Sfoglia per Autore
Neuropeptide S reduces mouse aggressiveness in the resident/intruder test through selective activation of the neuropeptide S receptor
2015 Ruzza, C; Asth, L; Guerrini, R; Trapella, C; Gavioli, E
JWH-018 impairs sensorimotor functions in mice
2015 Ossato, Andrea; Vigolo, A; Trapella, Claudio; Seri, C; Rimondo, C; Serpelloni, G; Marti, Matteo
Intrathecal administration of nociceptin/orphanin FQ receptor agonists in rats: A strategy to relieve chemotherapy-induced neuropathic hypersensitivity
file con accesso da definire2015 Micheli, Laura; Di Cesare Mannelli, Lorenzo; Rizzi, Anna; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo; Ghelardini, Carla
The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled Receptor
2015 Miller, Rebecca L.; Thompson, Aaron A.; Trapella, Claudio; Guerrini, Remo; Malfacini, Davide; Patel, Nilkanth; Han, Gye Won; Cherezov, Vadim; Calo', Girolamo; Katritch, Vsevolod; Stevens, Raymond C.
Physicochemical stability of cabazitaxel and docetaxel solutions
file con accesso da definire2015 Renzo, Lazzarini; Salvadori, Severo; Trapella, Claudio; Guerrini, Remo; Marzola, Erika; Giada, Pasini; Dalpiaz, Alessandro
Structure activity studies of nociceptin/orphanin FQ(1–13)-NH2 derivatives modified in position 5
2015 Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pacifico, Salvatore; Malfacini, Maria Camilla Cerlesi Davide; Ferrari, Federica; Bird, Mark Francis; Lambert, David George; Salvadori, Severo; Calo', Girolamo
Development and characterisation of novel fentanyl-delta opioid receptor antagonist based bivalent ligands
file con accesso da definire2015 Bird, Mf; Vardanyan, Rs; Hruby, Vj; Calo', Girolamo; Guerrini, Remo; Salvadori, Severo; Trapella, Claudio; Mcdonald, J; Rowbotham, Dj; Lambert, Dg
Novel halogenated derivates of JWH-018: Behavioral and binding studies in mice
2015 A., Vigolo; Ossato, Andrea; Trapella, Claudio; Vincenzi, Fabrizio; C., Rimondo; C., Seri; Varani, Katia; G., Serpelloni; Marti, Matteo
Letter to the Editor: Antimicrobial properties of mucus from the brown garden snail Helix aspersa
file con accesso da definire2016 Bortolotti, Daria; Trapella, Claudio; Bernardi, Tatiana; Rizzo, Roberta
Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist
file con accesso da definire2016 Rizzi, Anna; Cerlesi, Maria Camilla; Ruzza, Chiara; Malfacini, Davide; Ferrari, Federica; Bianco, Sara; Costa, Tommaso; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo
Studies of C-terminal naphthoquinone dipeptides as 20S proteasome inhibitors
2016 Scotti, A; Trapella, Claudio; Ferretti, Valeria; Gallerani, Eleonora; Gavioli, Riccardo; Marastoni, Mauro
Design, synthesis and biological characterization of novel mitochondria targeted dichloroacetate-loaded compounds with antileukemic activity
2016 Trapella, Claudio; Voltan, Rebecca; Melloni, Elisabetta; Tisato, Veronica; Celeghini, C; Bianco, Sara; Fantinati, Anna; Salvadori, Severo; Guerrini, Remo; Secchiero, Paola; Zauli, Giorgio
Synthetic cannabinoid JWH-018 and its halogenated derivatives JWH-018-Cl and JWH-018-Br impair Novel Object Recognition in mice: Behavioral, electrophysiological and neurochemical evidence
2016 Barbieri, Mario; Ossato, Andrea; Canazza, Isabella; Trapella, Claudio; Borelli, Andrea Celeste; Beggiato, Sarah; Rimondo, C; Serpelloni, G; Ferraro, Luca Nicola; Marti, Matteo
Effect of the novel synthetic cannabinoids AKB48 and 5F-AKB48 on “tetrad”, sensorimotor, neurological and neurochemical responses in mice. In vitro and in vivo pharmacological studies
2016 Canazza, Isabella; Ossato, Andrea; Trapella, Claudio; Fantinati, Anna; de Luca, Maria Antonietta; Margiani, Giulia; Vincenzi, Fabrizio; Rimondo, Claudia; Di Rosa, Fabiana; Gregori, Adolfo; Varani, Katia; Borea, Pier Andrea; Serpelloni, Giovanni; Marti, Matteo
