböly; Alicja, Kluczyk; Anna, Janecka
A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.
file con accesso da definire2014 Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pela', Michela; Molinari, Stefano; Cerlesi, Maria Camilla; Malfacini, Davide; Rizzi, Anna; Salvadori, Severo; Calo', Girolamo
Synthesis, enantiomeric separation and docking studies of spiropiperidine analogues as ligands of the nociceptin/orphanin FQ receptor
file con accesso da definire2014 Umberto M., Battisti; Sandra, Corrado; Claudia, Sorbi; Andrea, Cornia; Annalisa, Tait; Malfacini, Davide; Cerlesi, Maria Camilla; Calo', Girolamo; Livio, Brasili
Pharmacological Investigations of N-Substituent Variation in Morphine and Oxymorphone: Opioid Receptor Binding, Signaling and Antinociceptive Activity
file con accesso da definire2014 Ben Haddou, T; Béni, S; Hosztafi, S; Malfacini, Davide; Calo', Girolamo; Schmidhammer, H; Spetea, M.
1,4-Dioxolane-triazaspirodecanone derivatives as nociceptin/orphanin FQ receptor ligands
file con accesso da definire2014 S., Corrado; C., Sorbi; A., Tait; U. M., Battisti; Camarda, Valeria; Malfacini, Davide; Calo', Girolamo; L., Brasili
Exploring pharmacological activities and signaling of morphinans substituted in position 6 as potent agonists interacting with the μ opioid receptor
file con accesso da definire2014 Tanila Ben, Haddou; Malfacini, Davide; Calo', Girolamo; Mario D., Aceto; Louis S., Harris; John R., Traynor; Andrew, Coop; Helmut, Schmidhammer; Mariana, Spetea
Novel ligands and assays for nociceptin/orphanin FQ and classical opioid receptors
2015 Malfacini, Davide
The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled Receptor
2015 Miller, Rebecca L.; Thompson, Aaron A.; Trapella, Claudio; Guerrini, Remo; Malfacini, Davide; Patel, Nilkanth; Han, Gye Won; Cherezov, Vadim; Calo', Girolamo; Katritch, Vsevolod; Stevens, Raymond C.
Pharmacological profile of nociceptin/orphanin FQ receptors interacting with G-proteins and β-arrestins 2
2015 Malfacini, Davide; Ambrosio, C.; Gro', M. C.; Sbraccia, M.; Trapella, Claudio; Guerrini, Remo; Bonora, Massimo; Pinton, Paolo; Costa, T.; Calo', Girolamo
In vitro and in vivo pharmacological characterization of a neuropeptide S tetrabranched derivative
file con accesso da definire2015 Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Pulga, Alice; Pacifico, Salvatore; Salvadori, Severo; Trapella, Claudio; Reinscheid, Rainer K; Calo', Girolamo; Guerrini, Remo
In vitro and in vivo pharmacological characterization of Pronetupitant, a prodrug of the neurokinin 1 receptor antagonist Netupitant
file con accesso da definire2015 Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Molinari, Stefano; Giuliano, Claudio; Lovati, Emanuela; Pietra, Claudio; Calo', Girolamo
Synthesis and Structure–Activity Relationships of Triazaspirodecanone Derivatives as Nociceptin/Orphanin FQ Receptor Ligands
file con accesso da definire2015 Corrado, S; Battisti, Um; Sorbi, C; Tait, A; Malfacini, Davide; Camarda, Valeria; Calo', Girolamo; Brasili, L. 1.
In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations
file con accesso da definire2016 Ferrari, Federica; Cerlesi, Maria Camilla; Malfacini, Davide; Asth, Laila; Gavioli, Elaine C; Journigan, Blair V; Kamakolanu, Uma Gayathri; Meyer, Michael E; Yasuda, Dennis; Polgar, Willma E; Rizzi, Anna; Guerrini, Remo; Ruzza, Chiara; Zaveri, Nurulain T; Calo', Girolamo
Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist
file con accesso da definire2016 Rizzi, Anna; Cerlesi, Maria Camilla; Ruzza, Chiara; Malfacini, Davide; Ferrari, Federica; Bianco, Sara; Costa, Tommaso; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo
Characterisation of the novel mixed Mu-NOP peptide ligand dermorphin-N/OFQ (DeNo)
2016 Bird, Mark F.; Camilla Cerlesi, Maria; Brown, Mark; Malfacini, Davide; Vezzi, Vanessa; Molinari, Paola; Micheli, Laura; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Guerrini, Remo; Calo', Girolamo; Lambert, David G.
