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N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor 2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Saponaro,... Giulia; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea file con accesso da definire
Structure-activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A(3) adenosine receptor antagonists. 2008 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Botta, M; Bernardini, C; Tafi, A; Tuccinardi, T; Martinelli, A; Varani, Katia; Borea, Pier Andrea file con accesso da definire
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists 2008 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea file con accesso da definire
Design and Synthesis of New A2A and A3 Adenosine Receptors Antagonists 2009 Saponaro, Giulia
A3 adenosine receptor antagonists: History and future perspectives 2010 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Tabrizi, Mojgan Ag...hazadeh; Preti, Delia file con accesso da definire
New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A 3 adenosine receptor antagonists 2011 Baraldi, Pier Giovanni; Preti, Delia; Zaid, Na; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Bara...ldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Varani, Katia; Cosconati, S; Di Maro, S; Marinelli, L; Novellino, E; Borea, Pier Andrea file con accesso da definire
Water-Soluble Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines as Human A3 Adenosine Receptor Antagonists 2012 Baraldi, Pier Giovanni; Saponaro, Giulia; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Baraldi, S...tefania; A. R., Moorman; S., Cosconati; S., Di Maro; L., Marinelli; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea; Preti, Delia file con accesso da definire
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation 2012 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, S...tefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists 2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
Novel 1,3-Dipropyl-8-(3-benzimidazol-2-yl-methoxy-1-methylpyrazol-5-yl)xanthines as Potent and Selective A2B Adenosine Receptor Antagonists 2012 Baraldi, Pier Giovanni; Baraldi, Stefania; Saponaro, Giulia; Preti, Delia; Romagnoli, Romeo; Picc...agli, Laura; Cavalli, A; Recanatini, M; Moorman, Ar; Zaid, An; Varani, Katia; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan file con accesso da definire
Pyrrolo- and pyrazolo-[3,4-e][1,2,4]triazolo[1,5-c]pyrimidines as adenosine receptor antagonists 2012 Baraldi, Pier Giovanni; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Romagnoli..., Romeo; Moorman A., R; Varani, Katia; Borea, Pier Andrea; Preti, Delia file con accesso da definire
Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists 2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, R...omeo; Preti, Delia; Baraldi, Stefania; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia file con accesso da definire
Antinociceptive effects of the selective CB2 agonist MT178 in inflammatory and chronic rodent pain models. 2013 Vincenzi, Fabrizio; Targa, Martina; Corciulo, Carmen; AGHAZADEH TABRIZI, Mojgan; Merighi, Stefani...a; Gessi, Stefania; Saponaro, Giulia; Baraldi, Pier Giovanni; Borea, Pier Andrea; Varani, Katia file con accesso da definire
Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists. 2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; Moorman, Ar; Romagnoli, Rome...o; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Tintori, C; Tuccinardi, T; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia file con accesso da definire
Synthesis and Biological Evaluation of Novel 2-Amino-3-Aroyl-4-Neopentyl-5-Substituted Thiophene Derivatives as Allosteric Enhancers of the A1 Adenosine Receptor 2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Kimatra...i Salvador, M.; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Moorman, A. R.; Vincenzi, Fabrizio; Borea, A. P.; Varani, Katia file con accesso da definire
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene 2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; A. P., Ijzerman; A., Massink; O., Cruz Lopez; L. C., Lo...pez Cara; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; A. R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia file con accesso da definire
Transient receptor potential ankyrin 1 (TRPA1) antagonists 2015 Preti, Delia; Saponaro, Giulia; Szallasi, Arpad file con accesso da definire
One-pot reaction to obtain N,N'-disubstituted guanidines of pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine scaffold as human A3 adenosine receptor antagonists 2015 Baraldi, Pier Giovanni; Baraldi, Stefania; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Romagnoli..., Romeo; Ruggiero, Emanuela; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor 2015 Preti, Delia; Baraldi, Pier Giovanni; Saponaro, Giulia; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojg...an; Baraldi, Stefania; Cosconati, Sandro; Bruno, Agostino; Novellino, Ettore; Vincenzi, Fabrizio; Ravani, Annalisa; Borea, Pier Andrea; Varani, Katia
Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors 2015 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, D...elia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J. file con accesso da definire
Mostrati risultati da 1 a 20 di 23
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