Effect of JWH-250, JWH-073 and their interaction on “tetrad”, sensorimotor, neurological and neurochemical responses in mice
2016 Ossato, Andrea; Canazza, Isabella; Trapella, Claudio; Vincenzi, Fabrizio; De Luca, Maria Antonietta; Rimondo, Claudia; Varani, Katia; Borea, Pier Andrea; Serpelloni, Giovanni; Marti, Matteo
Structure-and conformation-Activity studies of nociceptin/orphanin FQ receptor dimeric ligands
2017 Pacifico, Salvatore; Carotenuto, Alfonso; Brancaccio, Diego; Novellino, Ettore; Marzola, Erika; Ferrari, Federica; Cerlesi, Maria Camilla; Trapella, Claudio; Preti, Delia; Salvadori, Severo; Calo', Girolamo; Guerrini, Remo
1‐cyclohexyl‐x‐methoxybenzene derivatives, novel psychoactive substances seized on the internet market. Synthesis and in vivo pharmacological studies in mice
2017 Fantinati, Anna; Ossato, Andrea; Bianco, Sara; Canazza, Isabella; De Giorgio, F; Trapella, Claudio; Marti, Matteo
Antinociceptive action of NOP and opioid receptor agonists in the mouse orofacial formalin test
file con accesso da definire2017 Rizzi, Anna; Ruzza, Chiara; Bianco, Sara; Trapella, Claudio; Calo', Girolamo
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism
2017 Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, Maria Camilla; Trapella, Claudio; Calo', Girolamo
Expeditious Synthesis and Biological Characterization of Enantio-Enriched (-)-Nutlin-3
2017 Fantinati, Anna; Bianco, Sara; Cristofori, Virginia; Cavazzini, Alberto; Catani, Martina; Zanirato, Vinicio; Pacifico, Salvatore; Rimondi, Erika; Milani, Daniela; Voltan, Rebecca; Secchiero, Paola; Trapella, Claudio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Neuropeptide S reduces mouse aggressiveness in the resident/intruder test through selective activation of the neuropeptide S receptor | 2015 | Ruzza, C; Asth, L; Guerrini, R; Trapella, C; Gavioli, E | |
JWH-018 impairs sensorimotor functions in mice | 2015 | Ossato, Andrea; Vigolo, A; Trapella, Claudio; Seri, C; Rimondo, C; Serpelloni, G; Marti, Matteo | |
Intrathecal administration of nociceptin/orphanin FQ receptor agonists in rats: A strategy to relieve chemotherapy-induced neuropathic hypersensitivity | 2015 | Micheli, Laura; Di Cesare Mannelli, Lorenzo; Rizzi, Anna; Guerrini, Remo; Trapella, Claudio; Calo...', Girolamo; Ghelardini, Carla | file con accesso da definire |
The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled Receptor | 2015 | Miller, Rebecca L.; Thompson, Aaron A.; Trapella, Claudio; Guerrini, Remo; Malfacini, Davide; Pat...el, Nilkanth; Han, Gye Won; Cherezov, Vadim; Calo', Girolamo; Katritch, Vsevolod; Stevens, Raymond C. | |
Physicochemical stability of cabazitaxel and docetaxel solutions | 2015 | Renzo, Lazzarini; Salvadori, Severo; Trapella, Claudio; Guerrini, Remo; Marzola, Erika; Giada, Pa...sini; Dalpiaz, Alessandro | file con accesso da definire |
Structure activity studies of nociceptin/orphanin FQ(1–13)-NH2 derivatives modified in position 5 | 2015 | Guerrini, Remo; Marzola, Erika; Trapella, Claudio; Pacifico, Salvatore; Malfacini, Maria Camilla ...Cerlesi Davide; Ferrari, Federica; Bird, Mark Francis; Lambert, David George; Salvadori, Severo; Calo', Girolamo | |
Development and characterisation of novel fentanyl-delta opioid receptor antagonist based bivalent ligands | 2015 | Bird, Mf; Vardanyan, Rs; Hruby, Vj; Calo', Girolamo; Guerrini, Remo; Salvadori, Severo; Trapella,... Claudio; Mcdonald, J; Rowbotham, Dj; Lambert, Dg | file con accesso da definire |
Novel halogenated derivates of JWH-018: Behavioral and binding studies in mice | 2015 | A., Vigolo; Ossato, Andrea; Trapella, Claudio; Vincenzi, Fabrizio; C., Rimondo; C., Seri; Varani,... Katia; G., Serpelloni; Marti, Matteo | |