Beta-arrestin 2 rather than G protein efficacy determines the anxiolytic- versus antidepressant-like effects of nociceptin/orphanin FQ receptor ligands
2016 Asth, L; Ruzza, Chiara; Malfacini, Davide; Medeiros, I; Guerrini, Remo; Zaveri, N. T; Gavioli, E. C; Calo', Girolamo
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Acute and chronic antiparkinsonian effects of the novel nociceptin/orphanin FQ receptor antagonist NiK-21273 in comparison with SB-612111 | 2013 | Marti, Matteo; Mela, Flora; Budri, Mirco; Volta, Mattia; Malfacini, Davide; Molinari, Stefano; N.... T., Zaveri; S., Ronzoni; P., Petrillo; Calo', Girolamo; Morari, Michele | file con accesso da definire |
| [D-Pen(p-tBuBzl)5]NPS, a novel ligand for the neuropeptide S receptor: structure activity and pharmacological studies | 2014 | Ruzza, Chiara; L., del Zoppo; Malfacini, Davide; Pela', Michela; Trapella, Claudio; P., Grieco; S...alvadori, Severo; Calo', Girolamo; Guerrini, Remo | file con accesso da definire |
| Pharmacological characterization of tachykinin tetrabranched derivatives | 2014 | Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Cerlesi, Maria Camilla; Ferrari, Federica; Marzola..., Erika; Caterina, Ambrosio; Cristina, Gro; Salvadori, Severo; Tommaso, Costa; Calo', Girolamo; Guerrini, Remo | file con accesso da definire |
| In vitro and in vivo pharmacological characterization of nociceptin/orphanin FQ tetrabranched derivatives | 2014 | Rizzi, Anna; Malfacini, Davide; Cerlesi, Maria Camilla; Ruzza, Chiara; Marzola, Erika; M. F., Bir...d; D. J., Rowbotham; Salvadori, Severo; Guerrini, Remo; D. G., Lambert; Calo', Girolamo | file con accesso da definire |
| Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues | 2014 | Renata, Perlikowska; Malfacini, Davide; Cerlesi, Maria Camilla; Calo', Girolamo; Justyna, Piekiel...na; Léonore, Floriot; Tiphaine, Henry; Jean Claude do, Rego; Csaba, Tömböly; Alicja, Kluczyk; Anna, Janecka | file con accesso da definire |
| A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ. | 2014 | Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pela', Michela; Molinari, Stefano; Cerlesi, Ma...ria Camilla; Malfacini, Davide; Rizzi, Anna; Salvadori, Severo; Calo', Girolamo | file con accesso da definire |
| Synthesis, enantiomeric separation and docking studies of spiropiperidine analogues as ligands of the nociceptin/orphanin FQ receptor | 2014 | Umberto M., Battisti; Sandra, Corrado; Claudia, Sorbi; Andrea, Cornia; Annalisa, Tait; Malfacini,... Davide; Cerlesi, Maria Camilla; Calo', Girolamo; Livio, Brasili | file con accesso da definire |
| Pharmacological Investigations of N-Substituent Variation in Morphine and Oxymorphone: Opioid Receptor Binding, Signaling and Antinociceptive Activity | 2014 | Ben Haddou, T; Béni, S; Hosztafi, S; Malfacini, Davide; Calo', Girolamo; Schmidhammer, H; Spetea, M. | file con accesso da definire |
| 1,4-Dioxolane-triazaspirodecanone derivatives as nociceptin/orphanin FQ receptor ligands | 2014 | S., Corrado; C., Sorbi; A., Tait; U. M., Battisti; Camarda, Valeria; Malfacini, Davide; Calo', Gi...rolamo; L., Brasili | file con accesso da definire |