Letter to the Editor: Antimicrobial properties of mucus from the brown garden snail Helix aspersa | 2016 | Bortolotti, Daria; Trapella, Claudio; Bernardi, Tatiana; Rizzo, Roberta | file con accesso da definire |
Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist | 2016 | Rizzi, Anna; Cerlesi, Maria Camilla; Ruzza, Chiara; Malfacini, Davide; Ferrari, Federica; Bianco,... Sara; Costa, Tommaso; Guerrini, Remo; Trapella, Claudio; Calo', Girolamo | file con accesso da definire |
Studies of C-terminal naphthoquinone dipeptides as 20S proteasome inhibitors | 2016 | Scotti, A; Trapella, Claudio; Ferretti, Valeria; Gallerani, Eleonora; Gavioli, Riccardo; Maraston...i, Mauro | |
Design, synthesis and biological characterization of novel mitochondria targeted dichloroacetate-loaded compounds with antileukemic activity | 2016 | Trapella, Claudio; Voltan, Rebecca; Melloni, Elisabetta; Tisato, Veronica; Celeghini, C; Bianco, ...Sara; Fantinati, Anna; Salvadori, Severo; Guerrini, Remo; Secchiero, Paola; Zauli, Giorgio | |
Synthetic cannabinoid JWH-018 and its halogenated derivatives JWH-018-Cl and JWH-018-Br impair Novel Object Recognition in mice: Behavioral, electrophysiological and neurochemical evidence | 2016 | Barbieri, Mario; Ossato, Andrea; Canazza, Isabella; Trapella, Claudio; Borelli, Andrea Celeste; B...eggiato, Sarah; Rimondo, C; Serpelloni, G; Ferraro, Luca Nicola; Marti, Matteo | |
Effect of the novel synthetic cannabinoids AKB48 and 5F-AKB48 on “tetrad”, sensorimotor, neurological and neurochemical responses in mice. In vitro and in vivo pharmacological studies | 2016 | Canazza, Isabella; Ossato, Andrea; Trapella, Claudio; Fantinati, Anna; de Luca, Maria Antonietta;... Margiani, Giulia; Vincenzi, Fabrizio; Rimondo, Claudia; Di Rosa, Fabiana; Gregori, Adolfo; Varani, Katia; Borea, Pier Andrea; Serpelloni, Giovanni; Marti, Matteo | |
Effect of JWH-250, JWH-073 and their interaction on “tetrad”, sensorimotor, neurological and neurochemical responses in mice | 2016 | Ossato, Andrea; Canazza, Isabella; Trapella, Claudio; Vincenzi, Fabrizio; De Luca, Maria Antoniet...ta; Rimondo, Claudia; Varani, Katia; Borea, Pier Andrea; Serpelloni, Giovanni; Marti, Matteo | |
Structure-and conformation-Activity studies of nociceptin/orphanin FQ receptor dimeric ligands | 2017 | Pacifico, Salvatore; Carotenuto, Alfonso; Brancaccio, Diego; Novellino, Ettore; Marzola, Erika; F...errari, Federica; Cerlesi, Maria Camilla; Trapella, Claudio; Preti, Delia; Salvadori, Severo; Calo', Girolamo; Guerrini, Remo | |
1‐cyclohexyl‐x‐methoxybenzene derivatives, novel psychoactive substances seized on the internet market. Synthesis and in vivo pharmacological studies in mice | 2017 | Fantinati, Anna; Ossato, Andrea; Bianco, Sara; Canazza, Isabella; De Giorgio, F; Trapella, Claudi...o; Marti, Matteo | |
Antinociceptive action of NOP and opioid receptor agonists in the mouse orofacial formalin test | 2017 | Rizzi, Anna; Ruzza, Chiara; Bianco, Sara; Trapella, Claudio; Calo', Girolamo | file con accesso da definire |
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism | 2017 | Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, M...aria Camilla; Trapella, Claudio; Calo', Girolamo | |
Expeditious Synthesis and Biological Characterization of Enantio-Enriched (-)-Nutlin-3 | 2017 | Fantinati, Anna; Bianco, Sara; Cristofori, Virginia; Cavazzini, Alberto; Catani, Martina; Zanirat...o, Vinicio; Pacifico, Salvatore; Rimondi, Erika; Milani, Daniela; Voltan, Rebecca; Secchiero, Paola; Trapella, Claudio |
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