| Exploring pharmacological activities and signaling of morphinans substituted in position 6 as potent agonists interacting with the μ opioid receptor | 2014 | Tanila Ben, Haddou; Malfacini, Davide; Calo', Girolamo; Mario D., Aceto; Louis S., Harris; John R...., Traynor; Andrew, Coop; Helmut, Schmidhammer; Mariana, Spetea | file con accesso da definire |
| Novel ligands and assays for nociceptin/orphanin FQ and classical opioid receptors | 2015 | Malfacini, Davide | |
| The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled Receptor | 2015 | Miller, Rebecca L.; Thompson, Aaron A.; Trapella, Claudio; Guerrini, Remo; Malfacini, Davide; Pat...el, Nilkanth; Han, Gye Won; Cherezov, Vadim; Calo', Girolamo; Katritch, Vsevolod; Stevens, Raymond C. | |
| Pharmacological profile of nociceptin/orphanin FQ receptors interacting with G-proteins and β-arrestins 2 | 2015 | Malfacini, Davide; Ambrosio, C.; Gro', M. C.; Sbraccia, M.; Trapella, Claudio; Guerrini, Remo; Bo...nora, Massimo; Pinton, Paolo; Costa, T.; Calo', Girolamo | |
| In vitro and in vivo pharmacological characterization of a neuropeptide S tetrabranched derivative | 2015 | Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Pulga, Alice; Pacifico, Salvatore; Salvadori, Seve...ro; Trapella, Claudio; Reinscheid, Rainer K; Calo', Girolamo; Guerrini, Remo | file con accesso da definire |
| In vitro and in vivo pharmacological characterization of Pronetupitant, a prodrug of the neurokinin 1 receptor antagonist Netupitant | 2015 | Ruzza, Chiara; Rizzi, Anna; Malfacini, Davide; Molinari, Stefano; Giuliano, Claudio; Lovati, Eman...uela; Pietra, Claudio; Calo', Girolamo | file con accesso da definire |
| Synthesis and Structure–Activity Relationships of Triazaspirodecanone Derivatives as Nociceptin/Orphanin FQ Receptor Ligands | 2015 | Corrado, S; Battisti, Um; Sorbi, C; Tait, A; Malfacini, Davide; Camarda, Valeria; Calo', Girolamo...; Brasili, L. 1. | file con accesso da definire |
| In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations | 2016 | Ferrari, Federica; Cerlesi, Maria Camilla; Malfacini, Davide; Asth, Laila; Gavioli, Elaine C; Jou...rnigan, Blair V; Kamakolanu, Uma Gayathri; Meyer, Michael E; Yasuda, Dennis; Polgar, Willma E; Rizzi, Anna; Guerrini, Remo; Ruzza, Chiara; Zaveri, Nurulain T; Calo', Girolamo | file con accesso da definire |
| Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist | 2016 | Rizzi, Anna; Cerlesi, Maria Camilla; Ruzza, Chiara; Malfacini, Davide; Ferrari, Federica; Bianco,... Sara; Costa, Tommaso; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo | file con accesso da definire |
| Characterisation of the novel mixed Mu-NOP peptide ligand dermorphin-N/OFQ (DeNo) | 2016 | Bird, Mark F.; Camilla Cerlesi, Maria; Brown, Mark; Malfacini, Davide; Vezzi, Vanessa; Molinari, ...Paola; Micheli, Laura; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Guerrini, Remo; Calo', Girolamo; Lambert, David G. | |
| Beta-arrestin 2 rather than G protein efficacy determines the anxiolytic- versus antidepressant-like effects of nociceptin/orphanin FQ receptor ligands | 2016 | Asth, L; Ruzza, Chiara; Malfacini, Davide; Medeiros, I; Guerrini, Remo; Zaveri, N. T; Gavioli, E.... C; Calo', Girolamo |
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